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1-(4-{[2-(1-methylpyrrolidin-2-yl)ethyl]amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
N-methyl-5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-(1,2-oxazol-5-ylmethyl)-1,2-oxazole-3-carboxamide
N1-(3-methanesulfonamidophenyl)piperidine-1,3-dicarboxamide
4-{1-[2-(pyridin-3-yloxy)propyl]-1H-imidazol-2-yl}quinoline
3,5-dimethyl-1-(1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}pyrrolidin-3-yl)-1H-pyrazole
1-{1-[(2-fluoro-4-methoxyphenyl)methyl]pyrrolidin-3-yl}-4-methylpiperazine
6-chloro-N-methyl-N-(thiophen-3-ylmethyl)imidazo[1,2-a]pyridine-2-carboxamide
1-[(3R,4S)-3-amino-4-(4-methoxyphenyl)pyrrolidin-1-yl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
(3S,4S)-4-cyclopropyl-1-(3-fluoro-4-methoxybenzenesulfonyl)pyrrolidine-3-carboxylic acid
1-[2-(3-phenylpyrrolidin-1-yl)ethyl]-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
3-ethoxy-N-ethyl-N-[(2E)-3-phenylprop-2-en-1-yl]propanamide
3-{2-oxo-2-[4-(pyrimidin-2-yloxy)piperidin-1-yl]ethyl}-2,3-dihydro-1H-isoindol-1-one
9-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
2-(4-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperazin-1-yl)-1,3-benzoxazole
5-ethyl-2-methyl-4-[4-(pyridin-4-yl)piperidin-1-yl]pyrimidine
3-[1-(5-carbamoylthiophen-3-yl)-1H-pyrazol-4-yl]benzoic acid
1-methyl-N-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}-1H-1,2,3-benzotriazole-5-carboxamide
1-[1-(oxan-4-yl)piperidin-3-yl]-4-phenylpiperazine
(1-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)(thiophen-2-yl)methanol
2-methoxy-5-{[3-(pyrrolidine-1-carbonyl)piperazin-1-yl]methyl}pyrimidine
2,6,8-trimethyl-4-[2-(pyridin-3-yl)piperidine-1-carbonyl]quinoline
(1R,3S)-7-[3-(difluoromethoxy)benzoyl]-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-1-ol
3-(pentan-2-yl)-8-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(3-{[(3-methylphenyl)methyl]sulfanyl}propyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
1-(cyclopropylmethyl)-5-(isoquinoline-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-2-(trifluoromethyl)pyrimidin-4-amine
5-[methyl(2-phenylethyl)amino]-2-[2-(3-methyl-4H-1,2,4-triazol-4-yl)ethyl]-2,3-dihydropyridazin-3-one
{2-[2-(1-cyclohexanecarbonylpiperidin-4-yl)-1H-imidazol-1-yl]ethyl}dimethylamine
N,2,6-trimethyl-N-[1-(1,2-oxazol-3-yl)ethyl]quinoline-3-carboxamide
(3aR,6aR)-2-acetyl-5-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-ethyl-4-{[methyl({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)amino]methyl}pyrrolidin-2-one
2-(pyridin-3-yl)-1-{3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}ethan-1-one
2-[(3-{[(4-hydroxy-3-methoxyphenyl)methyl]carbamoyl}phenyl)amino]acetic acid
N-{2-[({5-[(dimethylamino)methyl]furan-2-yl}methyl)sulfanyl]ethyl}-1-methylazepane-2-carboxamide
(3R,7S,8aS)-3-methyl-7-{[(3-methylphenyl)methyl]amino}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
(4aR,7aS)-1-acetyl-4-[3-(1H-pyrazol-1-yl)benzoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(2,5-dihydro-1H-pyrrole-2-carbonyl)-4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(pyrazin-2-yl)propanamide
1-[(1R,5R)-6-[(2-butyl-1H-imidazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
4-({[(2-aminopyrimidin-5-yl)methyl](methyl)amino}methyl)-N-(5-methyl-1,3-thiazol-2-yl)benzamide
N-[(3R,4S)-1-(carbamoylmethyl)-4-propylpyrrolidin-3-yl]-2,3-dimethoxybenzamide
N-methyl-2-(1-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}piperidin-4-yl)acetamide
2-[(thiolan-3-yl)amino]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-(4-fluorophenoxymethyl)-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}piperidine
(4aS,8aR)-1-[2-(cyclohex-1-en-1-yl)ethyl]-6-(oxan-4-yl)-decahydro-1,6-naphthyridin-2-one
2-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)-5-methylpyrazine
1-[2-(2-chloro-4-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-4-methylpiperidine
5-ethyl-N-[2-(4-phenylpiperidin-1-yl)ethyl]-1,3,4-oxadiazol-2-amine
1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine
(3S,4S)-4-cyclopropyl-1-[2-(4-methyl-1,4-diazepan-1-yl)acetyl]pyrrolidine-3-carboxylic acid