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N-{[3-(3-fluorophenyl)-1,2-oxazol-5-yl]methyl}-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
1-{4-[5-(3-fluorophenyl)-2-[(2-methoxyethyl)sulfanyl]pyrimidin-4-yl]piperidin-1-yl}-2-(1H-imidazol-1-yl)ethan-1-one
N-{4-methyl-2-[2-(pyridin-3-yloxy)acetamido]phenyl}pentanamide
3-{1-[(3-acetylphenyl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)propanamide
2-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-5-fluoropyridine
3-{1-[1-(2,3-dihydro-1H-indene-2-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-1-ol
2-tert-butyl-4-[4-(2-chlorophenyl)piperidin-4-yl]pyrimidine
methyl 2-[5-(pyrrolidin-2-yl)thiophene-2-amido]pyridine-4-carboxylate
[2-ethoxy-5-({[(4-fluorophenyl)methyl](prop-2-en-1-yl)amino}methyl)phenyl]methanol
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[1-(dimethyl-1,2-oxazole-4-carbonyl)piperidin-3-yl]piperazine
1-[2-({[2-(2-fluorophenyl)ethyl]amino}methyl)-5-methoxyphenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
N-[(1-methanesulfonylpiperidin-3-yl)methyl]-6-methyl-2-propylpyrimidin-4-amine
(4aS,8aR)-6-(3-cyclopropylpropanoyl)-1-[2-(1H-imidazol-4-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
4-[(2S)-1-[(3-chloro-4,5-dimethoxyphenyl)methyl]pyrrolidine-2-carbonyl]morpholine
(3aS,6aS)-2-acetyl-5-[3-(dimethylsulfamoyl)propyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-(1H-1,3-benzodiazol-2-yl)-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxylic acid
N-(2-hydroxyethyl)-N-[(5-methylthiophen-2-yl)methyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
(3aR,6aR)-2-(5-cyano-4,6-dimethylpyridin-2-yl)-5-(cyclobutylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(3-fluorophenyl)methyl]-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-ethyl-3-(piperidine-1-carbonyl)-N-(thiophen-3-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-{[(3aR,5S,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]methyl}-3,5-dimethyl-1,4-dihydropyridin-4-one
(3R,9aR)-8-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
dimethyl(2-{2-[1-(2-methyl-1H-1,3-benzodiazole-5-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)amine
4-{[2-(5-ethylfuran-2-yl)-1H-imidazol-1-yl]methyl}benzene-1-sulfonamide
3-({1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]pyrrolidin-3-yl}methyl)benzoic acid
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}piperazine
4-benzyl-1-[2-(morpholin-4-yl)-2-oxoethyl]pyrrolidin-2-one
3-(methanesulfonylmethyl)-1-(3-phenylpropyl)piperidine
5-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-2-carbonyl}-2-(methylsulfanyl)-3,4-dihydropyrimidin-4-one
1-[(2,3-difluoro-6-methoxyphenyl)methyl]-4-(1H-imidazol-1-ylmethyl)piperidine
3-(2-hydroxyphenyl)-3-(3-hydroxyphenyl)-N-(1-phenylcyclopropyl)propanamide
3-(2-chlorophenyl)-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)propanamide
N-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)-4-(6-ethylpyrimidin-4-yl)piperazine-1-carboxamide
9-hydroxy-7-(5-methylthiophen-2-yl)-N-(propan-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carboxamide
N-benzyl-7-cyclobutanecarbonyl-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(1S,5R)-N-[2-(2-fluorophenyl)ethyl]-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
9-[(2,3,4-trimethoxyphenyl)methyl]-3-oxa-9-azaspiro[5.5]undecane
1-{[2-(4-chlorophenyl)-7-methoxyquinolin-3-yl]methyl}piperidin-3-ol
5-(4-benzylpiperidin-1-yl)-1-ethyl-3-(4-methyl-1,4-diazepane-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-(2-oxopyrrolidin-1-yl)acetamide
1-acetyl-N-[2-(4-fluorobenzenesulfonyl)ethyl]piperidine-3-carboxamide
[1-(1-cycloheptanecarbonylpiperidin-4-yl)-1H-1,2,3-triazol-4-yl]methanol
5-benzyl-5-{1-[(2-phenyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
(3aR,7aS)-2-(5-ethyl-1,3-oxazole-4-carbonyl)-2,3,3a,4,7,7a-hexahydro-1H-isoindole
1-(3-chloropyridin-2-yl)-4-[(2,4-dimethoxyphenyl)methyl]piperazine
3,5-dimethyl-2-{[2-(4-methylpentyl)morpholin-4-yl]methyl}-1,4-dihydropyridin-4-one
1-[2-(4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)phenyl]ethan-1-one
1-(2-chloro-4-fluoro-5-methylphenyl)-3-[2-(5-cyclobutyl-1,2,4-oxadiazol-3-yl)ethyl]urea
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)benzamide
2-oxo-N-[2-(phenylsulfanyl)ethyl]-N-(propan-2-yl)-2,3-dihydro-1H-imidazole-4-carboxamide