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N-[(4-methoxyphenyl)methyl]-1-methyl-N-propyl-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
1-[(2,3-dimethoxyphenyl)methyl]-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
4-[(1-cyclopentylpiperidin-4-yl)oxy]-3-methoxybenzamide
1-(4-fluorophenyl)-4-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}butane-1,4-dione
ethyl 1-[1-(2-cyclooctyl-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl)piperidine-3-carbonyl]piperidine-4-carboxylate
1-(3-chlorothiophene-2-carbonyl)-4-[(dimethylamino)methyl]azepan-4-ol
N-[2-(dimethylsulfamoyl)ethyl]-1-(2-hydroxyethyl)-1H-1,3-benzodiazole-5-carboxamide
ethyl 4-[2-(6-methylquinolin-5-yl)-1H-imidazol-1-yl]piperidine-1-carboxylate
3-({2-[2-(5-ethylfuran-2-yl)-1H-imidazol-1-yl]ethyl}sulfanyl)-4-methyl-4H-1,2,4-triazole
1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-(4-{6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-1,4-diazepan-1-yl)-2-methoxyethan-1-one
2-(2-methoxyphenyl)-5-{[4-(3-methylpyridin-2-yl)piperazin-1-yl]methyl}pyrimidine
4-{2-oxo-4-[2-(2,3,6-trimethylphenoxy)acetyl]piperazin-1-yl}benzonitrile
2-(1H-imidazol-2-yl)-N-[(2-methylphenyl)methyl]-N-(oxolan-2-ylmethyl)benzamide
[2-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-1,3-thiazol-4-yl]methanol
5-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-1H-1,2,3-benzotriazole
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
7-(2-methoxyethyl)-2-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}-2,7-diazaspiro[4.5]decan-6-one
{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}[(3-chlorophenyl)methyl]methylamine
2-[1-(1-methylpiperidin-4-yl)-4-(2-methylquinolin-4-yl)piperazin-2-yl]ethan-1-ol
2-(3-hydroxypiperidin-1-yl)-1-[3-(2-methylphenoxy)azetidin-1-yl]ethan-1-one
4-[(3-methylphenyl)methyl]-1-[1-(pyridin-2-yl)piperidine-3-carbonyl]-1,4-diazepan-5-one
5-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine-1-carbonyl}-3,4-dihydropyrimidin-4-one
N-(4-ethoxy-2-fluorophenyl)-3-methoxypyrrolidine-1-carboxamide
1-{[6-(dimethylamino)pyridin-3-yl]methyl}azepan-3-amine
N-(2-phenylethyl)-3-(phenylmethanesulfonamidomethyl)piperidine-1-carboxamide
3-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-1-(2-methoxy-5-methylphenyl)-3-methylurea
3-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1-(4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)urea
N,N-dimethyl-1-{[2-(pyridine-4-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]sulfonyl}pyrrolidin-3-amine
N-(5-{[bis(2-methoxyethyl)carbamoyl]amino}-2-fluorophenyl)acetamide
3-(2,5-dioxoimidazolidin-4-yl)-N-[(8-methoxyquinolin-5-yl)methyl]-N-methylpropanamide
3-{1-[2-(4H-1,2,4-triazol-4-yl)ethyl]piperidin-3-yl}-N-[4-(trifluoromethyl)phenyl]propanamide
N-(1,3-dimethyl-1H-pyrazol-4-yl)-2-{2-ethyl-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}acetamide
1-ethyl-3-(2-methylpropyl)-N-[(3R,4R)-4-(morpholin-4-yl)oxolan-3-yl]-1H-pyrazole-5-carboxamide
9-(2-ethylpyrimidine-5-carbonyl)-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecane
N-methyl-2-(2-methyl-1,3-thiazol-4-yl)-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)acetamide
N-methyl-N-[(5-methylfuran-2-yl)methyl]morpholine-2-carboxamide
1-(4-ethylpiperazin-1-yl)-3-{1-[(2-fluoro-4-methoxyphenyl)methyl]piperidin-4-yl}propan-1-one
N-[(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-(dimethylamino)-N-[1-(4-methanesulfonylphenyl)propyl]-4-methylpyrimidine-5-carboxamide
N-[(3-methylthiophen-2-yl)methyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
3-[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-4,5,6,7-tetrahydro-1,2-benzoxazole
6-{4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-N,N-dimethylpyrimidin-4-amine
methyl[3-(1-methyl-1H-imidazol-2-yl)propyl][2-methyl-2-(piperidin-1-yl)propyl]amine
N-[2-(quinolin-8-yloxy)ethyl]-1H-pyrazole-4-carboxamide
4-({[(4-hydroxy-5,8-dimethylquinolin-2-yl)methyl]amino}methyl)benzene-1-sulfonamide
1-{1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-4-(2-methylphenyl)piperazine
2-[2-(1H-imidazol-4-yl)ethyl]-8-[(4-methylphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
3-[(3R,4S)-1-[(5-ethylfuran-2-yl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
3-[({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]-2,2-dimethylpropan-1-ol