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3-(4-fluorophenoxy)-1-(furan-3-carbonyl)azetidine
N,N,4-trimethyl-5-{4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine-1-carbonyl}pyrimidin-2-amine
6-cyclopentyl-N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
7-[(3-methylphenyl)methyl]-2-(6-methylpyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
ethyl 1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-4-(2-phenoxyethyl)piperidine-4-carboxylate
3-(ethanesulfinyl)-N-ethyl-N-{[4-(propan-2-yl)phenyl]methyl}propanamide
N-[(3S,7S,8aS)-3-(4-aminobutyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-methoxybenzamide
2-{4-[2-(benzylsulfanyl)-4-hydroxypyrimidine-5-carbonyl]morpholin-3-yl}acetamide
2-{3-[(2,3-dimethylquinoxalin-6-yl)formamido]propanamido}acetic acid
(2R,6R)-4-{2-[(propan-2-yl)amino]pyrimidine-5-carbonyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-[(3,5-dimethylphenyl)methyl]-4-(2-propoxypropanoyl)piperazin-2-one
N-ethyl-N-(1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-yl)acetamide
1,2-dimethyl-4-{6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carbonyl}piperazine
N-(prop-2-en-1-yl)-N-(pyridin-2-ylmethyl)-2-(pyrrolidin-1-yl)benzamide
N-[1-(3-cyanopyridin-2-yl)piperidin-4-yl]-2-(dimethylamino)-2-(4-methylphenyl)acetamide
1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N-cyclopropyl-3-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}oxy)-4-methoxybenzamide
5-[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]-N-(pyridin-3-ylmethyl)pyridin-2-amine
(1S,5R)-6-(cyclobutylmethyl)-3-[(6-methylpyridin-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
4-(dimethyl-1,3-thiazole-5-carbonyl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
(3aS,6aS)-2-[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(4-methyl-1,3-thiazol-2-yl)-4-(pyridin-4-yl)benzamide
4-(3-{3-[3-(pyridin-3-yl)phenyl]-1H-pyrazol-1-yl}propyl)morpholine
2-({[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl](methyl)amino}methyl)-3H,4H-thieno[3,2-d]pyrimidin-4-one
2-oxo-1-phenyl-N-[2-(1,3-thiazol-2-yl)ethyl]pyrrolidine-3-carboxamide
2-(2,2-dimethylpropanamido)-N-methyl-N-(oxan-4-yl)benzamide
2-(2-phenylethyl)-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-1,3-benzoxazole-5-carboxamide
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}cyclopropanamine
N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
2-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,6-dimethylpyrimidin-4-amine
1-(1-benzylpiperidin-4-yl)-4-(4-propyl-1H-1,2,3-triazol-1-yl)piperidine
5-{[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-N-methylfuran-2-carboxamide
4-ethyl-N-methyl-N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-1,2,3-thiadiazole-5-carboxamide
2-(cyclopentylmethyl)-6-methyl-1-[3-(2-oxopyrrolidin-1-yl)propyl]-3-(piperidine-1-carbonyl)-1,4-dihydropyridin-4-one
N-[(5-ethylpyridin-2-yl)methyl]-2-[(2-fluorophenyl)methyl]-1,3-benzoxazole-6-carboxamide
2-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pyrimidine
1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(4H-1,2,4-triazol-4-yl)piperidine
2-methyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
ethyl 1-[(2-aminopyrimidin-5-yl)methyl]-4-[(3-methoxyphenyl)methyl]piperidine-4-carboxylate
4-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-1,3-oxazolidin-2-one
N-[2-(pyridin-4-yl)ethyl]-6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
5-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)-2-(pyrrolidin-1-yl)benzonitrile
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)pyrimidin-2-amine
5-[4-(4-methoxyphenyl)-3,3-dimethylpiperazine-1-carbonyl]-2-methyl-3,4-dihydropyrimidin-4-one
N-[(2R,3R)-2-methoxy-1'-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
1-[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
4-(1,1-dioxo-1λ6-thiolan-3-yl)-N-(1-methyl-1H-indazol-6-yl)piperazine-1-carboxamide
3-(4-methyl-1,3-thiazol-5-yl)-1-[3-(pyridin-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]propan-1-one
methyl 2-[7-methyl-2-oxo-3-(piperidin-1-ylmethyl)-1,2-dihydroquinolin-1-yl]acetate
[1-(6-aminopyrimidin-4-yl)-3-(3-phenylpropyl)piperidin-3-yl]methanol