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9-benzoyl-4-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-1-methyl-1,4,9-triazaspiro[5.5]undecane
5-chloro-2-methyl-6-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyrimidin-4-ol
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-1H-imidazole-2-carboxamide
N-[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-2-oxo-2,3-dihydro-1H-imidazole-4-carboxamide
N-[2-(7-methyl-1H-indol-3-yl)ethyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
(4aS,8aR)-6-(4-amino-5-methylpyrimidin-2-yl)-1-(piperidin-4-ylmethyl)-decahydro-1,6-naphthyridin-2-one
7-(4-fluorophenyl)-2-[1-(2-methoxyethyl)-1H-imidazol-5-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
6-{1-[(1-methyl-5-phenyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-3,4-dihydropyrimidin-4-one
1-{2-[(3S,4R)-4-hydroxy-4-methyl-3-(2-methylpropyl)piperidin-1-yl]-2-oxoethyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-{2-[7-(thiophen-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}cyclohexanecarboxamide
2-(2,5-dioxoimidazolidin-4-yl)-N-{2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]ethyl}acetamide
4-ethyl-1-[2-(4-phenylpiperazin-1-yl)ethyl]-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{1'-[4-(dimethylamino)benzoyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
9-(5-ethyl-2-methylpyrimidin-4-yl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
N-[(3S,4R)-4-(propan-2-yl)-1-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]pyrrolidin-3-yl]acetamide
2-methyl-4-(4-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)-5-propylpyrimidine
5-{[1-butyl-3-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}imidazolidine-2,4-dione
4-{2,2-dimethyl-3-[4-(5-methylpyrimidin-4-yl)piperidin-1-yl]propyl}morpholine
1-(2,2-dimethylpropyl)-4-{[6-(propan-2-yl)-2-(trifluoromethyl)pyrimidin-4-yl]amino}pyrrolidin-2-one
2-[2-(trifluoromethoxy)phenyl]pyridine-3-carbonitrile
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-2-(piperidin-1-yl)acetamide
3-[(3-amino-1H-1,2,4-triazol-5-yl)formamido]-N-(4-methylphenyl)propanamide
N-(2-methoxyethyl)-2-(1-methylpiperidin-2-yl)-N-(naphthalen-1-ylmethyl)acetamide
2,6-diamino-4-(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)-5,6,7,8-tetrahydroquinoline-3-carbonitrile
(2,1,3-benzoxadiazol-4-ylmethyl)(2-methoxyethyl)({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)amine
ethyl 3-[(4-fluorophenyl)methyl]-1-(4-oxo-4-phenylbutanoyl)piperidine-3-carboxylate
1-({3-[(dimethylamino)methyl]phenyl}methyl)-3-(3-methyl-1,2,4-thiadiazol-5-yl)urea
3-(3-methoxyphenyl)-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(cyclohexylmethyl)-3-hydroxy-3-(1,2-oxazolidin-2-ylmethyl)piperidin-2-one
ethyl 3-[(3-chlorophenyl)methyl]-1-(1,3-thiazole-5-carbonyl)piperidine-3-carboxylate
N-(5-methoxy-2-methylphenyl)-3-oxopiperazine-1-carboxamide
3-[(2-methylphenyl)methyl]-1-(1,4-oxazepan-6-ylmethyl)urea
1-{[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-methoxypiperidine
1-[3-(4-{[methyl(naphthalen-1-ylmethyl)amino]methyl}phenoxymethyl)piperidin-1-yl]-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
7-(4-chlorophenyl)-2-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-yl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
5-{1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}-3-[2-(1-methylpyrrolidin-2-yl)ethyl]-5-propylimidazolidine-2,4-dione
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2-ethylpyridine-4-carboxamide
N-[4-(3-methoxyphenyl)phenyl]-1-(3-methylbut-2-enoyl)piperidine-3-carboxamide
5-(4-cyclohexylpiperazin-1-yl)-1-propyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
(2R,6S)-4-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-2,6-dimethylmorpholine
N-[(2,3-dimethoxyphenyl)methyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
3-(2-methoxyethyl)-1-(2,2,2-trifluoroethyl)-5-{1,3,6-trimethyl-1H-pyrazolo[3,4-b]pyridin-4-yl}-1H-1,2,4-triazole
2-[8-(butan-2-yl)-1-ethyl-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl]acetamide
5-({methyl[(1-methylpiperidin-3-yl)methyl]amino}methyl)-2-oxo-2,3-dihydro-1H-imidazole-4-carboxylic acid
3-{[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}benzonitrile
N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-amine
2,5-dimethyl-N-(3-phenylprop-2-yn-1-yl)-N-propyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
N-[2-(4,5,6,7-tetrahydro-1-benzothiophen-3-yl)ethyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-[(2-aminopyridin-3-yl)methyl]-3-(azetidine-1-carbonyl)benzene-1-sulfonamide