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N-{1-[(2-chlorophenyl)methyl]-1H-pyrazol-5-yl}-4-(2-methoxyethyl)piperazine-1-carboxamide
1-{3-[1-(4-methoxyphenyl)-1H-1,2,4-triazol-5-yl]phenyl}pyrrolidin-2-one
4-{4-[(2-fluorophenyl)methyl]-1,4-diazepane-1-carbonyl}-1-oxaspiro[4.4]nonan-2-one
N3-(1-benzylpyrrolidin-3-yl)-N5-methyl-1-(3-methylbutyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
(3S,9aR)-3-[(4-hydroxyphenyl)methyl]-8-(4-phenylbenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]methyl}-1H-indole
5-[benzyl(butyl)amino]-1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]azepan-2-one
N-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
4-cyano-N-[1-(pyrimidin-2-yl)piperidin-3-yl]benzene-1-sulfonamide
N-methyl-4-{[4-(pyrrolidin-3-yl)piperazin-1-yl]methyl}benzene-1-sulfonamide
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-[3-(morpholin-4-yl)propyl]piperidine-3,5-dicarboxamide
N-[(3-hydroxypyrrolidin-3-yl)methyl]-3,6-dimethyl-1-benzofuran-2-carboxamide
ethyl[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl](oxan-2-ylmethyl)amine
N-benzyl-2-(2-methylphenyl)pyrrolidine-1-sulfonamide
N-methyl-3-(6-oxo-1,6-dihydropyridazin-3-yl)-N-(quinolin-5-ylmethyl)propanamide
N-ethyl-N-[(2-fluorophenyl)methyl]-3-(3-hydroxy-3-methylbutyl)benzamide
3-(4-chloro-1H-pyrazol-1-yl)-1-[2-(3-methoxyphenyl)pyrrolidin-1-yl]propan-1-one
5-(1,5-dimethyl-1H-pyrazol-4-yl)-N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-1,2-oxazole-3-carboxamide
5-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridine-2-carbonitrile
7-{2-[3-(methylsulfanyl)phenyl]acetyl}-2,7-diazaspiro[4.4]nonane-1,3-dione
3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-methyl-N-(thiophen-3-ylmethyl)benzamide
2-(cyclohex-1-en-1-yl)-1-(4-{[4-(2-hydroxyethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)ethan-1-one
2-[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidine-1-carbonyl]-4H-chromen-4-one
3-[5-(1,3-benzoxazol-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]-1-(pyrrolidin-1-yl)propan-1-one
(1R,3S)-3-amino-N-methyl-N-[(4-phenoxyphenyl)methyl]cyclohexane-1-carboxamide
[(2-fluoro-5-methoxyphenyl)methyl](methyl)(oxan-2-ylmethyl)amine
5-[1-(cyclopentylmethyl)pyrrolidin-2-yl]-N-[(2-methylpyridin-4-yl)methyl]thiophene-2-carboxamide
{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}(methyl)(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)amine
3-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)pyridin-2-ol
(4aR,8aR)-2-[(5-chlorothiophen-2-yl)methyl]-7-(pyrrolidine-1-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
N-[(3R,4S)-1-cyclopentyl-4-propylpyrrolidin-3-yl]-1-(1H-imidazol-1-ylmethyl)cyclopropane-1-carboxamide
3-[(3R,7S,8aS)-3-[(benzylsulfanyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2,4-dichlorophenyl)urea
3-(1H-1,3-benzodiazol-1-yl)-1-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}propan-1-one
4-{[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]sulfamoyl}-N-(pyrrolidin-3-yl)benzamide
6-(2-chlorophenyl)-N-(cyclopropylmethyl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-{3-methoxy-4-[(1-methylpiperidin-4-yl)oxy]benzoyl}-1,2,3,4-tetrahydroisoquinoline
2-[1-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)azetidin-3-yl]pyridine
N-ethyl-6-[2-(4-fluorophenyl)morpholin-4-yl]-N-methylpyridine-3-carboxamide
1-{6-methylthieno[2,3-d]pyrimidin-4-yl}-N-[2-(1,3-thiazol-2-yl)ethyl]piperidin-4-amine
N-{[1-(piperidin-1-yl)cyclohexyl]methyl}-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(1-methyl-1H-pyrazole-4-carbonyl)pyrrolidine-3-carboxylic acid
3-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1-methyl-1,2-dihydroquinoxalin-2-one
2-(4-chloro-3-methyl-1H-pyrazol-1-yl)-1-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
(3aS,6aS)-2-cyclobutanecarbonyl-5-[2-(3-fluorophenyl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-hydroxy-3-{[methyl(pyridin-2-ylmethyl)amino]methyl}-1-[(3-methylphenyl)methyl]piperidin-2-one
N-{[2-(dimethylamino)-7-methoxyquinolin-3-yl]methyl}-2-fluoro-N-(2-methoxyethyl)benzamide
1-(cyclopropylmethyl)-2-oxo-3-{[(thiophen-2-ylmethyl)carbamoyl]methyl}-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
N-[(3R,4R)-1-(4-ethyl-5-methylthiophene-3-carbonyl)-3-hydroxypiperidin-4-yl]pyridine-2-carboxamide
1-(2-chlorophenyl)-3-{1-[1-(5-methoxyfuran-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
2-ethyl-N-[3-(3-hydroxypiperidin-1-yl)propyl]pyrimidine-5-carboxamide