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5-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
(1S,5R)-3-(oxan-4-yl)-6-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(3R,4S)-4-cyclopropyl-1-[3-(methylsulfanyl)propanoyl]pyrrolidin-3-yl]-2-oxo-2-phenylacetamide
3-(4-oxo-3,4-dihydroquinazolin-3-yl)-N-[4-(pyridin-3-yloxy)phenyl]propanamide
{[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}({[5-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl})amine
1-(2-ethylpyrimidine-5-carbonyl)-4-(hydroxymethyl)azepan-4-ol
(3aR,6aR)-2-(4-hydroxybenzoyl)-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[3-(2-methoxyphenyl)propyl]-1-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
N-cyclohexyl-5-(pyridin-3-yl)furan-2-carboxamide
1-(azocan-1-yl)-3-{5-[methoxy(phenyl)methyl]-1,3,4-oxadiazol-2-yl}propan-1-one
[(1-methyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)[3-(methylsulfanyl)butyl]amine
1-[2-({7-acetyl-2-cyclopropyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)ethyl]imidazolidin-2-one
methyl 4-(2-propyl-1,3-thiazole-4-carbonyl)piperazine-1-carboxylate
1-[2-(2H-1,3-benzodioxol-5-ylmethyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]piperidine-3-carboxamide
(4-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methanol
N-[(5-methylfuran-2-yl)methyl]-5-(morpholin-4-ylmethyl)furan-3-carboxamide
{[(3R,4S)-4-cyclopropyl-1-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]pyrrolidin-3-yl]sulfamoyl}dimethylamine
5-phenyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
1-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(propan-2-yloxy)ethan-1-one
3-[5-(2-methylpyrimidin-4-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-1-(morpholin-4-yl)propan-1-one
6-methyl-2-{2-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]-2-oxoethyl}-2,3-dihydropyridazin-3-one
1-[2-(furan-2-yl)pyrrolidin-1-yl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propan-1-one
2-[8-(3-methylbutyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]pyridine-3-carboxamide
N-(4-methoxyphenyl)-4-{[4-(pyrrolidin-1-ylmethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carboxamide
8-[(3-ethoxy-4-methoxyphenyl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
6-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-N,N-dimethylpyrimidin-4-amine
methyl 3-acetamido-1-[2-(1H-indol-3-yl)ethyl]-5-[(propan-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-(2,3-dimethylphenyl)-5-(pyrrolidine-1-carbonyl)pyridine
2-methoxy-6-{[methyl({[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl})amino]methyl}phenol
3-[(3-benzyl-1H-1,2,4-triazol-5-yl)methyl]-4,6-dimethyl-2,3-dihydro-1H-indol-2-one
5-phenoxy-N-(4H-1,2,4-triazol-4-yl)furan-2-carboxamide
5-[4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)piperidine-1-carbonyl]-1,3-benzothiazole
5-[(3-hydroxypiperidin-1-yl)methyl]-N-methyl-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
3-(2-propyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
2-(4-{[methyl(oxan-4-ylmethyl)amino]methyl}phenyl)-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
3-(phenoxymethyl)-5-{pyrazolo[1,5-a]pyridine-3-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N,N-dimethyl-2-{[1-(2-methylpropyl)piperidin-4-yl]amino}ethane-1-sulfonamide
2-fluoro-N-({4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)benzamide
1-(2-fluorophenyl)-N-(2-hydroxyethyl)-N-(3-methyl-1,1-dioxo-1λ6-thiolan-3-yl)cyclopropane-1-carboxamide
6-{[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]amino}-N-[(3-propyl-1,2-oxazol-5-yl)methyl]pyridine-3-carboxamide
4,6-dimethyl-5-{4-[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]piperidine-1-carbonyl}-2H-pyran-2-one
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-3-hydroxy-4-methoxybenzamide
5-fluoro-N4,N4-dimethyl-N2-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}pyrimidine-2,4-diamine
1-[1'-(4-methylquinolin-2-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
(2S,4R)-1-{[2-(cyclopentyloxy)phenyl]methyl}-4-acetamido-N-ethylpyrrolidine-2-carboxamide
4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(2-fluorophenyl)methyl]piperidine
1-methyl-4-[5-(pyrrolidine-1-carbonyl)pyridin-2-yl]piperazine-2-carboxylic acid
2-{4-[(2-ethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}pyridine-3-carbonitrile
(2-methoxyethyl)[(6-methoxypyridin-3-yl)methyl](thiophen-2-ylmethyl)amine
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-1-methyl-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide