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N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1-phenyl-1H-1,2,3-triazole-4-carboxamide
4-{1-azabicyclo[2.2.2]octan-3-yl}-N-(2-fluoro-4-methoxyphenyl)piperazine-1-carboxamide
(3R,5S)-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
methyl 3-({[2-(azocan-1-yl)pyridin-3-yl]methyl}carbamoyl)propanoate
methyl 5-(2,5-dimethylbenzoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
(2S,4R)-4-amino-1-(2-amino-4-phenylpyrimidine-5-carbonyl)-N,N-diethylpyrrolidine-2-carboxamide
2-[benzyl(methyl)amino]-N-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-indene-2-carboxamide
3-[4-({methyl[(5-methyl-1,2-oxazol-3-yl)methyl]amino}methyl)phenyl]prop-2-yn-1-ol
(3S,9aR)-3-methyl-8-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-(6-methoxynaphthalen-2-yl)-N,N-dimethylmorpholine-4-carboxamide
4-[3-(1,4-diazepane-1-sulfonyl)benzoyl]-1-methylpiperazin-2-one
5-methyl-4-{methyl[2-(4-methylphenoxy)ethyl]amino}-N-(oxolan-2-ylmethyl)thieno[2,3-d]pyrimidine-6-carboxamide
6-{1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}pyrimidin-4-ol
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
7-(cyclobutylmethyl)-2-[2-(cyclohex-1-en-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
8-[3-(3-methoxyphenoxy)propyl]-2-(propan-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
2-(2-methoxy-5-methylphenyl)-5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridine
7-(5-methoxy-4-oxo-1,4-dihydropyridine-2-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-[(E)-2-(furan-2-yl)ethenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-ethyl-4-{[3-(2-methylpiperidine-1-carbonyl)-1,2-oxazol-5-yl]methyl}piperazine
4-{2-[5-(1-ethyl-1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}pyridine
2-methoxy-N-({5-[4-methyl-6-(methylamino)pyrimidin-2-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide
4-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane-4-carbonyl]-1,2-dihydrophthalazin-1-one
1-{[1-(4-propylpyrimidine-5-carbonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxylic acid
6-(1-methyl-1H-imidazol-2-yl)-N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}pyridazin-3-amine
2-(4-fluorophenyl)-1-[7-(5-methylthiophen-2-yl)-9-(oxan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
2-(4-fluorophenyl)-N-(furan-3-ylmethyl)imidazo[1,2-a]pyridine-6-carboxamide
1-({5-[(4-methoxy-3-methylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,3-dimethylurea
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-(2-methylquinolin-4-yl)piperidin-3-yl]propanoic acid
3-ethyl-N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1H-pyrazole-4-carboxamide
2-(dimethylamino)-2-(2-methylphenyl)-1-[4-(pyridin-4-yl)piperazin-1-yl]ethan-1-one
1-[3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]-2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethan-1-one
N-[3-(2-methoxyphenyl)propyl]-4-(pyridin-2-yl)pyrimidin-2-amine
3-(4-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}phenyl)propanoic acid
1-(carbamoylmethyl)-N-[2-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
(3-{[1-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)pyrrolidin-3-yl]methyl}phenyl)methanol
4-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidine-1-carbonyl]-2-methoxyphenol
N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-3-{[(2S)-oxolan-2-ylmethyl]sulfamoyl}benzamide
N-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}thiolan-3-amine
(3aS,6aR)-5-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-(carbamoylmethyl)-N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}piperidine-3-carboxamide
1-{[3-cyclopropyl-1-(3-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-4-methyl-1,2-dihydroquinolin-2-one
5-[7-(3,6-dimethylpyrazin-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]-1,2-dihydropyridin-2-one
8-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decane
2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]acetamide
1-(5-ethyl-1,3-oxazole-4-carbonyl)-3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
(2R,3R)-3-{[(3-phenyl-1H-pyrazol-5-yl)methyl]amino}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
3-{1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole
N-[2-(dimethylamino)-2-(furan-2-yl)ethyl]-5-methoxy-4-oxo-1,4-dihydropyridine-2-carboxamide
1-(cyclopropylmethyl)-5-{1H-pyrazolo[1,5-a]imidazole-7-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid