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N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-(3-methylphenyl)acetamide
ethyl 4-[4-(pyridin-3-yl)pyrimidin-2-yl]piperazine-1-carboxylate
(5-{[2-(2-methoxyethyl)piperidin-1-yl]methyl}furan-2-yl)methanol
4-(3-fluorophenoxy)-1-[(5-methylfuran-2-yl)methyl]piperidine-4-carboxylic acid
4-[2-(8-chloroquinolin-2-yl)-1H-imidazol-1-yl]-N-ethylpiperidine-1-carboxamide
methyl 3-[1-(4-chlorophenyl)cyclopropaneamido]-5-{[(2-methyl-1,3-thiazol-4-yl)formamido]methyl}benzoate
2,6,8-trimethyl-4-[2-(1-methyl-1H-pyrazol-3-yl)piperidine-1-carbonyl]quinoline
3-methyl-N-[2-(3-phenylpropoxy)phenyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
1-cyclobutanecarbonyl-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)piperidine-4-carboxamide
1-[({1-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}carbamoyl)methyl]piperidine-4-carboxamide
(4aS,7aR)-1-(2-hydroxypyridine-3-carbonyl)-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]{[5-(oxan-2-yl)furan-2-yl]methyl}amine
4-{[1-methyl-3-(2-methylpropyl)-1H-pyrazol-5-yl]methyl}-1,4-oxazepane
N-[(3R,4S)-4-cyclopropyl-1-methanesulfonylpyrrolidin-3-yl]-5-methoxyfuran-2-carboxamide
1-(2,5-dimethylphenyl)-5-(2-methoxyethyl)-3-methyl-1H-1,2,4-triazole
N-(1-benzyl-1H-pyrazol-5-yl)-2-(5-phenyl-2H-1,2,3,4-tetrazol-2-yl)acetamide
3-(2-chlorophenyl)-N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-(3-hydroxyphenyl)propanamide
1-[1-(adamantan-2-yl)piperidin-3-yl]-4-(2-methoxyphenyl)piperazine
1-[2-(benzyloxy)ethyl]-4-(1-methyl-1H-imidazol-2-yl)-1H-1,2,3-triazole
1-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine
1-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
2-{3-chloro-6-methylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-8-methyl-2,8-diazaspiro[4.5]decane
4-[(carbamoylmethyl)sulfamoyl]-N-[3-(methylsulfanyl)propyl]benzamide
2,6-dimethyl-8-[4-(2-methylpyrimidin-4-yl)piperidin-1-yl]octan-2-ol
(4aS,8aR)-1-(3-methoxypropyl)-6-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
N-cyclopentyl-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
5-[2-(4-methylphenoxymethyl)furan-3-carbonyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
2-[2-(2,6-dimethoxy-4-methylphenyl)-4-methylphenoxy]acetamide
5-[4-(5-chloro-2-methylphenyl)piperazine-1-carbonyl]-1-cyclopentyl-N-ethyl-4-oxo-1,4-dihydropyridine-3-carboxamide
2-[ethyl({[(3R,4R)-4-(hydroxymethyl)-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}pyrrolidin-3-yl]methyl})amino]ethan-1-ol
methyl 5-(3-chloro-4-methoxyphenyl)pyridine-3-carboxylate
1-(2-methoxyphenyl)-N-[(5-methylpyrazin-2-yl)methyl]-1H-pyrazole-4-carboxamide
{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}({3-[5-(pyrrolidin-1-yl)pyridazin-3-yl]phenyl}methyl)amine
N-{[(3S,4S)-3-hydroxy-1-[(2-methylpyrimidin-5-yl)methyl]piperidin-4-yl]methyl}-2-methylbenzamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(3-methylbut-2-en-1-yl)pyrrolidin-3-yl]-1,3,5-trimethyl-1H-pyrazole-4-carboxamide
1-cyclopropanecarbonyl-4-[(1-methyl-1H-indol-5-yl)methyl]-1,4-diazepan-6-ol
3-[1-(benzenesulfonyl)cyclopropanecarbonyl]-3,9-diazaspiro[5.5]undecane
2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]-N-[2-(pyridin-2-yl)ethyl]acetamide
1-[benzyl(methyl)amino]-3-[4-({[(2-methoxyphenyl)methyl]amino}methyl)phenoxy]propan-2-ol
1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxy-3-{[(prop-2-en-1-yl)amino]methyl}piperidin-2-one
8-{2-[4-(dimethylamino)phenyl]acetyl}-2-ethyl-2,8-diazaspiro[4.5]decan-3-one
2-{[5-(2-fluorophenyl)furan-2-yl]methyl}-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
N-methyl-1-{6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carbonyl}pyrrolidine-3-carboxamide
4-(3,5-dimethyl-1H-pyrazol-4-yl)-6-(4-methylpiperazin-1-yl)pyrimidin-2-amine
4-{[2-(dimethylamino)ethyl]amino}-5-methyl-N-(3-methylbutyl)thieno[2,3-d]pyrimidine-6-carboxamide
3-(5-methylthiophen-2-yl)-N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-1H-pyrazole-5-carboxamide
4-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)-1H-imidazol-1-yl]benzamide
(4aR,7aS)-1-{2-[2-(4H-1,2,4-triazol-4-yl)phenoxy]acetyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione