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N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
1-{2-methoxy-5-[({[1-(propan-2-yl)piperidin-4-yl]methyl}amino)methyl]phenoxy}-3-(4-methylpiperazin-1-yl)propan-2-ol
4-(1-tert-butyl-1H-pyrrole-3-carbonyl)-1-(4-methylphenyl)piperazin-2-one
2-[1-(2,5-dichlorophenyl)-5-(methanesulfonamidomethyl)-1H-1,2,4-triazol-3-yl]acetamide
1-{4-[(cyclohex-1-en-1-ylmethyl)amino]-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}-2-methoxyethan-1-one
N-{[2-(dimethylamino)-7-methoxyquinolin-3-yl]methyl}-N-(2-methoxyethyl)cyclopropanecarboxamide
[2-ethoxy-5-(7-methyl-1H-1,3-benzodiazol-2-yl)phenyl]methanol
2-(2,4-dimethoxybenzenesulfonyl)-8-methyl-2,8-diazaspiro[4.5]decane
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-{2-[(3-methoxyphenyl)methyl]morpholin-4-yl}ethan-1-one
N,N-dimethyl-2-[(1S,5R)-6-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
4-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-1-oxaspiro[4.5]decan-2-one
6-methyl-1-[3-({5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)propyl]-1,2-dihydropyridin-2-one
4-{[(1S,6R)-3-methyl-4-oxo-3,9-diazabicyclo[4.2.1]nonan-9-yl]methyl}-1H-pyrazole-3-carboxylic acid
(3R,4S)-4-cyclopropyl-1-(5-phenyl-1,2,4-oxadiazol-3-yl)pyrrolidin-3-amine
4-[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]-1-phenylpiperazin-2-one
N-[3-(cyclohexyloxy)propyl]-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
N-(2-{1-[4-(5-methylpyrimidin-2-yl)phenyl]-1H-imidazol-4-yl}ethyl)acetamide
1-[4-(ethylsulfanyl)phenyl]-3-[1-(pyridin-3-ylmethyl)piperidin-4-yl]urea
1-(3-chlorophenyl)-4-(2,3-dihydro-1H-indene-5-carbonyl)piperazin-2-one
N-[2-(3-fluorophenyl)ethyl]-2-(4-{4-[(oxan-4-yl)amino]piperidin-1-yl}phenyl)acetamide
5-[4-(2,4-difluorophenyl)piperazine-1-carbonyl]quinoxaline
3-(3-methylphenyl)-1-[6-(4H-1,2,4-triazol-4-yl)pyridin-3-yl]-1H-pyrazole-4-carboxylic acid
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-{2-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]ethyl}acetamide
5-methyl-4-(1-methyl-1H-pyrazol-5-yl)-2-(4-methylpiperazin-1-yl)pyrimidine
[(6-chloropyridin-3-yl)methyl](methyl){[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}amine
N-(2-fluoroethyl)-1-(4-methoxyphenyl)-2,2-dimethylcyclopropane-1-carboxamide
2-[(1S,5R)-3-(5-chlorothiophene-2-carbonyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
3-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}propanoic acid
N-[2-(2,3-dimethoxyphenyl)ethyl]-7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-(pyridin-2-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
1-[(1-{6-[(2-methoxybutyl)amino]pyridine-3-carbonyl}piperidin-4-yl)methyl]pyrrolidin-2-one
8-(2-chloro-6-methylbenzenesulfonyl)-2-ethyl-2,8-diazaspiro[4.5]decan-3-one
1-ethyl-4-[(4-methoxypyridin-2-yl)methyl]piperazine-2,3-dione
(1H-imidazol-2-ylmethyl)[(2-methylphenyl)methyl](prop-2-en-1-yl)amine
N'-ethyl-N'-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N,N-dimethylbutanediamide
2-(3-fluorophenyl)-2-{[1-(4-fluorophenyl)cyclopropyl]formamido}acetic acid
(4aR,8aR)-2-cyclopentanecarbonyl-7-[2-(phenylsulfanyl)ethyl]-decahydro-2,7-naphthyridin-4a-ol
1-cyclohexyl-N-cyclopropyl-5-(3-methylpiperidine-1-carbonyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
methyl (2R,4S)-4-hydroxy-1-(3-methoxybenzenesulfonyl)piperidine-2-carboxylate
2-methyl-4-{3-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidine-1-carbonyl]phenyl}butan-2-ol
{1-[(2-chloro-4,5-dimethoxyphenyl)methyl]piperidin-2-yl}methanol
5-(1-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidin-2-yl)-3-phenyl-1,2,4-oxadiazole
3-{5-[(2E)-but-2-en-1-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-N-[2-(5,7-difluoro-2-methyl-1H-indol-3-yl)ethyl]acetamide
N-(1H-indol-3-yl)-2-(pyrrolidin-1-yl)benzamide
3-(2-ethyl-1H-imidazol-1-yl)-1-[3-(2-fluorophenoxymethyl)piperidin-1-yl]propan-1-one
2,6-dimethyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}pyrimidine-4-carboxamide
(2S,4S)-4-amino-1-(4-ethenylbenzoyl)-N-methylpyrrolidine-2-carboxamide
1-cyclopentanecarbonyl-N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]piperidine-4-carboxamide