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2-butyl-8-[3-(1H-imidazol-1-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
(1S,6R)-9-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}-3-methyl-3,9-diazabicyclo[4.2.1]nonan-4-one
2-(2H-1,3-benzodioxol-5-yl)-1-[9-methoxy-7-(6-methoxypyridazin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
2-({2-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
N-{1-[2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]pyrrolidin-3-yl}acetamide
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-2-(2-methyl-1H-imidazol-1-yl)propanamide
3-{[2-(1-phenylethyl)-1H-imidazol-1-yl]methyl}pyridine
6-tert-butyl-1-methyl-N-[2-(pyridin-2-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
{2-methoxy-5-[6-(methylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]phenyl}methanol
4-[2-(4-fluoro-2-methylphenyl)acetyl]-1-(4-methylphenyl)piperazin-2-one
N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2,5-dimethylfuran-3-carboxamide
1,4-dimethyl-2-[3-(2-methylphenoxy)azetidine-1-carbonyl]-1H-indole
7-(quinoxalin-2-yl)-2,7-diazaspiro[4.4]nonane-1,3-dione
(1R,5S,8R)-N-(4-acetylphenyl)-8-(dimethylamino)-3-azabicyclo[3.2.1]octane-3-carboxamide
N-[(5-methyl-1,2-oxazol-3-yl)methyl]-2-(oxolane-2-carbonyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
1'-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-1-methyl-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
3-{2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-1-(pyrrolidin-1-yl)propan-1-one
1,3-dimethyl-N-[2-(pyrrolidin-1-yl)ethyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-(4-fluorophenyl)-2-[4-(4-methoxybenzoyl)piperazin-1-yl]acetic acid
2-cyclopentyl-4-{4-[2-(4-fluorophenyl)acetyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
N-{[1-(cyclohexylmethyl)-2-cyclopropylmethanesulfonyl-1H-imidazol-5-yl]methyl}-N-methyloxolan-3-amine
N-[2-(5,7-difluoro-2-methyl-1H-indol-3-yl)ethyl]-2-ethylpyrimidine-5-carboxamide
(3aS,6aS)-5-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{3-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidine-1-carbonyl]phenyl}pyrrolidin-2-one
2-cyclobutyl-N-[(3R,4S)-4-propyl-1-(pyrimidin-2-ylmethyl)pyrrolidin-3-yl]acetamide
(2S,4R)-4-amino-1-[1-(2-fluorophenyl)piperidin-4-yl]-N-methylpyrrolidine-2-carboxamide
1-[3-(dimethylamino)phenyl]-3-(2-propoxypropyl)urea
(2R,3R,6R)-5-[(2-butyl-1H-imidazol-4-yl)methyl]-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(3-methyl-4-{[3-(2-methylpiperidin-1-yl)azetidin-1-yl]methyl}-1H-pyrazol-1-yl)ethan-1-ol
2-[(3-methoxyphenyl)methyl]-4-(pyrazin-2-yl)morpholine
2-(2-methoxyethyl)-9-[6-(trifluoromethyl)pyridin-2-yl]-2,9-diazaspiro[5.5]undecan-3-one
2-(3-{[2-(3-methoxyphenyl)azetidin-1-yl]methyl}-2-methyl-1H-indol-1-yl)acetamide
2-amino-4-(3,5-dimethyl-1H-pyrazol-4-yl)-6-(1H-pyrrol-2-yl)pyridine-3-carbonitrile
3-(dimethyl-1,2-oxazol-4-yl)-1-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]propan-1-one
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[1-(3-methylpyridin-2-yl)propan-2-yl]-1,3-oxazole-4-carboxamide
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-3-(1-methylpiperidin-2-yl)propanamide
1-(4-chloro-1,3-dimethyl-1H-pyrazole-5-carbonyl)-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
1-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
6-methyl-N-(3-methyl-4-pentanamidophenyl)-1-(propan-2-yl)-1H-pyrazolo[3,4-b]pyridine-4-carboxamide
5-[(2S)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-2-(4-methylphenyl)pyrimidin-4-ol
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-({[(3-methylpyridin-2-yl)methyl]amino}methyl)piperidin-2-one
methyl (1S,3S,3aR,6aS)-5-methyl-3-(3-methylthiophen-2-yl)-4,6-dioxo-1-phenyl-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
2-[3-(2-methoxyethyl)-5-[2-(methylamino)pyridin-4-yl]-1H-1,2,4-triazol-1-yl]acetic acid
N-[(3S,7S,8aS)-3-ethyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-fluoro-3-(trifluoromethyl)benzamide
N-[2-(3-phenylpyrrolidin-1-yl)ethyl]oxane-4-carboxamide
4-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
5-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-4-propylpyrimidine
1-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]-3-(pyrrolidin-1-yl)propan-1-one
1-{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidine-3-carbonitrile
4-[6-(2-fluoro-5-methylphenyl)pyrimidin-4-yl]morpholine