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7-[3-(2-ethoxyphenyl)propyl]-2-oxa-7-azaspiro[4.5]decan-8-one
2-methyl-6-{3-[1-(pyridin-3-ylmethyl)piperidin-4-yl]pyrrolidine-1-carbonyl}pyridine
3-hydroxy-3-({methyl[2-(1H-pyrazol-4-yl)ethyl]amino}methyl)-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
2-(1H-pyrazol-1-yl)-N-{2-[(trifluoromethyl)sulfanyl]ethyl}butanamide
5-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine-2-carbonitrile
1-[3-(1-methyl-5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]cyclopropane-1-carboxamide
4-{5-[2-(1H-imidazol-2-yl)phenyl]-1,2,4-oxadiazol-3-yl}pyridine
1-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-ethyl-4-{[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]methyl}-1H-pyrrole-2-carbonitrile
2-[4-({2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}methyl)phenyl]ethan-1-amine
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-5-(oxolan-2-yl)thiophene-2-carboxamide
9-(2-methoxy-4-methylbenzoyl)-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
(2S,4R)-4-amino-N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]pyrrolidine-2-carboxamide
4-(4-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carbonyl}phenyl)-2-methylbut-3-yn-2-ol
2-(ethylsulfanyl)-5-{1-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1H-imidazol-2-yl}pyrimidine
N-[(3-methylphenyl)methyl]-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
1-[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidin-1-yl]-2-cyclobutylethan-1-one
3-(1-benzyl-1H-imidazol-2-yl)-1-[3-(4-methyl-1H-pyrazol-1-yl)propyl]piperidine
methyl 1-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-3-(2-methylpropyl)-2-oxo-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylate
3-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)-1H,2H,5H,6H,7H-cyclopenta[b]pyridin-2-one
4-[2-(1H-imidazol-1-ylmethyl)pyrrolidine-1-carbonyl]-6-methyl-2-(1H-pyrazol-4-yl)quinoline
2-[3-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]pyrazine
N-[2-(3,4-dimethoxyphenyl)ethyl]-5-(oxolan-2-yl)thiophene-2-carboxamide
{2-[(2H-1,3-benzodioxol-4-ylmethyl)(thiophen-3-ylmethyl)amino]ethyl}dimethylamine
N-{[5-(2-amino-6-tert-butyl-3-cyanopyridin-4-yl)furan-2-yl]methyl}-N-methylmethanesulfonamide
(2R)-2-{[5-(2-fluorophenoxymethyl)-1H-pyrazol-3-yl]formamido}propanamide
1-[2-(3-phenylpropyl)morpholin-4-yl]-3-(pyrazin-2-yl)propan-1-one
3-[1-(3-chloropyridin-2-yl)piperidin-4-yl]-N-[(1-ethylpyrrolidin-2-yl)methyl]propanamide
5-[4-(2,6-dimethylpyridin-4-yl)piperazine-1-carbonyl]-2-methyl-1H-1,3-benzodiazole
4-ethoxy-N-[(5-methylpyrazin-2-yl)methyl]pyrimidin-2-amine
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]piperidin-2-one
2-{[1-(2-ethoxyethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl]formamido}acetamide
2-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-6,7-dimethoxy-1-methyl-1,2,3,4-tetrahydroisoquinoline
methyl (2S,4S,5R)-2-ethyl-5-(4-fluorophenyl)-1-methyl-4-{[(1r,4r)-4-hydroxycyclohexyl]carbamoyl}pyrrolidine-2-carboxylate
(3R)-3,4,4-trimethyl-1-(5-methyl-2H-1,2,3-triazole-4-carbonyl)pyrrolidin-3-ol
5-(naphthalen-1-yl)-N-[1-(pyrazin-2-yl)propan-2-yl]-1,2,4-triazin-3-amine
6-(benzyloxy)-1-cyclohexyl-4-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-1,4-diazepan-2-one
3-methyl-N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)-5,6-dihydro-1,4-dioxine-2-carboxamide
1-(2,1,3-benzoxadiazol-4-ylmethyl)-4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-5-one
2-(dimethylamino)-2-(2-methylphenyl)-N-[(1-propyl-1H-pyrazol-4-yl)methyl]acetamide
N-cyclohexyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-5-(morpholin-4-ylmethyl)furan-3-carboxamide
2-methyl-2-({1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidin-3-yl}formamido)propanamide
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]oxan-4-amine
N-[(3R,5S)-5-(ethylcarbamoyl)-1-(2-phenylethyl)pyrrolidin-3-yl]-2-methyl-1H-pyrrole-3-carboxamide
(3S,4R)-N,N-dimethyl-4-(propan-2-yl)-1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-3-amine
(2S)-N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]pyrrolidine-2-carboxamide
1-[1-(2-hydroxyacetyl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-3-carboxamide
1-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-9-yl]-2-(pyridin-4-yl)ethan-1-one
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)morpholine-2-carboxamide