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N-(1,3-benzothiazol-2-yl)-3-[4-hydroxy-4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]propanamide
N-methyl-6-oxo-1-[2-(pyridin-2-yl)ethyl]-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)piperidine-3-carboxamide
4-(1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1H-imidazol-2-yl)pyridine
2-(4-{[2-(trifluoromethoxy)phenyl]methyl}morpholin-2-yl)ethan-1-amine
5-(4-methylnaphthalen-1-yl)pyrimidin-2-amine
methyl N-{2-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-oxoethyl}carbamate
4-(3-chlorophenyl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}pyrimidin-2-amine
N-[2-(dimethylsulfamoyl)ethyl]imidazo[1,2-a]pyridine-2-carboxamide
[1-({2-[(2-chloro-6-fluorophenyl)methoxy]phenyl}methyl)pyrrolidin-3-yl]methanamine
2-(2-hydroxyethyl)-9-{2-[4-(hydroxymethyl)phenyl]acetyl}-2,9-diazaspiro[5.5]undecan-3-one
N-[(5-amino-1,3,4-thiadiazol-2-yl)(phenyl)methyl]-1-phenyl-1H-1,2,3-triazole-4-carboxamide
methyl({[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}){[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}amine
4-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-2-ethyl-1-(propan-2-yl)piperazine
N-cyclopropyl-3-{5-[(3-methoxyphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
5-methyl-N-[2-(phenylsulfanyl)ethyl]-1-propyl-1H-pyrazole-4-carboxamide
3-(4-hydroxyphenyl)-N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-1H-pyrazole-5-carboxamide
2-(2-chloro-4-fluorophenoxymethyl)-N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-1,3-oxazole-4-carboxamide
N-(pyridin-3-yl)-5-(quinolin-8-yl)furan-2-carboxamide
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-{[methyl(thiophen-2-ylmethyl)amino]methyl}piperidin-2-one
6-[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]pyridine-3-carbonitrile
[1-({2-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)azepan-2-yl]methanol
7-(5-methylthiophen-2-yl)-4-[(2R)-pyrrolidine-2-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[2-(4-methoxyphenyl)phenyl]-3-(5-oxo-1-propylpyrrolidin-3-yl)urea
5-ethyl-N4-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-6-methylpyrimidine-2,4-diamine
4-(4-chlorophenyl)-1-[(2S)-2-(morpholine-4-carbonyl)pyrrolidin-1-yl]butan-1-one
3-(3-hydroxy-3-methylbutyl)-N-methyl-N-[(3-methylpyridin-2-yl)methyl]benzamide
(2S,4S)-4-amino-1-(2,8-dimethylquinoline-3-carbonyl)-N-methylpyrrolidine-2-carboxamide
3-[5-(cyclopropanesulfonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]-1-(pyrrolidin-1-yl)propan-1-one
3-ethyl-3-(hydroxymethyl)-N-(3-phenyl-1,2,4-thiadiazol-5-yl)piperidine-1-carboxamide
1-[4-(dimethylamino)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-hydroxypropan-1-one
N-[2-(dimethylamino)ethyl]-6-(methoxymethyl)-N,1-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-methyl-1-[4-({[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amino}methyl)piperidin-1-yl]propan-1-one
3-({4-[(2,3-dihydro-1H-inden-5-yloxy)methyl]piperidin-1-yl}methyl)piperidin-3-ol
N-[2-(1-methylpiperidin-3-yl)ethyl]-2-(pyridin-3-yloxy)acetamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N-methylbenzamide
1-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidin-3-yl)-4-(2-methoxyphenyl)piperazine
N'-cyclopentyl-N-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}butanediamide
1-ethyl-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-N,5-dimethyl-1H-pyrazole-4-carboxamide
1-(propan-2-yl)-4-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}piperidine
(2H-1,3-benzodioxol-5-ylmethyl)(methyl)({4-methyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)amine
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)piperidine-1-carboxamide
3-(azepane-1-carbonyl)-1-ethyl-N-[(3-methoxyphenyl)methyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
(4aS,8aR)-1-(2-aminoethyl)-6-[(8-fluoroquinolin-2-yl)methyl]-decahydro-1,6-naphthyridin-2-one
4-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}morpholine
1-[2-(4-chloro-2-methylphenoxy)ethyl]-4-(1-methylpyrrolidine-3-carbonyl)piperazine
5-(1H-pyrazol-5-yl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}furan-2-sulfonamide
4-methoxy-N-{1-[1-(3-methylbut-2-enoyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
N,5,7-trimethyl-N-(3-methylbutyl)pyrido[2,3-d]pyrimidin-4-amine
(1S,4S)-2-(3-chlorophenyl)-5-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-2,5-diazabicyclo[2.2.1]heptan-3-one
4-methyl-2-(4-methyl-3-phenylpiperazin-1-yl)pyrimidine