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5-methyl-4-(4-methyl-1H-imidazole-2-carbonyl)-1-(3-phenylphenyl)piperazin-2-one
[(1-cyclopentylpiperidin-3-yl)methyl]({[5-(methoxymethyl)furan-2-yl]methyl})[2-(piperidin-1-yl)ethyl]amine
2-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-N-(propan-2-yl)pyridine-4-carboxamide
3-[(3R,4S)-1-(7-fluoro-3-methyl-1H-indole-2-carbonyl)-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
1-[3-({2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}amino)propyl]pyrrolidin-2-one
1-(cyclopropylmethyl)-N-ethyl-5-(thiolan-3-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-({1-[6-(3-methylpiperazin-1-yl)pyridine-3-carbonyl]piperidin-4-yl}methyl)pyrrolidin-2-one
N-[(3R,7S,8aS)-3-(hydroxymethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-methoxybenzamide
N-[1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(2-oxopyrrolidin-1-yl)benzamide
2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]-N-(2-phenylethyl)piperidine-1-carboxamide
N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-1-(oxan-4-yl)piperidine-3-carboxamide
4-chloro-3-({[1-(6-methylpyridin-3-yl)ethyl]carbamoyl}amino)-N-(propan-2-yl)benzamide
2-{1-cyclopropyl-2,5-dioxo-3-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl}-N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-N-methylacetamide
N-methyl-2-(4-methyl-1H-pyrazol-1-yl)-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
(2R,3R)-3-(dimethylamino)-1'-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
8-[(4-chloro-2-fluorophenyl)methyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
7-methoxy-N-(3-methoxypropyl)-N,4-dimethylquinazolin-2-amine
(3R,5R)-N-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
[2-({[2-(methoxymethyl)pyrimidin-5-yl]methyl}[(5-methylthiophen-2-yl)methyl]amino)ethyl]dimethylamine
5,6-dimethyl-2-oxo-N-[1-(thian-4-yl)piperidin-4-yl]-1,2-dihydropyridine-3-carboxamide
N-[(1-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}piperidin-3-yl)methyl]-4-fluorobenzamide
N-(1H-1,3-benzodiazol-2-yl)-2-{[(1-methyl-1H-imidazol-2-yl)methyl](propyl)amino}acetamide
7-(3-chlorophenyl)-4-[(3-methylpyridin-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(cyclohexylmethyl)-N,N-dimethyl-5-(morpholin-4-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
5-(2-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}-2-oxoethyl)-2-methyl-3,4-dihydropyrimidin-4-one
(4aS,8aR)-6-(2-cyclopropyl-4-methylpyrimidine-5-carbonyl)-1-propyl-decahydro-1,6-naphthyridin-2-one
3-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propanoic acid
N-(2-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)-6-oxo-1,6-dihydropyridine-3-carboxamide
8-methoxy-2-methyl-5-[6-(thiomorpholin-4-yl)pyridazin-3-yl]quinoline
3-(diphenylmethyl)-5-(oxolan-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
3-({2-[1-(2-hydroxyethyl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}(methyl)amino)-1λ6-thiolane-1,1-dione
7-(4-{2-cyclobutyl-3H-imidazo[4,5-b]pyridin-3-yl}piperidine-1-carbonyl)-2,3-dimethyl-1H-indole
({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)[3-(1H-pyrazol-1-yl)propyl](pyridin-3-ylmethyl)amine
3-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-ylmethyl}phenol
3-fluoro-5-methyl-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
3-chloro-N-[2-(dimethylamino)ethyl]-4-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]oxy}benzamide
3-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-[4-(1H-1,2,4-triazol-1-yl)phenyl]urea
N-(pyrazin-2-yl)-2-({1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}amino)acetamide
9-(5-acetylpyridin-2-yl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
methyl 3-({[3-(4-fluorophenyl)phenyl]formamido}methyl)-5-(pyrazine-2-amido)benzoate
N-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-{[4-(3-chlorophenyl)-5-({methyl[(2E)-3-phenylprop-2-en-1-yl]amino}methyl)-4H-1,2,4-triazol-3-yl]sulfanyl}propan-1-ol
1-methanesulfonyl-N-(4-methoxy-4-methylpentan-2-yl)piperidin-4-amine
2-(dimethylamino)-4-methyl-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]pyrimidine-5-carboxamide
1-(2-methoxyethyl)-4-{1-[4-(1H-pyrazol-1-yl)phenyl]piperidin-4-yl}piperazine
N-(2-{1-[(4-methylthiophen-2-yl)sulfonyl]piperidin-2-yl}ethyl)acetamide
2-(3-hydroxypiperidin-1-yl)-1-[4-(quinazolin-4-yl)piperazin-1-yl]ethan-1-one
N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}pyrimidin-2-amine
N,N-dimethyl-4-(2-oxo-5,5-diphenylpiperidin-1-yl)butanamide
N-[(2-fluorophenyl)methyl]-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide