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2-[(1H-indol-3-ylmethyl)({[4-(methylsulfanyl)phenyl]methyl})amino]ethan-1-ol
3-[(4-{4-[hydroxy(1-methyl-1H-imidazol-2-yl)methyl]piperidin-1-yl}-6-methylpyrimidin-2-yl)amino]phenol
[(2-ethoxynaphthalen-1-yl)methyl](methyl)[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amine
N-{1-[3-methyl-1-(4-methylpyridin-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}-N-phenylmethanesulfonamide
N-{[7-(5-acetyl-2-fluorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-methyl-1,2,3-thiadiazole-5-carboxamide
4-[2-(4-methoxyphenyl)ethyl]-3-(1-methylpiperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-6-methyl-2-(pyridin-3-yl)pyrimidin-4-amine
3-(benzyloxy)-1-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidine
6-methyl-3-(3-methylpiperidine-1-carbonyl)-2-(2-phenylethyl)-1-(pyridin-4-ylmethyl)-1,4-dihydropyridin-4-one
7-cyclohexyl-2-[(3-hydroxy-4-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
4-[1-(4-chlorophenyl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]-1λ6-thiane-1,1-dione
2,2-dimethyl-N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)-4-oxo-3,4-dihydro-2H-pyran-6-carboxamide
1'-(3,5-dimethyl-1H-indole-2-carbonyl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
1-[(2,6-difluorophenyl)methyl]-N-{[1-(hydroxymethyl)cyclopentyl]methyl}-N-methyl-1H-1,2,3-triazole-4-carboxamide
2-({2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}amino)acetamide
1-cyclobutanecarbonyl-N-[(4,6-dimethylpyrimidin-2-yl)methyl]piperidine-4-carboxamide
6-{[methyl(thiophen-3-ylmethyl)amino]methyl}-N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
4-[3-(benzyloxy)propyl]-1-(4-methylphenyl)piperazin-2-one
2-[2-methyl-4-(pyrrolidin-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]-1,3-thiazole-4-carboxamide
5-fluoro-2-{[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-3-methyl-1H-indole
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-2-propyl-1,3-thiazole-4-carboxamide
1-(5-chloro-2-methylphenyl)-4-[4-(1H-pyrazol-3-yl)benzoyl]piperazine
N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2,3-dihydro-1-benzofuran-2-carboxamide
N-[(3R,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-phenyl-5-propyl-1H-pyrazole-4-carboxamide
3-{[3-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl}pyridin-2-amine
N-[(3R,4S)-4-cyclopropyl-1-(6-cyclopropylpyrimidin-4-yl)pyrrolidin-3-yl]cyclobutanecarboxamide
4-[6-amino-2-(butylsulfanyl)pyrimidin-4-yl]piperazin-2-one
8-[2-(3-chlorophenyl)acetyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
4-{1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-1H-pyrazole-4-carbonyl}thiomorpholine
methyl (2S,4R)-4-hydroxy-1-{[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}pyrrolidine-2-carboxylate
N-[(2-chloro-6-fluorophenyl)methyl]-6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-ethyl-N-(2-methoxyethyl)-6-(piperidin-4-yl)pyrimidin-4-amine
2-ethyl-N-[(3R,4S)-1-methanesulfonyl-4-propylpyrrolidin-3-yl]-4-methyl-1,3-oxazole-5-carboxamide
6-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pyrimidin-4-amine
1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-4-phenylbutan-1-one
N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-(2-cyclopropylacetyl)pyrrolidine-2-carboxamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-5-methyl-4-{[3-(2-oxopyrrolidin-1-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
5-[4-(2-methylphenyl)-1,4-diazepane-1-carbonyl]isoquinoline
5-methoxy-2-{[({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}phenol
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(4-oxo-3,4-dihydrophthalazin-1-yl)propanamide
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-4-methylpyridine-3-carboxamide
N-[2-(2-methoxyphenoxy)ethyl]-N-methyl-2-[(prop-2-en-1-yl)amino]benzamide
(1-methoxypropan-2-yl)[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]amine
1-(5-cyanopyridin-2-yl)-4-(quinolin-6-yloxy)piperidine-4-carboxylic acid
2,4-dimethyl-5-{4-[3-(trifluoromethyl)phenoxy]piperidine-1-carbonyl}pyrimidine
3-{1-[3-(3-hydroxy-3-methylbut-1-yn-1-yl)benzoyl]piperidin-3-yl}-1-(morpholin-4-yl)propan-1-one
2-[1-(3-methylpyridin-4-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]-5-(1H-1,2,3,4-tetrazol-1-yl)phenol
N-(1-{1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-methylbutanamide
5-{2-oxo-2-[3-oxo-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-9-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-ethyl-3-{[({1-[ethyl(methyl)amino]cyclopentyl}methyl)carbamoyl]amino}-2-methylbenzamide