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N-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-4-(thian-4-yl)piperazine-1-carboxamide
N-[3-({[2-(methylsulfamoyl)ethyl]carbamoyl}methoxy)phenyl]propanamide
3-[(2R,3R,6R)-5-[(6-methylpyridin-2-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
N-{1-[(5-fluoro-2-methylphenyl)carbamoyl]ethyl}-N'-[2-(propan-2-yl)phenyl]butanediamide
(2S,4R)-N-{[2-(2,3-difluoro-4-methylphenoxy)pyridin-3-yl]methyl}-4-hydroxypyrrolidine-2-carboxamide
N-{[1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
8-fluoro-N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]quinoline-2-carboxamide
2-[4-(4-aminopyridin-3-yl)-1H-pyrazol-1-yl]-N-[1-(propan-2-yl)-1H-1,2,3-triazol-4-yl]acetamide
4-[5-methyl-2-oxo-4-(3-phenylpropanoyl)piperazin-1-yl]benzonitrile
N-{2-[4-(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]-2-oxoethyl}benzamide
N-[(dimethyl-1,3-thiazol-2-yl)methyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
4-{[2-(3-methoxyphenyl)piperidin-1-yl]methyl}-2-(propan-2-yl)pyrimidine
2-methoxy-5-(2-phenoxyethyl)benzamide
N-methyl-N-[2-(1,2,4-oxadiazol-3-yl)ethyl]-2-oxo-2-(pyridin-3-yl)acetamide
1-(2-cyclohexylethyl)-3-hydroxy-3-({[(2-hydroxypyridin-3-yl)methyl]amino}methyl)piperidin-2-one
4-(4-chlorophenyl)-N-{2-[(2S)-pyrrolidin-2-yl]ethyl}butanamide
2-[3-(pyridin-4-yl)-5-{2H,3H-thieno[3,4-b][1,4]dioxin-5-yl}-1H-1,2,4-triazol-1-yl]acetic acid
N-(pyridin-2-ylmethyl)-1-[1-(thiophen-2-ylmethyl)piperidin-4-yl]piperidine-4-carboxamide
3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-1-[3-(1H-imidazol-2-yl)piperidin-1-yl]propan-1-one
4-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazin-2-one
N-(3-{[(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethyl)carbamoyl]methoxy}phenyl)propanamide
2-(2-chloro-4-fluorophenoxymethyl)-N-methyl-N-(oxan-2-ylmethyl)-1,3-oxazole-4-carboxamide
4-(1,3-benzothiazole-6-carbonyl)-5-methyl-1-(4-methylphenyl)piperazin-2-one
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
2-{3-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidine-1-carbonyl]phenoxy}acetamide
3-{1-[5-(2-chloro-4-methoxyphenoxymethyl)-1,2-oxazole-3-carbonyl]pyrrolidin-2-yl}-4-methyl-1,2,5-oxadiazole
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-benzyl-4-{[(2,4-difluorophenyl)methyl]amino}pyrrolidine-2-carboxamide
3-[(cyclopropylamino)methyl]-1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxypiperidin-2-one
N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-2-(trimethyl-1H-pyrazol-1-yl)acetamide
2-({6-[3-(4-chlorobenzoyl)piperidin-1-yl]pyrimidin-4-yl}amino)ethan-1-ol
(3S,4R)-4-phenyl-1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]pyrrolidine-3-carboxylic acid
(2R)-2-amino-3-methoxy-1-[4-(4-methylphenoxy)piperidin-1-yl]propan-1-one
3-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1H-indazole
[(3R,4R)-4-(piperidin-1-ylmethyl)-1-[3-(pyridin-4-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-yl]methanol
2-{4-[1-(4-chloro-1H-pyrazole-3-carbonyl)pyrrolidin-3-yl]piperidin-1-yl}pyrimidine
1-{[4-(benzyloxy)-2-methoxyphenyl]methyl}azepan-4-ol
(2R,6R)-10-methoxy-4-(5-methylthiophene-2-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
3-(2-methoxy-5-phenylphenyl)-1-methyl-1-[2-(oxan-2-yl)ethyl]urea
N,6-dimethyl-2-{4-[4-(piperidin-1-ylmethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}pyrimidin-4-amine
1-{2-[2-(ethylamino)pyrimidin-5-yl]-6-fluoroquinoline-4-carbonyl}piperidine-3-carbonitrile
N-[2-(5-cyclobutyl-1,2,4-oxadiazol-3-yl)ethyl]-1H-indazole-3-carboxamide
2-{[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}-5-methoxypyridin-4-ol
3-{3-[3-(dimethylamino)pyrrolidin-1-yl]propyl}-8-(1-methyl-1H-pyrazole-5-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
7-{3-[(3-fluorophenyl)amino]piperidine-1-carbonyl}quinolin-8-ol
methyl 5-{2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-5-oxopentanoate
1-[2-(dimethylamino)ethyl]-4-[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]pyrrolidin-2-one
3,5-dimethyl-N-(5-oxo-1-phenylpyrrolidin-3-yl)-1,2-oxazole-4-sulfonamide
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-{[methyl(3-methylbutyl)amino]methyl}piperidin-2-one
6-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-5,6-dihydro-1,6-naphthyridin-5-one
(2E)-N-[(5-{[2-(dimethylamino)ethyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]-3-(thiophen-2-yl)prop-2-enamide