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4-[5-(4-chlorophenoxy)-1,3-dimethyl-1H-pyrazol-4-yl]-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
N-cyclopropyl-2-methyl-N-({3-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)-1,3-thiazole-4-carboxamide
1-(5-methyl-1H-indazole-3-carbonyl)azepan-4-amine
1-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-3-[3-(furan-2-yl)-1H-1,2,4-triazol-5-yl]-1-methylurea
{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}({[2-(methylsulfanyl)pyrimidin-5-yl]methyl})amine
8-[4-(1H-pyrazol-3-yl)benzoyl]-1-oxa-8-azaspiro[4.5]decane
2-ethyl-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]pyridine-4-carboxamide
({5-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonane-3-carbonyl]-2-ethylfuran-3-yl}methyl)diethylamine
9-methoxy-7-(4-methylphenyl)-4-(oxolane-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
6-amino-2-(2-{4-[2-methyl-4-(1H-pyrazol-1-yl)phenyl]-1H-1,2,3-triazol-1-yl}ethyl)pyrimidin-4-ol
(3S,4S)-1-(3-fluorobenzoyl)-4-(naphthalen-2-yl)piperidin-3-ol
1-[2-(dimethylamino)ethyl]-N-methyl-5-oxo-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)pyrrolidine-3-carboxamide
N,N-dimethyl-2-(3-phenylpiperazine-1-carbonyl)-2,3-dihydro-1H-inden-2-amine
2-{1-[(5-methylfuran-2-yl)methyl]-4-(oxan-4-yl)piperazin-2-yl}ethan-1-ol
5-methyl-2-(naphthalen-1-yl)-4-{[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methyl}-1,3-oxazole
6-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
3-methyl-7-{5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl}-5,6,7,8-tetrahydro-2,7-naphthyridine-4-carbonitrile
(3S,4S)-4-cyclopropyl-1-(3,5-dichloro-2-methoxybenzoyl)pyrrolidine-3-carboxylic acid
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-4-methyl-1,3-oxazole-5-carboxamide
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-(3-methyl-1,2-oxazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-cyclopropyl-1-[1-(5-fluoropyridine-2-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
3-[2-oxo-2-(piperidin-1-yl)ethyl]-4-[(3-phenoxyphenyl)methyl]piperazin-2-one
8-(2-methylquinolin-4-yl)-1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1,8-diazaspiro[4.5]decane
8-(1,3-benzothiazol-2-ylmethyl)-1-methyl-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{[1-(azepan-1-yl)propan-2-yl]amino}-N-(propan-2-yl)acetamide
(4aS,7aR)-1-[(3,4-dimethoxypyridin-2-yl)methyl]-4-ethyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-1,3-dimethyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-[(4-fluorophenyl)methyl]-1-(5-methyl-1,2-oxazole-3-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
2-methyl-4-(piperidin-4-yl)-6-[3-(pyridine-2-carbonyl)piperidin-1-yl]pyrimidine
1-{4-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-4-oxobutyl}pyrrolidin-2-one
5-{3-[1-(3-methylbut-2-en-1-yl)-1H-pyrazol-3-yl]phenyl}pyrimidine
2-(1-{[3-(2-methylpropyl)-3H-imidazo[4,5-b]pyridin-2-yl]methyl}cyclopentyl)-1-(morpholin-4-yl)ethan-1-one
3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[3-(methylsulfanyl)propyl]piperidine
6-methyl-5-{5-[(2S)-1-methylpyrrolidin-2-yl]-1,2,4-oxadiazol-3-yl}-1,2,3,4-tetrahydro-2,7-naphthyridine
1-tert-butyl-N-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidine-3-carboxamide
[(5-{[(3-fluorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl](methyl)(pyridin-4-ylmethyl)amine
6-(3-fluorophenyl)-N-(2-methoxybutyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-[3-(cyclohexylsulfanyl)propyl]-5-methyl-1,3,4-oxadiazol-2-amine
1-[(1S,5R)-6-[3-(5-methylfuran-2-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
3-(2-ethyl-1H-1,3-benzodiazol-6-yl)-1-(2-methoxyethyl)-1-[(3-methylthiophen-2-yl)methyl]urea
N-[3-(4H-1,2,4-triazol-4-yl)propyl]pyridin-3-amine
methyl (2S)-1-{[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}pyrrolidine-2-carboxylate
3-(azepane-1-carbonyl)-1-methyl-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[(3-methoxyphenyl)methyl]-N-(2-methylpropyl)-3-(2-oxooxolan-3-yl)propanamide
4-(2-methylpropyl)-3-{2-oxo-2-[4-(thiomorpholin-4-yl)piperidin-1-yl]ethyl}piperazin-2-one
1-{6-[7-(3,6-dimethylpyrazin-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]pyridin-3-yl}ethan-1-one
3-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-3-methyl-1-[4-(2-methyl-5-oxopyrrolidin-1-yl)phenyl]urea
3-[(5-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]methyl}furan-2-yl)sulfanyl]-4-methyl-4H-1,2,4-triazole