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4-[5-(isoquinolin-5-yl)-4-phenyl-1H-imidazol-1-yl]butan-1-amine
8-(2,6-dimethoxypyrimidine-4-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
2-methoxyethyl 2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecane-9-carboxylate
2-[({4-[(dimethylamino)methyl]phenyl}methyl)(methyl)amino]-2-(2-methoxy-5-methylphenyl)acetic acid
1,3-dimethyl-2,6-dioxo-N-{[2-(trifluoromethoxy)phenyl]methyl}-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-{[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]amino}pyridine-3-carboxamide
2-cyclopentyl-N-(2-methoxyethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-(2,3-dihydro-1-benzofuran-2-carbonyl)-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
N-(1-{2-[cyclohexyl(methyl)amino]-4-methylpyrimidin-5-yl}ethyl)-6-oxo-1,6-dihydropyridine-3-carboxamide
(1S,6R)-3-[4-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-3,9-diazabicyclo[4.2.1]nonane
1-[(2-fluorophenyl)methyl]-6-oxo-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}piperidine-3-carboxamide
4-[3-(4-fluorophenyl)pyrrolidine-1-carbonyl]-3-(3-methoxyphenyl)-1H-pyrazole
4-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
(5S,9aS,9bS)-5-(5-acetylthiophen-3-yl)-2-(2,3-dihydro-1H-inden-2-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-(1-{1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-4-yl}ethyl)morpholine
8-[4-(4-fluorophenyl)butanoyl]-2,8-diazaspiro[4.5]decan-3-one
2-{1-[(2-ethoxyphenyl)methyl]-4-(propan-2-yl)piperazin-2-yl}ethan-1-ol
4-{[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]amino}-5-methyl-N-(1,3-thiazol-2-ylmethyl)thieno[2,3-d]pyrimidine-6-carboxamide
5-(propan-2-yl)-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
(4aR,8aS)-1-(2,2-diphenylethyl)-6-[(2-methoxyphenyl)methyl]-decahydro-1,6-naphthyridin-2-one
4-phenyl-5-[3-(phenylamino)piperidine-1-carbonyl]pyrimidin-2-amine
3-[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]-1-[3-(2-methylpyrimidin-4-yl)phenyl]urea
2-(4-acetylphenoxy)-1-{3-[(4-methoxyphenyl)amino]piperidin-1-yl}ethan-1-one
1-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(trimethyl-1H-pyrazol-1-yl)propan-1-one
3-[(3R,4S)-1-(2-ethoxybenzoyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
2-[5-(4-methoxyphenyl)furan-2-yl]-1-(oxolan-3-ylmethyl)-1H-imidazole
4-[(2,3-dihydro-1-benzofuran-5-ylmethyl)amino]-1-[2-(4-fluorophenyl)ethyl]pyrrolidin-2-one
ethyl 4-[2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamido]piperidine-1-carboxylate
2-methyl-6-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-2,3-dihydropyridazin-3-one
2-[(2,6-dichlorophenyl)methyl]-N-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-hydroxypyrimidine-5-carboxamide
[4-({4-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)-1-methylpiperazin-2-yl]methanol
4-[(1S,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]benzonitrile
3-{2-[bis(propan-2-yl)carbamoyl]phenyl}-1H-1,2,4-triazole-5-carboxamide
1,3-dimethyl-N-[1-(morpholin-4-yl)propan-2-yl]-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
1-{3-[({6-[(propan-2-yl)amino]pyrimidin-4-yl}amino)methyl]pyridin-2-yl}piperidin-3-ol
3-(2H-1,3-benzodioxol-5-yl)-3-phenyl-N-[2-(pyrrolidin-1-yl)ethyl]propanamide
4,5-dimethyl-6-{1H-pyrrolo[2,3-b]pyridin-4-yl}-2-(trifluoromethyl)pyrimidine
(1S,5R)-6-(3-fluoropyridine-4-carbonyl)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
7-(3,6-dimethylpyrazin-2-yl)-4-[3-(1H-imidazol-1-yl)propyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(2-phenoxyethyl)-4-(3-propyl-1H-pyrazole-4-carbonyl)piperazine
2-(pyridin-3-yl)-1-{4-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]piperazin-1-yl}ethan-1-one
[7-(2,5-dimethylpyrimidin-4-yl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methanamine
1-[2-chloro-5-(trifluoromethyl)benzoyl]-4-(4H-1,2,4-triazol-3-yl)piperidine
3-methyl-5-[4-phenyl-1-(pyridin-2-ylmethyl)-1H-imidazol-5-yl]-1,2-benzoxazole
(2R,6R)-10-methoxy-4-[(3-methylphenyl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-4-(pyridin-2-ylmethyl)piperazine
1-[3-(3-methoxypropyl)piperidin-1-yl]-2-(thiophen-3-yl)ethan-1-one
N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-3-propanamidobenzamide
4-(4-{[3-(2-hydroxyethyl)-4-[1-(propan-2-yl)piperidin-4-yl]piperazin-1-yl]methyl}phenyl)but-3-yn-1-ol
methyl (1R,3S,3aR,6aS)-1,5-dimethyl-4,6-dioxo-3-[3-(1H-pyrazol-1-ylmethyl)phenyl]-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate