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N-(1-benzylpyrrolidin-3-yl)-3-{1-[2-(furan-2-yl)-2-oxoacetyl]piperidin-4-yl}propanamide
1-(adamantan-1-yl)-3-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}urea
[1-(3,4-dimethoxyphenyl)propan-2-yl](methyl){2-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}amine
(4aS,8aR)-1-(3-hydroxypropyl)-6-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-decahydro-1,6-naphthyridin-2-one
6-(4-methoxy-3,5-dimethylphenyl)-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
N,N-diethyl-1-[(1s,4s)-4-(3,4-dimethoxybenzamido)cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
3-[(oxolan-3-yl)sulfamoyl]-N-[2-(pyrazin-2-yl)ethyl]benzamide
2-[2-(3-chloro-2,6-difluorophenyl)acetyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
N-[(1-ethylpyrrolidin-2-yl)methyl]-6-(methoxymethyl)pyrimidin-4-amine
5-(quinolin-3-yl)pyrazin-2-amine
5-{1-[(2Z)-2-fluoro-3-phenylprop-2-enoyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-(pyridin-2-yl)imidazolidine-2,4-dione
6-(4-chlorophenyl)-N-methyl-N-(1-methylpyrrolidin-3-yl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
{4-[({[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)methyl]oxan-4-yl}methanol
3-methoxy-N-[2-(3-methylphenyl)-1,3-benzoxazol-6-yl]pyrrolidine-1-carboxamide
3-(2-{3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}-2-oxoethyl)-1,3-oxazolidin-2-one
5-methoxy-2-{[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-4H-pyran-4-one
1-(2-benzyl-1,3-thiazole-4-carbonyl)-4-methanesulfonyl-1,4-diazepane
1-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]-3-(1H-pyrazol-1-yl)propan-1-one
2-{[2-(3,4-dichlorophenyl)morpholin-4-yl]methyl}-5-methoxy-4H-pyran-4-one
N-{[4-(pyrrolidine-1-carbonyl)phenyl]methyl}thiolan-3-amine
(3S,4R)-1-cyclopentyl-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
5-acetyl-N-[1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]thiophene-2-carboxamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
1-(piperidin-4-ylmethyl)-3-[5-(thiophen-2-yl)-1,3,4-thiadiazol-2-yl]urea
4-chloro-3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1-methyl-1H-indazole
N-[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]-2-methyl-1,3-thiazole-4-carboxamide
1-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
2-(2,5-dimethylphenyl)-1-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
(1S,5R)-6-(3-fluoro-4-methoxybenzoyl)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-{2-[4-(3-chlorophenyl)-3-oxopiperazin-1-yl]-2-oxoethyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-[4-hydroxy-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-1-yl]ethan-1-one
(1R,5R)-N,N-dimethyl-6-(3-propyl-1H-pyrazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
3-(2,3-difluorophenyl)-5-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
1-{2-[2-(cyclohex-3-en-1-yl)-1H-imidazol-1-yl]ethyl}-3,5-dimethyl-1H-1,2,4-triazole
N3-methyl-N5-[(3-methylphenyl)methyl]-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
[(5-fluoro-1H-indol-2-yl)methyl](methyl){[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amine
(2R,3R,6R)-3-(2-methoxyphenyl)-5-(pyrimidin-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-[2-(dimethylamino)ethyl]-8-(2,2-dimethylpropyl)-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(5-amino-1H-1,2,4-triazol-3-yl)methyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
3-[(2-fluorophenyl)methoxy]-1-(6-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)azetidine
4-ethyl-3-[(1-{6-[(propan-2-yl)amino]pyrimidin-4-yl}piperidin-4-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
[(3-fluorophenyl)methyl]({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(2-methoxyethyl)amine
3-[(3S,7S,8aS)-3-[(2S)-butan-2-yl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(naphthalen-1-yl)urea
(3S,4S)-4-cyclopropyl-1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]pyrrolidine-3-carboxylic acid
(3S,4R)-1-[2-(4-methyl-1H-pyrazol-1-yl)acetyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
N-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4-oxopentanamide
3-[methyl({8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl})amino]propane-1,2-diol
4-methyl-N-[2-methyl-4-(pyrrolidine-1-carbonyl)phenyl]-1,4-diazepane-1-carboxamide
5-fluoro-3-methyl-2-{4-[2-(pyridin-4-yl)ethyl]piperazine-1-carbonyl}-1H-indole
1-cyclopentyl-N3-[1-(furan-2-yl)ethyl]-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide