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6-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]pyridine-3-carboxamide
({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)[(1-ethyl-1H-pyrazol-4-yl)methyl]methylamine
2-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-1-(morpholin-4-yl)ethan-1-one
5-[4-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]-1-[2-(pyridin-2-yl)ethyl]piperidin-2-one
(4aR,8aR)-2-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-7-(pyrrolidine-1-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
4-[1-(4-{1H-[1,2,3]triazolo[4,5-b]pyridin-6-yl}phenyl)ethyl]morpholine
(2S,4R)-1-[(3-chlorophenyl)methyl]-4-[(2,3-dihydro-1H-inden-2-yl)amino]-N-[2-(2-fluorophenyl)ethyl]pyrrolidine-2-carboxamide
N-[(2-ethoxyphenyl)methyl]-4,4,4-trifluoro-N-(prop-2-en-1-yl)butanamide
N-(4-hexylphenyl)-3-(hydroxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carboxamide
4-[1-(6-oxo-1,6-dihydropyrimidine-5-carbonyl)piperidin-3-yl]benzoic acid
N-{2-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}oxolane-2-carboxamide
2-cyclopropyl-4-methyl-N-[(3R,4S)-1-[(methylcarbamoyl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]pyrimidine-5-carboxamide
4-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]pyridine-2-carboxylic acid
4,4-difluoro-N-(3-phenyl-1,2,4-thiadiazol-5-yl)piperidine-1-carboxamide
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
3-(3,4-dimethoxyphenyl)-1-{[1-(propan-2-yl)piperidin-3-yl]methyl}urea
2-(2-oxo-1,3-oxazolidin-3-yl)-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}acetamide
1-(carbamoylmethyl)-N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]piperidine-3-carboxamide
7-[3-(3-methoxyquinoxalin-2-yl)propanoyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
2-{4-[2-(4-chlorophenoxy)ethyl]phenyl}acetamide
1-[2-({[4-ethoxy-3-(prop-2-en-1-yl)phenyl]methyl}amino)ethyl]piperidine-3-carboxamide
3-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-1-[4-(3-methyl-2-oxoimidazolidin-1-yl)phenyl]urea
4-[2-(2-chlorophenyl)ethyl]-11-{[3-(pyrrolidin-1-yl)propyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-[(5-methylthiophen-2-yl)methyl]piperazin-2-yl}ethan-1-ol
7-chloro-4-methyl-2-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]quinoline
1-(cyclopropylmethyl)-2-oxo-3-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
1-[2-(4-chlorophenyl)ethyl]-6-oxo-N-(pyridin-4-ylmethyl)piperidine-3-carboxamide
N-{[7-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)propanamide
N-[2-(3-chlorophenoxy)ethyl]-6-(methoxymethyl)-N-methylpyridine-2-carboxamide
1-(cyclohexylmethyl)-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-[2-(1,3-thiazol-4-yl)ethyl]azepan-4-amine
N-[(1S)-1-[1-(2,3-dihydro-1H-inden-5-yl)-3-methyl-1H-1,2,4-triazol-5-yl]-2-(1H-imidazol-4-yl)ethyl]acetamide
4-(methoxymethyl)-N,5-dimethyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,2-oxazole-3-carboxamide
N-{2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-1-(pyridin-2-ylmethyl)piperidin-4-amine
2-[({1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-2-oxopiperidin-3-yl}methyl)amino]-N,N-dimethylacetamide
N,N-dimethyl-2-[(4,4,4-trifluorobutanamido)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
N-[2-(piperidin-1-yl)ethyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
5-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]pyridine-2,4-diol
3-cyclopropyl-N-(2-methylpropyl)-1-phenyl-1H-1,2,4-triazole-5-carboxamide
N-(1-hydroxybutan-2-yl)-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
1-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]-4-(1-methyl-1H-imidazol-2-yl)piperidine
N-[(3R,5S)-5-(diethylcarbamoyl)-1-propanoylpyrrolidin-3-yl]-2-(methylamino)pyrimidine-5-carboxamide
4-hydroxy-2-({methyl[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]amino}methyl)quinoline-6-carboxamide
methyl 1-[(3S,5S)-5-{[2-(4-fluorophenyl)ethyl]carbamoyl}-1-[(6-methylpyridin-2-yl)methyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
5-fluoro-2-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}pyrimidine
5-methoxy-2-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]-4H-pyran-4-one
{1-[(1-pentylpiperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}(phenyl)methanol
9-{7-methylimidazo[1,2-a]pyridine-2-carbonyl}-1-oxa-9-azaspiro[5.5]undecan-5-ol
[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl][(5-methylpyrazin-2-yl)methyl]amine
8-{[3-(furan-2-yl)phenyl]methyl}-1-methyl-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione