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N-[4-({[1-(pyridin-4-yl)propan-2-yl]carbamoyl}methyl)phenyl]butanamide
N-{2-[(5-methyl-2-phenyl-1H-imidazol-4-yl)formamido]ethyl}acetamide
2-(cyclopropylmethyl)-8-(6-oxo-1,6-dihydropyrimidine-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[1-(carbamoylmethyl)piperidin-4-yl]-4-hydroxy-2-(phenoxymethyl)pyrimidine-5-carboxamide
5-[3-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-4-ethyl-1,3-thiazol-2-amine
dimethyl[(4-methyl-5-{1-[3-(trifluoromethyl)pyridin-2-yl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]amine
3-chloro-2-{4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine
2-(3-hydroxyphenyl)-1-[(1S,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
5-[(2E)-2-methylpent-2-en-1-yl]-N-phenyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-{2-[5-(2-methylpropyl)thiophen-2-yl]-1H-imidazol-1-yl}propan-1-ol
N-[2-(4-chlorobenzenesulfonamido)ethyl]-5-methyl-1,2-oxazole-3-carboxamide
1-({1-[(4-methoxy-2,5-dimethylphenyl)methyl]piperidin-3-yl}methyl)-4-methylpiperazine
5-{3-[2-(2,6-difluorophenyl)ethyl]piperidine-1-carbonyl}-2-(propan-2-yl)-3,4-dihydropyrimidin-4-one
(4aR,7aS)-4-[2-(4-fluorophenoxy)ethyl]-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
N-[(2,5-difluorophenyl)methyl]-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-{[2,4-bis(prop-2-en-1-yloxy)phenyl]methyl}-4-(1H-imidazol-1-ylmethyl)piperidin-4-ol
(1R,2S)-2-({5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)cyclopentan-1-ol
[(3S,5S)-1-[(2-aminopyridin-3-yl)methyl]-5-[(4-methyl-1,4-diazepan-1-yl)methyl]piperidin-3-yl]methanol
7-chloro-3,5-dimethyl-N-[2-(methylsulfanyl)ethyl]-1-benzofuran-2-carboxamide
(2S,4R)-4-(benzylamino)-1-(2,3-dihydro-1H-inden-2-yl)-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
(1S,5R)-3-[(4-fluorophenyl)methyl]-6-(1H-imidazol-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-(furan-2-ylmethyl)-3-(1,2-oxazinan-2-yl)-N-(pyridin-4-ylmethyl)propanamide
[(3R,4S)-1-[(1-ethyl-1H-indol-4-yl)methyl]-4-[(4-ethylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
2-{3-[(1S,4S)-2-azabicyclo[2.2.1]heptan-2-ylmethyl]-6-chloroimidazo[1,2-a]pyridine-2-carbonyl}-1,2,3,4-tetrahydroisoquinoline
2-ethoxy-5-(2-{[(3-methylpyridin-2-yl)methyl]amino}pyrimidin-4-yl)benzoic acid
1-[3-(1H-imidazol-1-yl)propyl]-4-(4-methoxy-2,3-dimethylphenyl)-1H-1,2,3-triazole
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-{[methyl(2-methylpropyl)amino]methyl}piperidin-2-one
3-[2-(4-cyclopentylpiperazin-1-yl)-2-oxoethyl]-4-[(2-fluorophenyl)methyl]piperazin-2-one
1-(4-{8-methyl-9-oxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carbonyl}phenyl)pyrrolidin-2-one
4-(1H-imidazol-2-yl)-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}piperidine
7-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)-3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]acetamide
2-(furan-3-yl)-5,8-dimethoxy-4-methylquinoline
5-(2H-1,3-benzodioxol-5-ylmethyl)-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
N-[(2,4-dimethoxyphenyl)methyl]-3-[1-(3-phenylpropyl)piperidin-3-yl]propanamide
(4aS,7aR)-1-(4-fluorobenzoyl)-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4,4,4-trifluoro-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]butanamide
1-[4-(4-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}piperazin-1-yl)phenyl]ethan-1-one
7-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-2-oxa-7-azaspiro[4.5]decan-8-one
(1R,2R)-2-[3-(ethoxymethyl)-5-{imidazo[2,1-b][1,3]thiazol-6-yl}-1H-1,2,4-triazol-1-yl]cyclohexan-1-ol
2-(2-methoxy-4-methylphenoxymethyl)-N-methyl-N-[(3-methylpyridin-4-yl)methyl]-1,3-oxazole-4-carboxamide
{1-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]piperidin-4-yl}(pyridin-2-yl)methanol
1-[(3-methylphenyl)methyl]-4-{4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carbonyl}piperazin-2-one
9-(cyclopropylmethyl)-1-methyl-4-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
4-{[(3-methoxyphenyl)methyl]amino}-N,5-dimethyl-N-(oxolan-3-yl)thieno[2,3-d]pyrimidine-6-carboxamide
N4-(2-methoxyethyl)-N1,N1-dimethyl-N4-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidine-1,4-dicarboxamide
N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carboxamide
1-{1-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]piperidin-3-yl}pyrrolidin-2-one
{2-[3-(3-methoxyphenoxymethyl)piperidin-1-yl]-2-oxoethyl}urea
1-cyclopentyl-N-ethyl-4-oxo-5-[4-(thiophen-2-ylmethyl)piperazine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide