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2-(furan-2-yl)-5-({2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}methyl)pyrimidine
1-(1-{5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carbonyl}piperidin-4-yl)pyrrolidin-2-one
N-[4-methyl-3-(3-methylbenzamido)phenyl]-1H-indole-3-carboxamide
3-ethyl-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]-1,2-oxazole-5-carboxamide
3-[2-(dimethylamino)-N-methyl-2-(3-methylphenyl)acetamido]-N-methylpropanamide
1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-3-(1-methyl-1H-pyrazol-5-yl)propan-1-one
1-methyl-4-[4-(1H-1,2,4-triazol-3-yl)benzoyl]piperazine-2-carboxylic acid
N-[(4-ethoxyphenyl)methyl]-N-(quinolin-2-ylmethyl)cyclopropanamine
(2S,4R)-4-amino-N-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidine-2-carboxamide
4-{5-[(4-hydroxypiperidin-1-yl)methyl]-1,2-oxazole-3-carbonyl}-1λ6-thiomorpholine-1,1-dione
4-{4-phenyl-1-[2-(1H-1,2,3,4-tetrazol-5-yl)ethyl]-1H-imidazol-5-yl}-1-(propan-2-yl)piperidine
(2R,6R)-4-(1H-imidazol-4-ylmethyl)-10-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
3-(2-{[(3,4-difluorophenyl)methyl]carbamoyl}ethyl)-N-(4-methoxyphenyl)piperidine-1-carboxamide
3-{5-[(6-chloropyridin-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
(1S,2R)-N2-tert-butyl-N1-cyclopropyl-N1-[(1-methyl-1H-imidazol-2-yl)methyl]cyclohexane-1,2-dicarboxamide
1-oxo-2-[2-(pyridin-4-yl)ethyl]-N-(1,3-thiazol-2-ylmethyl)-2,3-dihydro-1H-isoindole-5-carboxamide
1-[5-(1H-imidazol-2-yl)imidazo[2,1-b][1,3]thiazole-6-carbonyl]piperidine
1-[3-(1H-imidazol-5-yl)phenyl]-3-[2-(pyrrolidin-1-yl)ethyl]urea
N-(1-cycloheptylpiperidin-3-yl)-2-(trifluoromethyl)benzamide
N-(1-hydroxybutan-2-yl)-N-(pyridin-4-ylmethyl)-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
4-{2-oxo-2-[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]ethyl}-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
N-cyclopropyl-1-[1-(6-cyclopropylpyrimidin-4-yl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
1-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-4-phenylbutane-1,4-dione
1-[(4,8-dimethoxynaphthalen-1-yl)methyl]-4-fluoropiperidine
(3R,4R)-1-(3-chloro-4-fluorobenzenesulfonyl)-3,4-dimethylpyrrolidin-3-ol
4-(2-{[5-(methanesulfonylmethyl)pyridin-2-yl]oxy}hex-5-en-1-yl)morpholine
(4aR,7aS)-1-cyclobutanecarbonyl-4-(quinolin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(2-methoxyphenyl)-3-{1-[1-(2,2,3,3-tetramethylcyclopropanecarbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
N-ethyl-2-[2-(2-methoxyethyl)morpholin-4-yl]pyrimidin-4-amine
2-(2-methoxy-4-{[4-(pyridin-4-yl)piperazin-1-yl]methyl}phenoxy)propanoic acid
1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-4-(pyrrolidine-1-sulfonyl)piperazine
1-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-ol
4-(1-{1-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-imidazol-2-yl)quinoline
1-(4-methyl-1H-pyrrole-2-carbonyl)-3-(3-methylphenoxymethyl)piperidine
3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[3-(methylsulfanyl)propyl]benzamide
(2R,6R)-4-(5-fluoro-2-methylbenzoyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
2-[4-(thiophene-3-carbonyl)morpholin-2-yl]ethan-1-ol
N-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)oxane-2-carboxamide
8-[2-(2-methoxyethoxy)acetyl]-2-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
2-[6-oxo-1-(pentan-3-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl]benzonitrile
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-2-methylfuran-3-carboxamide
1-[1-(pyrimidin-2-yl)piperidin-3-yl]-3-(1,2,3-thiadiazol-5-yl)urea
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-[6-oxo-4-(piperidin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
(1S,5R)-3-(3,5-dimethyl-1H-indole-2-carbonyl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
8-[3-amino-3-(3,4-dimethoxyphenyl)propanoyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
6-ethyl-4-{2-[2-(thiophen-2-yl)ethyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
1-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-1,2,4-triazole
1-{[2,5-dimethoxy-4-(methylsulfanyl)phenyl]methyl}-3-phenylpyrrolidin-3-ol
{2-[(E)-2-phenylethenyl]phenyl}methanamine
3-butyl-4-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}-1-methylpiperazin-2-one