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2-[1-(propan-2-yl)piperidin-4-yl]-N-[1-(1-propyl-1H-1,2,4-triazol-5-yl)ethyl]acetamide
N-({1-[(3,4-dimethylphenyl)methyl]piperidin-3-yl}methyl)-2,2-dimethylpropanamide
8-(1,3-benzothiazole-6-carbonyl)-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
[(3R,4R)-4-[(dimethylamino)methyl]-1-[1-(4-methylphenyl)piperidin-4-yl]pyrrolidin-3-yl]methanol
ethyl 2-(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidin-1-yl)acetate
5-ethyl-N4-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]pyrimidine-2,4-diamine
4-[1-(furan-2-ylmethyl)piperidin-4-yl]-2-[(4-methoxyphenyl)methyl]morpholine
(2S,4R)-N-ethyl-4-(5-ethylthiophene-3-amido)-1-(1H-imidazol-4-ylmethyl)pyrrolidine-2-carboxamide
2-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-4-(pyrimidin-4-yl)morpholine
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-3-(1-methylpiperidin-3-yl)propanamide
2-{[(3-ethoxyphenyl)methyl]({2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl})amino}ethan-1-ol
2-(3-ethyl-1,2,4-oxadiazol-5-yl)-5-methoxy-1-methyl-1H-indole
N-[(3R,4R)-1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-3-hydroxypiperidin-4-yl]pyridine-3-carboxamide
4-(2-methoxyethoxy)-1-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperidine
methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]{[7-methyl-2-(morpholin-4-yl)quinolin-3-yl]methyl}amine
2-{4-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]piperazin-1-yl}-1,3-benzothiazole
1-(4-{[4-(5-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}phenyl)ethan-1-one
2-(1-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidine-3-carbonyl)pyridine
1-(2,6-dimethylpyridin-4-yl)-4-(3-methoxy-5-methylthiophene-2-carbonyl)piperazine
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-[4-(1H-pyrazol-1-yl)butan-2-yl]piperidine
2-{ethyl[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]amino}-2-(2-methoxy-5-methylphenyl)acetic acid
2-{[methyl({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amino]methyl}quinolin-4-ol
(1R,3S)-3-methoxy-7-[3-methyl-5-(phenoxymethyl)furan-2-carbonyl]-7-azaspiro[3.5]nonan-1-ol
N-{[1-(2-fluorophenyl)pyrrolidin-3-yl]methyl}imidazo[1,2-a]pyridine-6-carboxamide
N-(3,4-dimethoxyphenyl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidin-3-amine
1-{[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-2-(4-fluorophenyl)piperidine
4-(1,3-benzothiazol-2-yl)-2-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}phenol
methyl({[1-(3-methylbutyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl})[1-(1,2-oxazol-3-yl)ethyl]amine
1-cyclobutanecarbonyl-N-{2-[4-(dimethylamino)phenyl]ethyl}piperidine-4-carboxamide
(3-{[1-(5-chlorothiophene-2-carbonyl)pyrrolidin-3-yl]methyl}phenyl)methanol
4-[2-(morpholin-4-ylmethyl)piperidine-1-carbonyl]benzene-1-sulfonamide
1-[3-(1H-pyrazol-1-yl)propyl]-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
3-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidine-1-carbonyl]-6-ethyl-1,5-dimethyl-1,2-dihydropyridin-2-one
(3S,4S)-1-{[2-(butylsulfanyl)pyrimidin-5-yl]methyl}-4-methylpiperidine-3,4-diol
(3aS,6aS)-2-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-3-propoxypiperidine
6-ethyl-1,5-dimethyl-3-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]-1,2-dihydropyridin-2-one
2-[2-chloro-4-(pyrrolidin-1-ylmethyl)phenoxy]-6-(trifluoromethyl)pyridine
(3S,9aR)-2,3-dimethyl-8-{[1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-(4-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1,4-diazepan-1-yl)-2-methoxyethan-1-one
8-(5-methyl-1,3,4-thiadiazol-2-yl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}pyrrolidine-3-carboxamide
(2S,4S)-4-cyclobutaneamido-N-[(3,4-dimethoxyphenyl)methyl]-1-methylpyrrolidine-2-carboxamide
1-[(1R,3S,4S)-3-hydroxy-4,7,7-trimethylbicyclo[2.2.1]heptane-1-carbonyl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-3-(piperidin-3-yl)benzamide
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(2-methyl-4-phenylpyridine-3-carbonyl)pyrrolidin-3-yl]methanol
3-(1H-imidazol-1-ylmethyl)-1-(1H-imidazol-4-ylmethyl)piperidine
3-(2H-1,3-benzodioxol-5-yl)-5-{[3-(methylsulfanyl)phenyl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
{3-[(2,4-difluorophenyl)methyl]-1-[1-(2-phenylethyl)piperidin-4-yl]piperidin-3-yl}methanol
6-ethyl-N-[3-(1H-imidazol-1-yl)propyl]-2-methylquinoline-4-carboxamide