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N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-1,5-dimethyl-1H-pyrazole-3-carboxamide
2-cyclopentyl-N-{[2-(dimethylamino)-7-methoxyquinolin-3-yl]methyl}-N-(2-methoxyethyl)acetamide
(3S,7S,8aS)-3-[(benzyloxy)methyl]-7-{[(3-chloro-1-benzothiophen-2-yl)methyl]amino}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
1-[2-(1H-imidazol-1-yl)ethyl]-2-(5-phenylthiophen-2-yl)-1H-imidazole
5-(azepan-1-yl)-1-ethyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-[(pyrrolidin-3-yl)amino]pyridine-3-carboxamide
2-methoxy-5-[3-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]pyridine
(3R,4R)-4-(azepan-1-yl)-1-[(4-fluoro-2-methoxyphenyl)methyl]piperidin-3-ol
4-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidine-1-carbonyl]-2,6,8-trimethylquinoline
2-(4-methyl-1H-imidazol-5-yl)-1-(2,2,2-trifluoroethyl)-1H-imidazole
(2R)-4-[(6,8-dimethoxy-4-methylquinolin-2-yl)amino]-2-methylbutan-1-ol
1-(3,5-dimethylphenyl)-4-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperazin-2-one
4-{2-[2-(4-fluorophenyl)piperidin-1-yl]-2-oxoethyl}-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
(3aS,7aR)-5-methyl-2-[(3-phenyl-1,2-oxazol-5-yl)methyl]-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
2-(9-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl)acetamide
methyl 3-[1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-8-yl]propanoate
3-{[3-hydroxy-3-(piperidin-1-ylmethyl)pyrrolidin-1-yl]methyl}-7-methyl-1,2-dihydroquinolin-2-one
4-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
(2E)-3-(3-fluorophenyl)-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]prop-2-enamide
N-(3-methylbutyl)-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(propan-2-yloxy)ethan-1-one
5-[3-(5-methyl-1,2,4-oxadiazol-3-yl)benzoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
2-(pyridin-4-ylmethyl)-9-(trimethyl-1H-pyrazole-4-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
2-fluoro-N-[(5-methylthiophen-2-yl)methyl]-N-(prop-2-en-1-yl)-5-sulfamoylbenzamide
8-({9-hydroxy-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-(1-{[2-(methylsulfanyl)phenyl]methyl}pyrrolidin-3-yl)piperidine
3-(5-chloro-2-methoxybenzoyl)piperidine
8-[2-(methylamino)acetyl]-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-2-(pyridin-3-yl)acetamide
(4aR,8aS)-1-(2H-1,3-benzodioxol-5-ylmethyl)-6-[(4-methoxy-3-methylphenyl)methyl]-decahydro-1,6-naphthyridin-2-one
5-{[benzyl(methyl)amino]methyl}-N-[2-(methylamino)ethyl]-1,2-oxazole-3-carboxamide
(2R)-2-amino-1-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-phenylethan-1-one
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[2-(pyridin-4-yl)ethyl]acetamide
1-cyclobutanecarbonyl-N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}piperidine-4-carboxamide
4-ethyl-1-[(2-methylphenyl)methyl]-1,4-diazepan-5-one
methyl 1-{2-[(3-methoxyphenyl)amino]butanoyl}piperidine-4-carboxylate
methyl 3-[(butan-2-yl)(pyridin-4-ylmethyl)carbamoyl]propanoate
1-(2-{2-azaspiro[4.4]nonan-2-yl}-2-oxo-1-phenylethyl)-4-butylpiperazine-2,3-dione
1,3-dimethyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1H-indole-2-carboxamide
(2S)-2-[4-(4-fluoro-3-methoxyphenyl)-1H-1,2,3-triazol-1-yl]-4-(methylsulfanyl)butanoic acid
2-methyl-N-[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-4,5,6,7-tetrahydro-1,3-benzothiazol-4-amine
3-(2-oxo-2-{4-[2-(1H-pyrrol-1-yl)ethyl]piperazin-1-yl}ethyl)imidazolidine-2,4-dione
2-chloro-4-({[(1-cyclohexylpiperidin-3-yl)methyl](pyridin-3-ylmethyl)amino}methyl)phenol
8-[2-(prop-2-en-1-yloxy)benzoyl]-2,8-diazaspiro[4.5]decan-3-one
2-methoxy-N-{[5-(quinolin-6-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}acetamide
7-(1-benzothiophen-3-yl)-4-(oxolane-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(2S)-1-{5-[(4-benzylpiperidin-1-yl)methyl]-1,2-oxazole-3-carbonyl}pyrrolidine-2-carboxamide
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(2-oxopiperidin-1-yl)ethyl]acetamide
3-[(4-hydroxy-1,2,3,4-tetrahydroisoquinolin-2-yl)methyl]-6-methoxy-1,2-dihydroquinolin-2-one