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2-[1-(3,5-difluoropyridine-2-carbonyl)piperidin-4-yl]-1,2,3,4-tetrahydroisoquinoline
5-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-1-ethyl-3-methyl-1H-pyrazole
4-(1H-imidazol-1-yl)-1-[4-(3-methoxybenzoyl)piperazin-1-yl]butan-1-one
5-{3-[(2H-1,3-benzodioxol-5-yl)amino]piperidine-1-carbonyl}-2-(propan-2-yl)-3,4-dihydropyrimidin-4-one
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
methyl (2S)-1-{2-[4-(4-{[2-(furan-2-yl)ethyl]amino}piperidin-1-yl)phenyl]acetyl}pyrrolidine-2-carboxylate
N-methyl-1-(1-methylpiperidin-4-yl)-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-(1,3-benzothiazol-5-yl)-2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine-1-carboxamide
4-fluoro-N-(3-methoxypropyl)-N-{[6-(2-methylphenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}benzamide
2,2-difluoro-1-[(2R,3R)-2-hydroxy-3-(1H-imidazol-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]propan-1-one
(3R,4R)-1-(5-amino-4-chloro-1H-pyrazole-3-carbonyl)-3-methyl-4-(oxan-4-yl)piperidin-4-ol
(1H-imidazol-2-ylmethyl)[(5-methylthiophen-2-yl)methyl](pyridin-4-ylmethyl)amine
2-{3-methyl-4-[(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]-1H-pyrazol-1-yl}ethan-1-ol
7-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-2-(dimethylamino)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-methyl-2-(morpholin-4-yl)-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-2-(pyridin-3-yl)acetamide
N-ethyl-1-(5-phenyl-1,2,4-oxadiazol-3-yl)-N-(pyridin-4-ylmethyl)piperidin-3-amine
7-fluoro-3-[1-methyl-6-oxo-3-(pyridin-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl]-1,2-dihydroquinolin-2-one
1-[2-(cyclohex-1-en-1-yl)ethyl]-2-(4-methyl-1H-imidazol-5-yl)-1H-imidazole
(3S,4S)-3-[2-(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)-1H-imidazol-1-yl]-4-hydroxy-1λ6-thiolane-1,1-dione
1-(1-methylpiperidin-4-yl)-N-[2-(1,3-thiazol-2-yl)ethyl]piperidine-3-carboxamide
[(8-chloroquinolin-2-yl)methyl](methyl)[(1-methylpyrrolidin-2-yl)methyl]amine
3-(1,3-dihydro-2-benzofuran-5-yl)-1-(oxolan-2-ylmethyl)urea
(2S,4S)-4-cyclobutaneamido-N-[2-(1H-indol-3-yl)ethyl]-1-methylpyrrolidine-2-carboxamide
(2S,4S)-4-[4-(4-methoxyphenyl)-1H-1,2,3-triazol-1-yl]pyrrolidine-2-carboxylic acid
1-[(4-fluoro-3-methoxyphenyl)methyl]-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-4-ol
1-(2-chloroprop-2-en-1-yl)-3-[(cycloheptylamino)methyl]-6,7-dimethoxy-1,2-dihydroquinolin-2-one
6-methyl-2-({[1-(5-methylpyridin-2-yl)ethyl]amino}methyl)quinolin-4-ol
2-(dimethylamino)-N-(5-oxo-1-propylpyrrolidin-3-yl)-2,3-dihydro-1H-indene-2-carboxamide
N-ethyl-3-[(3R)-3-hydroxypiperidin-1-yl]-N-phenylpropanamide
2-(dimethylamino)-4-methyl-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}pyrimidine-5-carboxamide
2-ethoxy-1-[(3S,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidin-1-yl]ethan-1-one
8-(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-[2-(4-ethyl-1,3-thiazol-2-yl)ethyl]-1-(6-fluoropyridin-3-yl)urea
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-[1-(propan-2-yl)-1H-pyrrole-2-carbonyl]piperidin-3-yl]propan-1-ol
1-[(4-methylphenyl)methyl]-5-oxo-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}pyrrolidine-3-carboxamide
1-(4-methylphenyl)-4-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperazin-2-one
1-(cyclopropylmethyl)-5-[(2R)-2-phenylbutanoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
(2R)-2-amino-N-ethyl-3-phenyl-N-[(2E)-3-phenylprop-2-en-1-yl]propanamide
1-[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]-2-(2-methyl-1H-imidazol-1-yl)ethan-1-one
1-benzyl-4-oxo-5-(4-phenylpiperidine-1-carbonyl)-N-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
methyl[(1-methylpyrrolidin-2-yl)methyl]{[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}amine
2-{[(1-ethylpiperidin-4-yl)amino]methyl}-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
2-(3-fluorophenyl)-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
6-(2,6-dimethoxyphenyl)-3,4-dihydro-2H-1,4-benzoxazin-3-one
methyl 2-[(cyclohexylmethyl)sulfamoyl]-6-(1,3-thiazole-5-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-(cyclohexylmethyl)-N3,N3-dimethyl-N5-[(2-methylphenyl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
4-[(1S,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carbonyl]-1,2-dihydroisoquinolin-1-one
4-{1-[4-(5-methylfuran-2-yl)benzoyl]piperidin-4-yl}thiomorpholine
N-[1-(4-fluorophenyl)-2-hydroxyethyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
[3-(3-methoxypropyl)-1-(morpholine-4-carbonyl)piperidin-3-yl]methanol