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1-ethyl-3-methyl-N-[(2-methylphenyl)methyl]-N-(prop-2-en-1-yl)-1H-pyrazole-5-carboxamide
6-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]quinoline
4-{1-[3-(2-oxopyrrolidin-1-yl)propanoyl]piperidin-3-yl}benzoic acid
3-[2-amino-4-(azocan-1-yl)-6-methylpyrimidin-5-yl]propanoic acid
N-[(1-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}piperidin-3-yl)methyl]cyclobutanecarboxamide
8-(4-methyl-5-phenylthiophene-2-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(2R,6R)-4-methanesulfonyl-10-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)-6-oxo-1,6-dihydropyridine-3-carboxamide
2-cyano-N-methyl-N-[1-(pyridin-3-yl)ethyl]benzamide
4-{[2-(2-butyl-1H-imidazol-4-yl)-1H-imidazol-1-yl]methyl}pyridine
2-(3-methyl-1,2-oxazol-5-yl)-1-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
(3R,4R)-3-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)piperidin-4-ol
1-[4-(2,5-dihydro-1H-pyrrol-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)ethan-1-one
4-[(3-fluorophenyl)methyl]-1-[1-(2-phenylethyl)piperidin-4-yl]-1,4-diazepan-5-one
7-(4-methylphenyl)-4-[2-(1H-pyrrol-1-yl)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-(4-methoxypyridin-2-yl)-5-[2-(piperidin-2-yl)ethyl]phenol
4-hydroxy-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2-(2-methyl-1,3-thiazol-4-yl)pyrimidine-5-carboxamide
3,3-dimethyl-1-[(3S,4R)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)-4-(propan-2-yl)pyrrolidin-3-yl]urea
N-[(1-{[2-(2,2-dimethylpropanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}piperidin-3-yl)methyl]acetamide
3-(1-propyl-1H-1,2,3-triazol-4-yl)-1-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}urea
1-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}-2,2-dimethylpropan-1-one
1-[(3ar,6ar)-octahydropyrrolo[3,4-c]pyrrole-3a-carbonyl]-4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]piperidine
3-(1-methylpiperidin-2-yl)-N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
3-(2-fluorophenyl)-N-[1-(methoxymethyl)cyclopentyl]-1H-pyrazole-4-carboxamide
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(6-methoxypyridin-2-yl)benzamide
(1S,5R)-3-benzyl-6-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
1-(piperidin-1-yl)-2-{2-[1-(pyrrolidin-3-yl)-1H-imidazol-2-yl]phenoxy}ethan-1-one
8-[(4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazin-1-yl)methyl]quinoline
(3R,5S)-N3-[(3,4-dimethylphenyl)methyl]-N5-(6-methylpyridin-3-yl)piperidine-3,5-dicarboxamide
3-(hydroxymethyl)-1-(2,4,5-trimethylbenzoyl)piperidin-3-ol
N-(1-benzylpyrrolidin-3-yl)-3-{1-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]piperidin-4-yl}propanamide
4-{1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)sulfonyl]piperidin-3-yl}benzoic acid
N-cyclohexyl-N-[(3,4-dimethoxyphenyl)methyl]oxane-2-carboxamide
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-3-(3-hydroxy-3-methylbutyl)benzamide
N,N-dimethyl-4-{4-[(4-methylphenyl)methyl]-3-oxopiperazine-1-carbonyl}piperidine-1-carboxamide
4-(2-methoxy-5-methylphenyl)-3-(1-methoxyethyl)-4H-1,2,4-triazole
N-[(2-methylphenyl)methyl]-5-(naphthalen-1-yl)-1,2,4-triazin-3-amine
N-(6-chloropyridin-3-yl)-3-(morpholin-4-yl)azetidine-1-carboxamide
(4-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine-1-carbonyl}phenyl)methanamine
N-(4-chloro-3-methylphenyl)-2-({[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}amino)acetamide
(3S,4S)-1-(1-methyl-5-phenyl-1H-pyrrole-2-carbonyl)-4-propylpyrrolidine-3-carboxylic acid
(2R,3R)-3-(morpholin-4-yl)-1'-(pyrimidin-2-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-(2-hydroxyethyl)-N-methyl-1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-3-carboxamide
4-{[3-(2-chlorophenoxy)azetidin-1-yl]methyl}-2-methyl-1,3-oxazole
6-methyl-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-{5-acetyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(pyridin-3-yl)ethan-1-one
2-methyl-3-{2-[2-(oxolan-3-yl)-1H-imidazol-1-yl]ethyl}-1-azatricyclo[6.3.1.04,12]dodeca-2,4,6,8(12)-tetraene
4-(cyclopropylmethyl)-1-(1-ethyl-1H-indole-5-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
methyl 3-[1-benzyl-2,4-dioxo-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decan-8-yl]propanoate