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N-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]-5-fluoro-1H-indole-2-carboxamide
1-ethyl-N-[(4-fluorophenyl)methyl]-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-{2-[3-(morpholin-4-yl)-3-oxopropyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}propanamide
4-(2-oxopyrrolidin-1-yl)-N-[1-(2-phenylethyl)piperidin-3-yl]benzamide
3-(5-{2-[2-(6-methyl-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]ethyl}-1,2,4-oxadiazol-3-yl)pyridine
4-(2-amino-6-ethyl-5-methylpyrimidin-4-yl)-1-(3,5-dimethylphenyl)piperazin-2-one
(3S,4R)-1-({[2-(2-methoxyphenyl)ethyl]carbamoyl}methyl)-4-phenylpyrrolidine-3-carboxylic acid
5-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-N,N-dimethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-{1-[(2-methoxypyrimidin-5-yl)methyl]piperidin-3-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1'-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
4-({3-[(3-fluorophenyl)amino]piperidin-1-yl}methyl)phenol
4-methoxy-N-(2-{7-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
N-[2-(ethylsulfanyl)phenyl]-4-[(4-fluorophenyl)methyl]-3-oxopiperazine-1-carboxamide
2-{1-[1-(propan-2-yl)piperidin-4-yl]-4-(pyrazin-2-yl)piperazin-2-yl}ethan-1-ol
(3aR,6aR)-2-cyclopentyl-N-[2-(ethanesulfonyl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)benzoic acid
5-methyl-N-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}pyrazolo[1,5-a]pyrimidin-7-amine
2-[(2-{[2-(dimethylamino)ethyl](oxolan-2-ylmethyl)carbamoyl}phenyl)amino]acetic acid
N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-2,1,3-benzothiadiazole-4-sulfonamide
5-[(dimethylamino)methyl]-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1,3,4-oxadiazole-2-carboxamide
N-methyl-N-(pyrimidin-4-ylmethyl)-2-(pyrrolidin-3-yl)benzamide
1-{3-[5-(2-fluorophenyl)-2-(pyridin-3-yl)pyrimidin-4-yl]piperidin-1-yl}ethan-1-one
4-({1-[1-(4-fluorophenyl)cyclopropanecarbonyl]piperidin-4-yl}oxy)pyridine
3-[1-(7-chloro-3,5-dimethyl-1-benzofuran-2-carbonyl)pyrrolidin-2-yl]-4-methyl-1,2,5-oxadiazole
(3S,4S)-4-(4-fluorophenyl)-1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}piperidin-3-ol
2-chloro-4-({4-[(4-ethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenol
4-({5-[1-(6-ethylpyrimidin-4-yl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)morpholine
2-[(7-methanesulfonyl-4-methylquinazolin-2-yl)(methyl)amino]-N-methylacetamide
2-(3-cyclopentyl-5-{2,5,7-trimethylpyrazolo[1,5-a]pyrimidin-3-yl}-1H-1,2,4-triazol-1-yl)pyridine
2-fluoro-6-[4-(pyrrolidin-2-yl)phenyl]benzamide
N,N-dimethyl-1-{[5-(2-methylpropyl)thiophen-2-yl]methyl}pyrrolidin-3-amine
[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]({[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-4-(1H-pyrazol-4-yl)butanamide
1-[(5-methylfuran-2-yl)methyl]-3-(pyrrolidin-1-yl)piperidine
4-acetyl-N-{3-[(2-methylpiperidin-1-yl)methyl]phenyl}-1,4-diazepane-1-carboxamide
5-methoxy-N,1-dimethyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-1H-indole-2-carboxamide
5-methanesulfonyl-1'-(pyridin-2-ylmethyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-[(2S)-oxolan-2-ylmethyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
ethyl 4-[1-(4-methyl-1H-pyrrole-2-carbonyl)piperidin-3-yl]piperazine-1-carboxylate
6-[(diethylamino)methyl]-N-(pyrrolidin-3-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
6-(benzyloxy)-1-(2-methylpropyl)-4-[3-(6-oxo-1,6-dihydropyridazin-3-yl)propanoyl]-1,4-diazepan-2-one
2-(5-chloro-2-methoxyphenyl)-2-[4-(thiophen-3-ylmethyl)piperazin-1-yl]acetic acid
1-[2,3-dimethyl-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}urea
N-cyclohexyl-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N3-[2-(3-chlorophenyl)ethyl]-N5-cyclohexyl-1-(2-methoxyethyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-(adamantan-1-yl)-4-hydroxy-N-(pyridin-4-ylmethyl)pyrimidine-5-carboxamide
1-methyl-8-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-{2-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
N-[2-(pyrrolidine-1-sulfonyl)ethyl]-1H-1,2,3-triazole-5-carboxamide
(2R,4S)-4-hydroxy-1-(quinoline-2-carbonyl)piperidine-2-carboxylic acid