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5-{[2-(2-cyclohexylpyrimidin-5-yl)-1H-imidazol-1-yl]methyl}-N,N-dimethylfuran-2-carboxamide
1-(2-methoxy-5-{[methyl(pyrazin-2-ylmethyl)amino]methyl}phenoxy)-3-(piperidin-1-yl)propan-2-ol
2-[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propanoic acid
ethyl 4-{2-[2-({[4-(methoxycarbonyl)phenyl]methyl}amino)ethyl]-5-oxopyrrolidin-1-yl}piperidine-1-carboxylate
N,N-dimethyl-5-(1-methyl-1H-1,3-benzodiazole-5-carbonyl)-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
4-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-N,N-dimethylaniline
4-[4-(2-methoxyphenyl)-6-methyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carbonyl]-1λ6-thiomorpholine-1,1-dione
3-{1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-1-(4-methylpiperazin-1-yl)propan-1-one
3-[5-(4-chlorophenyl)-1H-pyrrol-2-yl]-1-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}propan-1-one
N-benzyl-2,7-dioxo-N-(1,3-thiazol-2-ylmethyl)-1,3-diazepane-4-carboxamide
1-(2-benzyl-1,3-thiazole-4-carbonyl)-4-hydroxypiperidine-4-carboxylic acid
N-[2-(dimethylamino)ethyl]-N'-(4-methylphenyl)-N-(oxolan-2-ylmethyl)propanediamide
9-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-hydroxyethyl)-N-methylacetamide
(3S,4R)-1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
(3aS,6aS)-2-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
{2-fluoro-5-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]phenyl}methanol
[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]({[2-(ethylsulfanyl)pyrimidin-5-yl]methyl})methylamine
3-(3-hydroxy-3-methylbutyl)-N-(2-hydroxyethyl)-N-(2-methylpropyl)benzamide
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-1,2,3-thiadiazole-4-carboxamide
4-{4-[3-(4-fluorophenoxy)propyl]piperazine-1-carbonyl}-N-methylpyridin-2-amine
2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]-N-[(4-methylphenyl)methyl]-N-(propan-2-yl)acetamide
methyl 2-(cyclopentylsulfamoyl)-6-(1-phenylcyclopropanecarbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(pyrazin-2-yl)piperazin-2-one
1-cyclohexyl-3-[(4-methoxyphenyl)methyl]-5-(4H-1,2,4-triazol-4-ylmethyl)-1H-1,2,4-triazole
[(3R,5R)-5-[(dimethylamino)methyl]-1-(4,6-dimethylpyridine-3-carbonyl)piperidin-3-yl]methanol
3-[(3R,4S)-3-(3-methyl-1-propyl-1H-pyrazole-4-amido)-4-(propan-2-yl)pyrrolidin-1-yl]propanoic acid
2-[2-({3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}methyl)phenoxy]acetic acid
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-1-(2-hydroxyethyl)-1H-1,3-benzodiazole-5-carboxamide
N4-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-5-ethyl-N4-methylpyrimidine-2,4-diamine
N-(1-carbamoylcycloheptyl)-1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
N-[2-(1-methylpiperidin-2-yl)ethyl]-6-(pyridin-4-yl)pyridine-3-carboxamide
1-{3-[6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}-2-(propylsulfanyl)ethan-1-one
1-{3-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-2-(furan-2-yl)ethane-1,2-dione
2-methoxy-1-(4-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-1-carbonyl}piperidin-1-yl)ethan-1-one
methyl 3-[(3S,4R)-4-(4-methylpiperazin-1-yl)-1-(1-methylpiperidin-4-yl)piperidin-3-yl]propanoate
2-[(4-chlorophenyl)methyl]-N-[1-(pyrimidin-4-yl)ethyl]-1,3-benzoxazole-5-carboxamide
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-N-(furan-2-ylmethyl)oxolane-2-carboxamide
5-methyl-1-(3-methylphenyl)-4-[2-(methylsulfanyl)pyridine-3-carbonyl]piperazin-2-one
N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
2-chloro-N-methyl-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}pyridine-4-carboxamide
N-cyclopropyl-2-[2-methyl-4-oxo-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
N-(1-hydroxypropan-2-yl)-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
N-[(3S,7S,8aS)-3-[(benzyloxy)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-fluorobenzamide
benzyl (1S,5R)-7-oxo-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxylate
5-(2-methoxyacetamido)-1-methyl-N-{[1-(2-methylpropyl)piperidin-4-yl]methyl}-2-(pyridin-4-yl)-1H-1,3-benzodiazole-7-carboxamide
[(2S,6S)-4-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
1-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-4-{[2-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
(1S,5R)-6-benzyl-3-[(3-methyl-1-phenyl-1H-pyrazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-(propan-2-yl)-2-(3,4,5-trimethoxyphenyl)pyrimidin-4-amine