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N-[(3R,4S)-1-[2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
5-[1-(2-phenylethyl)piperidin-4-yl]-5-(pyridin-3-yl)imidazolidine-2,4-dione
N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepine-3-carboxamide
1-(propan-2-yl)-4-{1-[4-(1H-pyrazol-1-yl)phenyl]piperidin-4-yl}-1,4-diazepane
1-ethyl-4-(5,6,7,8-tetrahydro-1,6-naphthyridine-6-carbonyl)pyrrolidin-2-one
2-[1-(hydroxymethyl)-9-[2-(1H-pyrazol-1-yl)acetyl]-3,9-diazaspiro[5.5]undecan-3-yl]acetamide
4-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1,3λ6,4-oxathiazinane-3,3-dione
1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
5-({3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}methyl)-N-methyl-1,2,4-oxadiazole-3-carboxamide
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-2-(trimethyl-1H-pyrazol-1-yl)acetamide
1-[2-(2,6-dimethoxyphenoxy)ethyl]-3-methyl-1,2-dihydroquinoxalin-2-one
2-(furan-2-yl)-1-[4-(1H-pyrazol-5-yl)phenyl]-1H-imidazole
3-oxo-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-1,2,3,4-tetrahydroquinoxaline-6-carboxamide
5-ethyl-N4-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]pyrimidine-2,4-diamine
1-[4-(3-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-(1H-1,2,3,4-tetrazol-5-yl)ethan-1-one
2-[4-(1H-imidazol-2-yl)-2-methoxyphenoxy]acetamide
6-[4-(1-cyclopropyl-1H-pyrrole-2-carbonyl)piperazin-1-yl]pyridine-3-carbonitrile
8-[(4-hydroxyphenyl)methyl]-1-(2-phenylethyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]-5-[3-(trifluoromethyl)phenyl]pyrimidine
2-{2-methyl-6-[3-(pyridine-2-carbonyl)piperidin-1-yl]pyrimidin-4-yl}ethan-1-amine
N-methyl-N-(2-phenylethyl)-1-(thiophen-3-ylmethyl)piperidin-3-amine
2-[3-(2,5-difluorobenzoyl)piperidin-1-yl]pyridine-3-carbonitrile
1-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-3-(1,2,3-thiadiazol-5-yl)urea
5-(4-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperazin-1-yl)-2,3-dihydropyridazin-3-one
4-[(2,3-dimethyl-1H-indol-7-yl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
3-(dimethyl-1,2-oxazol-4-yl)-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-4-ylmethyl)propanamide
(2S,4R)-4-amino-N,N-diethyl-1-[5-(trifluoromethyl)pyridin-2-yl]pyrrolidine-2-carboxamide
2-[(1,1-dioxo-1λ6-thiolan-3-yl)(methyl)amino]-N-ethyl-N-(2-methylprop-2-en-1-yl)acetamide
1-[benzyl(methyl)amino]-3-[2-methoxy-5-({[3-(methylsulfanyl)propyl]amino}methyl)phenoxy]propan-2-ol
4-{1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]piperidine-4-carbonyl}piperazin-2-one
2-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-1-(6-methyl-1,2,3,4-tetrahydroquinolin-1-yl)ethan-1-one
N-[1-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]-2-(2,4-dichlorophenoxy)acetamide
(3S,4S)-1-[2-(2-methyl-1H-imidazol-1-yl)acetyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
{4-[1-ethyl-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]phenyl}methanol
1-(3-methylpiperidin-1-yl)-3-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}propan-1-one
(2S,4S)-1-[(4-chlorophenyl)methyl]-N-(2-methoxyethyl)-4-{[(3-methylphenyl)methyl]amino}pyrrolidine-2-carboxamide
3-(dimethyl-1H-1,2,4-triazol-1-yl)-N,2-dimethyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
1-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]-N-(pyridin-2-ylmethyl)piperazine-2-carboxamide
7-(2-{[(2-methyl-1,3-thiazol-4-yl)methyl]amino}propoxy)-2H-chromen-2-one
2-[4-({[1-(furan-2-yl)ethyl](methyl)amino}methyl)phenyl]-6-(pyridin-4-yl)-3,4-dihydropyrimidin-4-one
5-(4-methoxyphenyl)-N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H-pyrazole-3-carboxamide
4-(1-butyl-1H-imidazol-2-yl)-1-(4-fluoro-3-methoxybenzoyl)piperidine
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-2-fluoro-5-sulfamoylbenzamide
1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-4-(pyridin-3-ylmethyl)-1,4-diazepane
5-[3-(1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-1-cyclopentyl-4-oxo-N-(prop-2-en-1-yl)-1,4-dihydropyridine-3-carboxamide
1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]-4-(pyridin-4-ylmethyl)piperazine
5-(2-{2-[2-(ethylamino)pyrimidin-5-yl]-1H-imidazol-1-yl}ethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
[(2-chloro-4-fluorophenyl)methyl]({[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl})methylamine
2-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-4-methylpyrimidine
N'1-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}cyclopropane-1,1-dicarboxamide