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4-[(3-fluorophenyl)methyl]-11-{[3-(1H-imidazol-1-yl)propyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-[3-(dimethylamino)pyrrolidin-1-yl]-N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]acetamide
6-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
5-{[(5-fluoro-2-methylphenyl)methyl]amino}-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
1-({5-[(3-fluoro-2-methylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,3-dimethylurea
1-(3-cyano-4-methoxyphenyl)-3-{3-[cyclopentyl(methyl)amino]propyl}urea
2-[7-(cyclobutylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]acetic acid
1-[1-(4-fluorobenzoyl)piperidin-3-yl]-3-phenylpropan-1-one
5-methyl-N-[(6-methylquinolin-5-yl)methyl]pyrimidin-2-amine
6-{4-[(4-cyclopentyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}-1H-indole
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}pyrazolo[1,5-a]pyrimidine-2-carboxamide
methyl 4-(4-ethyl-5-methylpyrimidin-2-yl)piperazine-1-carboxylate
N-[4-({[2-(dimethylamino)ethyl](oxolan-2-ylmethyl)carbamoyl}methyl)phenyl]butanamide
3-[({[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}amino)methyl]pyrrolidin-3-ol
4-[2-(1-benzylpiperidin-4-yl)acetyl]piperazine-2-carboxylic acid
5-(methoxymethyl)-N-[1-(3-methylbutan-2-yl)-1H-pyrazol-5-yl]furan-2-carboxamide
2-fluoro-N-{3-[2-(4-fluorophenyl)-3-oxopiperazin-1-yl]-3-oxopropyl}benzamide
1-ethyl-N-[2-(4-fluorobenzenesulfonyl)ethyl]-5-oxopyrrolidine-3-carboxamide
2,5,6-trimethyl-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}pyrimidin-4-amine
4-{2-[(5-fluoropyrimidin-2-yl)oxy]hex-5-en-1-yl}thiomorpholine
2-methyl-9-(quinolin-6-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
ethyl({[2-(naphthalen-2-yl)pyrimidin-5-yl]methyl})(pyridin-4-ylmethyl)amine
3-(3-fluorophenyl)-4-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]piperazin-2-one
1-{[1-(2,3-dihydro-1H-inden-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-N,N-dimethylpyrrolidin-3-amine
N,N-dimethyl-5-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
3-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]benzonitrile
dimethyl(2-{[(2-methylphenyl)methyl](pyridin-3-ylmethyl)amino}ethyl)amine
1-[5-(2-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
N,5-dimethyl-N-[2-(1H-pyrazol-4-yl)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-N-[2-(4-fluorophenyl)ethyl]-5-(methoxymethyl)-1H-pyrazole-4-carboxamide
(1S,5R)-N-benzyl-7-oxo-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
(1R,6S)-3-[(3-ethenylphenyl)methyl]-9-methyl-3,9-diazabicyclo[4.2.1]nonane
N-[3-(1,3-thiazol-4-yl)phenyl]-1-[2-(4H-1,2,4-triazol-4-yl)ethyl]piperidine-4-carboxamide
8-(3-fluoropropyl)-2-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
9-(3-chloro-4-methoxybenzoyl)-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
(4-{[1-(naphthalene-2-carbonyl)pyrrolidin-3-yl]methyl}phenyl)methanol
5-(3,5-dimethyl-1H-indole-2-carbonyl)-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
1-[4-(2-fluorophenyl)piperazin-1-yl]-2-[2-({methyl[1-(1,3-thiazol-2-yl)ethyl]amino}methyl)-4-phenylphenoxy]ethan-1-one
4-(2-methylbutan-2-yl)-N-(1,4-oxazepan-6-ylmethyl)benzene-1-sulfonamide
1-[3-(4-methoxyphenyl)-1H-pyrazole-5-carbonyl]-4-[2-(1H-pyrrol-1-yl)ethyl]piperazine
(4aS,7aR)-1-(1H-imidazol-4-ylmethyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-oxo-4H-chromene-2-carboxamide
8-[4-(4-methylphenyl)benzoyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]-N-[2-(pyrrolidin-1-yl)ethyl]piperidine-3-carboxamide
4-{5-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-yl]-1-[(3-methylphenyl)methyl]-1H-1,2,4-triazol-3-yl}benzamide
methyl 5-{[(2E)-2-methylbut-2-en-1-yl]amino}-3-(oxolane-3-amido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-ethyl-3-{1-[2-(4-methanesulfonylphenyl)acetyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[1-(pyrazin-2-yl)propan-2-yl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
2-[1-(2-chlorophenyl)-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(furan-3-ylmethyl)acetamide
(2R,6R)-4-[2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid