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1-{imidazo[1,2-a]pyridine-6-carbonyl}-3-(propoxymethyl)pyrrolidine
N-[2-(pyrrolidine-1-sulfonyl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
dimethyl[2-({[2-(3-methylphenyl)pyrimidin-5-yl]methyl}(oxolan-2-ylmethyl)amino)ethyl]amine
1-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-3-[5-(thiophen-2-yl)-1,3,4-thiadiazol-2-yl]urea
3-[2-(dimethylamino)ethyl]-1-ethyl-8-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(3-carboxybenzoyl)pyrrolidine-3-carboxylic acid
2-chloro-N-{1-[1-(2-hydroxyethyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
(4aS,8aR)-6-(3-fluoropyridin-2-yl)-1-[3-(methylsulfanyl)propyl]-decahydro-1,6-naphthyridin-2-one
(4aS,8aR)-6-[(3,5-dimethyl-1-benzofuran-2-yl)methyl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
2-{[(2-fluorophenyl)methyl](methyl)amino}-1-[6-hydroxy-4-(2-hydroxyethyl)-1,4-diazepan-1-yl]ethan-1-one
N-cyclopropyl-2-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]pyridine-4-carboxamide
4-{[4-(oxan-4-yl)piperazin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
3-(cyclohexylsulfamoyl)-5-(1H-pyrazol-1-yl)benzoic acid
ethyl 2-[2-({1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazol-4-yl}formamido)ethyl]-1,3-thiazole-4-carboxylate
(3R,4S)-1-cyclobutanecarbonyl-4-cyclopropylpyrrolidin-3-amine
4-[(3-fluorophenyl)methyl]-11-{[(1-methyl-1H-pyrazol-4-yl)methyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-[(1-phenyl-1H-pyrazol-4-yl)methyl]pyrazolo[1,5-a]pyridine-7-carboxamide
1-{2-[4-(3-methyl-3-phenylpiperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}piperazine
2-amino-4-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-5H,6H,7H-pyrrolo[2,3-h]quinoline-3-carbonitrile
2-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-4-(trifluoromethyl)pyridine
3,3,3-trifluoro-1-{3-[2-(4-methoxyphenyl)ethyl]piperidin-1-yl}propan-1-one
3-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-5-propyl-1,2-oxazole
3,5-dimethoxy-2-({methyl[(5-methylfuran-2-yl)methyl]amino}methyl)benzoic acid
methyl 5-{[5-(1,2-oxazol-5-yl)furan-2-yl]sulfonyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
6-[(4-methoxy-2,3-dimethylphenyl)methyl]-2-methyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
4-(2,6-dimethyl-4-oxo-1,4-dihydropyridine-3-carbonyl)-1-[(4-methoxyphenyl)methyl]piperazin-2-one
N-(2-methylpropyl)-1-[(1s,4s)-4-[(pyridin-3-ylmethyl)amino]cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
3-({[(2S)-5-oxopyrrolidin-2-yl]methyl}(pyridin-2-ylmethyl)carbamoyl)benzoic acid
(3aR,6aS)-5-(5-cyclopropyl-1,2-oxazole-3-carbonyl)-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1'-{furo[3,2-c]pyridin-4-yl}-1-methyl-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
4-(3,4-dichlorophenyl)-3-(1-methoxyethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
4-{[(benzylsulfamoyl)amino]methyl}-N-methylbenzamide
1-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-4-ethyl-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(furan-2-yl)-1-{3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}propan-1-one
2-(1-methyl-1H-imidazol-2-yl)-N-[2-(1-methylpiperidin-3-yl)ethyl]benzamide
methyl 3-(3-cyanopiperidine-1-carbonyl)-5-(cyclobutylmethoxy)benzoate
1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-4-[(4-methoxyphenyl)methyl]-1,4-diazepan-5-one
2-(1-tert-butyl-1H-pyrazol-4-yl)-N,5,7-trimethyl-N-(propan-2-yl)quinoline-4-carboxamide
1-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-5-oxopyrrolidine-3-carboxylic acid
4-(3,4-dimethoxybenzoyl)-2-(4-methylpentyl)morpholine
N-ethyl-3,6-dimethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
(2R,3R)-3-amino-1'-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-[2-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-oxoethyl]-1,2-dihydropyridin-2-one
2-methyl-N-[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]thieno[2,3-d]pyrimidin-4-amine
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(4-methyl-1H-imidazole-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N,2,2-trimethyl-4-oxo-3,4-dihydro-2H-pyran-6-carboxamide
1-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-4-(thiophen-2-ylmethyl)-1,4-diazepane
(4S)-1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
1-(cyclohexylmethyl)-N5-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N3,N3-dimethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1'-[(5-methoxy-1H-indazol-3-yl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol