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N-{1-[(methylcarbamoyl)methyl]-1H-pyrazol-4-yl}-4-[(3-methylpiperidin-1-yl)methyl]benzamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}benzamide
N-[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
5-[3-(pyridin-2-yl)azetidine-1-carbonyl]-2-(pyridin-3-yl)pyrimidine
2-(4-{[2-(difluoromethoxy)phenyl]methyl}-1-[(3-methoxyphenyl)methyl]piperazin-2-yl)ethan-1-ol
8-chloro-2-({2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidin-1-yl}methyl)quinoline
(4aS,8aR)-6-(2H-1,3-benzodioxole-5-carbonyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
5-({[(3-{2-[4-(3-chlorobenzoyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)amino}methyl)pyrrolidin-2-one
methyl 4-[3-(5-cyano-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl)propanamido]benzoate
3-[3-(dimethylamino)-2,2-dimethylpropyl]-1-(4-ethenylphenyl)urea
5-[(4-methylpiperazin-1-yl)methyl]-N-(pyridin-3-ylmethyl)furan-2-carboxamide
(2S,4S)-4-amino-N-[3-(1,3-benzothiazol-2-yl)propyl]-1-methylpyrrolidine-2-carboxamide
1-methyl-4-[5-(trifluoromethyl)pyridin-2-yl]-1,4,9-triazaspiro[5.6]dodecan-10-one
(2S,4R)-N-(3-chloro-4-propoxyphenyl)-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidine-1-carboxamide
N-(propan-2-yl)-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
9-(5-ethyl-2,6-dimethylpyrimidin-4-yl)-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-{methyl[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amino}-N-(pyridin-3-yl)propanamide
N-cyclopentyl-2-fluoro-N-{[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl}benzene-1-sulfonamide
(4aR,6R,8aS)-8a-(methoxymethyl)-2-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-6-(morpholin-4-yl)-decahydroisoquinoline
1-amino-N-(2-{1-[(4,5-dimethylfuran-2-yl)methyl]piperidin-3-yl}ethyl)cyclopropane-1-carboxamide
1-[4-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-(pyrimidin-2-ylsulfanyl)ethan-1-one
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)furan-2-carboxamide
2-(2,4-dioxoimidazolidin-1-yl)-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]acetamide
[(3R,4R)-1-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methyl-1,3-thiazole-5-carboxamide
1-(cyclohexylmethyl)-5-{3-[(4-methylpiperazin-1-yl)methyl]-1,2,4-oxadiazol-5-yl}piperidin-2-one
5-fluoro-2-methyl-3-(2-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}ethyl)-1H-indole
(1R,5S,6R)-3-{[6-(dimethylamino)pyridin-3-yl]methyl}-3-azabicyclo[3.1.0]hexane-6-carboxylic acid
1-[(6-chloropyridin-3-yl)methyl]-2-methyl-4-phenylpiperazine
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidin-4-amine
5-[1-(6-cyanopyridine-3-carbonyl)pyrrolidin-2-yl]-N-cyclopropylthiophene-2-carboxamide
(4-{[4-phenyl-5-(pyridin-4-yl)-1H-imidazol-1-yl]methyl}phenyl)methanol
[(3R,4R)-1-(2-chloro-4-fluorobenzoyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
methyl 3-(cyclobutylmethoxy)-5-{[1-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]carbamoyl}benzoate
3-[1-(2,2-dimethyl-4-oxo-3,4-dihydro-2H-pyran-6-carbonyl)piperidin-3-yl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
(4-{[methyl(oxolan-3-ylmethyl)amino]methyl}oxan-4-yl)methanol
N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-amino-6-(2,2-dimethyloxan-4-yl)-5-ethyl-4-(2-methoxypyrimidin-5-yl)pyridine-3-carbonitrile
N5,N5,N6-trimethyl-N6-[(3-methyl-1,2-oxazol-5-yl)methyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
1-{4-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidine-1-carbonyl]phenyl}ethan-1-one
(3S,9aR)-8-[(3,4-dimethylphenyl)methyl]-2,3-dimethyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-(3-methyl-1H-pyrazole-4-carbonyl)-7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-6-one
2-[(5-methylpyrazin-2-yl)methyl]-9-(6-methylpyrimidin-4-yl)-2,9-diazaspiro[5.5]undecan-3-one
1-[5-(3,4-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]-2-(methoxymethyl)piperidine
N-(2-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}ethyl)-2-(trifluoromethyl)benzamide
2,3-dimethyl-N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}quinoxaline-6-carboxamide
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
2-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-6-methylpyridine-3-carboxylic acid
1-(1-benzylpiperidin-4-yl)-1,4-diazepane-6-carboxylic acid