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6-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-9H-purine
4-[(2-chlorophenyl)methyl]-9-methoxy-7-(4-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-ethyl-3-{1-[2-(methylamino)pyridine-3-carbonyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{5-[3-(pyrazin-2-yl)-1H-pyrazol-1-yl]quinolin-8-yl}acetamide
2-(2-{[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}phenoxy)ethan-1-ol
6-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-3-(8-methoxy-2-methylquinolin-5-yl)-1-methyl-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
9-[(5-fluoro-2-methylphenyl)methyl]-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{4-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]phenyl}-4-methylpiperazine
2-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]quinoline
2-ethyl-4-({4-[4-(methylsulfanyl)phenyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)pyrimidine
7-[(5-chlorothiophen-2-yl)methyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
2-{5-[2-(5-methylfuran-2-yl)propyl]-4-phenyl-1H-imidazol-1-yl}acetamide
4-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-1-(propan-2-yl)pyrrolidin-2-one
N-(adamantan-2-ylmethyl)-6-({methyl[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]amino}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
4-{[(2,3-dimethoxyphenyl)methyl]amino}-N,N-diethyl-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
1-{3-[(diethylamino)methyl]phenyl}-3-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-methylurea
[(3R,4R)-1-(2-fluoro-4-methylbenzoyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
[(3R,4R)-1-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)pyrrolidin-3-yl]methanol
N,N-dimethyl-2-{4-[1-(2-methylphenyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}acetamide
1-methyl-3-phenyl-8-(pyridin-4-ylmethyl)-1,8-diazaspiro[4.5]decan-2-one
N-(4-chlorophenyl)-2-[2-({methyl[1-(1,3-thiazol-2-yl)ethyl]amino}methyl)-4-phenylphenoxy]acetamide
3-[(1-{2-methylimidazo[1,2-a]pyridine-3-carbonyl}pyrrolidin-3-yl)methyl]benzoic acid
(3R,4R)-1-{[2-(adamantan-1-yl)-1,3-thiazol-4-yl]methyl}-4-aminopiperidin-3-ol
N-(oxolan-2-ylmethyl)-N-{[3-(thiophen-3-ylmethoxy)phenyl]methyl}pyridine-4-carboxamide
5-(2H-1,3-benzodioxole-5-carbonyl)-3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
1-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-4-[(3-fluorophenyl)methyl]piperazine
N-methyl-2-({[4-methyl-3-(propan-2-yl)phenyl]carbamoyl}amino)pentanamide
N-[4-(5-chloro-3-methyl-1H-pyrazol-1-yl)phenyl]-2-(morpholin-3-yl)acetamide
[(4-chlorophenyl)methyl]({3-[4-(morpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]propyl})amine
(3aR,6aR)-2-(2,4-difluorobenzoyl)-5-(2-methoxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[(1S,5R)-6-(cyclopropylmethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]-4,6-dimethylpyridine-3-carbonitrile
4-{[(1R)-1-carbamoylethyl]amino}-N-[(2-methoxyphenyl)methyl]pyridine-2-carboxamide
2-{1-[2-(adamantan-1-yl)acetyl]-3-oxopiperazin-2-yl}-N-methylacetamide
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)propanamide
5-[(2R)-2-amino-2-phenylacetyl]-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
(1S,5R)-N-(3-methoxyphenyl)-3-methyl-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
1-[(2,3-dimethyl-1H-indol-7-yl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
methyl 1-[(3R,5S)-1-(cyclohexylmethyl)-5-({[3-(trifluoromethyl)phenyl]methyl}carbamoyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
1-ethyl-5-({4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}methyl)-1H-indole
3-({3-[(dimethylamino)methyl]-3-hydroxypiperidin-1-yl}methyl)-2-methoxy-6-(propan-2-yl)-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
N'-({1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-3-yl}methyl)ethanediamide
N-[(2-methoxyphenyl)methyl]-3-oxo-N-propyl-2,3-dihydro-1H-indene-1-carboxamide
N-[(2-methoxyphenyl)methyl]-6-methyl-2-(pyridin-3-yl)pyrimidin-4-amine
4-methyl-2-[4-(thiophen-3-ylmethyl)piperazin-1-yl]-6-(trifluoromethyl)pyrimidine
N-(2-{imidazo[1,2-a]pyridin-3-yl}ethyl)-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
N-(3-methoxypropyl)-3-{[(5-methyl-1,2-oxazol-3-yl)methyl]sulfamoyl}benzamide
N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
4-({1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]piperidin-2-yl}methyl)morpholine
1-({5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)cyclopropan-1-amine
methyl 2-(2-{3-methyl-1-phenyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}phenoxy)acetate