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N-[3-({3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}sulfonyl)phenyl]acetamide
ethyl 1-[5-(1H-imidazol-2-yl)thiophene-2-carbonyl]-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylate
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(1-methylcyclopropyl)propan-1-one
4-{[6-(dimethylamino)pyridin-3-yl]methyl}-1-(4-methoxyphenyl)-3-methylpiperazin-2-one
benzyl(cyclopropylmethyl){[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl}amine
N-[(3S,5S)-5-(diethylcarbamoyl)-1-(1H-imidazol-4-ylmethyl)pyrrolidin-3-yl]-1-methyl-1H-pyrrole-2-carboxamide
N-({1-[(2-methylphenyl)methyl]pyrrolidin-3-yl}methyl)-4-(1H-pyrazol-4-yl)butanamide
4-benzyl-3-(1-{thieno[3,2-d]pyrimidin-4-yl}piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-butyl-4-ethyl-2-methyl-N-(pyridin-4-ylmethyl)-1,3-thiazole-5-carboxamide
(1S,5R)-6-(3-fluorobenzenesulfonyl)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-(2,1,3-benzoxadiazol-5-ylmethyl)-2-(2-ethyl-1H-1,3-benzodiazol-1-yl)butanamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-(1H-1,2,4-triazol-1-yl)benzamide
2-ethyl-4-({4-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)morpholine
2-amino-N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-2-methylpropanamide
1-ethyl-N-[3-(3-ethylphenoxy)propyl]-N,5-dimethyl-1H-pyrazole-4-carboxamide
N-(2-methoxyethyl)-N-methyl-1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carboxamide
N-[(2-propyl-1,3-thiazol-4-yl)methyl]-4-(pyridin-2-yl)pyrimidin-2-amine
3-{1-[(carboxymethyl)carbamoyl]piperidin-3-yl}benzoic acid
2-[1-(2-chloro-6-methylbenzenesulfonyl)azetidin-3-yl]pyridine
1-methyl-N-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
N-{[(3S,4S)-1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-3-hydroxypiperidin-4-yl]methyl}cyclopropanecarboxamide
N-[(2,5-difluorophenyl)methyl]-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[4-(2,2-dimethoxyethyl)piperazin-1-yl]-2-(methylsulfanyl)ethan-1-one
1-[1-(2-oxo-2H-chromene-3-carbonyl)piperidin-4-yl]-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
(2S,4R)-4-amino-N-(furan-2-ylmethyl)-N-[2-(morpholin-4-yl)ethyl]pyrrolidine-2-carboxamide
2-[6-hydroxy-4-(3-methylbutanoyl)-1,4-diazepan-1-yl]pyridine-4-carbonitrile
8-[2-(methylamino)pyrimidine-5-carbonyl]-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
methyl[2-(morpholin-4-yl)ethyl]({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)amine
1-{3-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]-3-oxopropyl}-6-methyl-1,2-dihydropyridin-2-one
4-{[3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]methyl}-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
1'-{2-oxo-1H,2H,5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
2-[4-(hydroxymethyl)phenyl]-4,6-dimethylpyridine-3-carbonitrile
N-[(3S,4R)-1-[(2-aminopyridin-3-yl)methyl]-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
N-(2-methoxyethyl)-2-(pyrrolidin-3-yl)-N-(thiophen-3-ylmethyl)acetamide
ethyl 3-(2-phenoxyethyl)-1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidine-3-carboxylate
1-[(3R,4S)-3-amino-4-propylpyrrolidin-1-yl]-2-(3-methoxyphenyl)ethan-1-one
ethyl 2-[1-(3-methanesulfonylbenzoyl)piperidin-2-yl]acetate
(1R,3S)-1-hydroxy-3-(2-hydroxyethoxy)-N-[(2-methylphenyl)methyl]-7-azaspiro[3.5]nonane-7-carboxamide
({6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)[5-(morpholin-4-yl)pentyl]amine
N-[2-(4-chlorophenyl)ethyl]-2-[4-(propan-2-yl)morpholin-2-yl]acetamide
(3S,4S)-1-(cyclopropylmethyl)-4-(naphthalen-2-yl)piperidin-3-ol
2-fluoro-N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}-5-sulfamoylbenzamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N-methyl-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
1-{2-amino-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-5-yl}-3-(1H-indol-3-yl)propan-1-one
N-methyl-2-(N-phenylmethanesulfonamido)-N-(prop-2-yn-1-yl)propanamide
2-[2-(2-methylpropyl)-3-oxo-2,8-diazaspiro[4.5]decan-8-yl]pyridine-3-carboxamide
2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-[1-(pyridin-2-yl)propan-2-yl]acetamide
1-methyl-3-{2-oxa-7-azaspiro[4.5]decane-7-carbonyl}-1,2-dihydroquinoxalin-2-one
N-{2-[1-(1H-imidazol-4-ylmethyl)piperidin-3-yl]ethyl}-2,2-dimethylpropanamide
3-(2H-1,3-benzodioxol-5-yl)-N-[3-(2-methyl-1H-imidazol-1-yl)propyl]-3-phenylpropanamide