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3,5-dichloro-N-[2-(ethanesulfonyl)ethyl]-4-methylbenzamide
[(3-tert-butyl-1H-pyrazol-5-yl)methyl](methyl){[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amine
3-(dimethylamino)-N-[4-(2-methoxyphenoxy)phenyl]pyrrolidine-1-carboxamide
3-(4-{5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl}piperazine-1-carbonyl)-4,5,6,7-tetrahydro-1,2-benzoxazole
1-methyl-3-(2-methylpropyl)-5-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl}-1H-pyrazole
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-2-(trimethyl-1H-pyrazol-1-yl)acetamide
3-[2-(methylsulfanyl)ethyl]-5-[1-(1H-1,2,4-triazol-1-yl)ethyl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
1,6-dimethyl-N-(4-phenylbutyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N,N-dimethyl-4-[2-({[3-(trifluoromethyl)phenyl]methyl}carbamoyl)ethyl]piperidine-1-carboxamide
1-[2-(4-fluorophenyl)ethyl]-4-[(thian-4-yl)amino]pyrrolidin-2-one
9-[(3-fluoro-4-methylphenyl)methyl]-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
4-hydroxy-N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
5-[({[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}(propan-2-yl)amino)methyl]pyrrolidin-2-one
N-[(2-chloropyridin-3-yl)methyl]-6-methoxy-N-methylpyrimidin-4-amine
4-({4-[(4-fluorophenyl)methyl]piperidin-1-yl}methyl)pyrimidine
N-methyl-N-[(5-methylfuran-2-yl)methyl]-2,1-benzoxazole-3-carboxamide
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-(2-methyl-1H-imidazol-1-yl)acetamide
6-methyl-8-{8-methyl-2,8-diazaspiro[4.5]decane-2-carbonyl}-4-oxa-2,5-diazatricyclo[7.3.0.03,7]dodeca-1(9),2,5,7-tetraene
3-[(4-ethyl-1,3-thiazol-2-yl)methyl]-1-[3-(piperidine-1-carbonyl)phenyl]urea
[2-(3,6-dimethylpyrazin-2-yl)phenyl]methanol
1-(2-methylfuran-3-carbonyl)-4-(2-methylphenyl)-1,4-diazepane
1-[(4-fluorophenyl)methyl]-5-(4-methylpiperidin-1-yl)azepan-2-one
N-ethyl-5-{[4-(2-fluoro-5-methylphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyrimidin-2-amine
2-[1-(1-benzylpiperidin-4-yl)-3-oxopiperazin-2-yl]-N-methylacetamide
N-[1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carboxamide
N-[2-(1H-1,2,4-triazol-1-yl)ethyl]-1H-1,3-benzodiazole-2-carboxamide
8-{2-[4-(2-methoxyethoxy)piperidin-1-yl]-2-oxoethyl}-8-azaspiro[4.5]decane-7,9-dione
1-{[2,5-dimethoxy-4-(methylsulfanyl)phenyl]methyl}piperidine-3-carbonitrile
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)cyclopentanamine
5-[1-(2H-1,3-benzodioxol-5-yl)propan-2-yl]-1-cyclopentyl-1H,4H-pyrazolo[3,4-d]imidazole
2-[(1,4-dioxan-2-ylmethyl)(methyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
1-(4-ethylpiperazin-1-yl)-3-[3-({methyl[(3-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]propan-2-ol
4-methyl-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]pyrimidin-2-amine
1-[1-(cyclohex-3-en-1-ylmethyl)azetidin-3-yl]-3,5-dimethyl-1H-pyrazole
4-[2-(dimethylamino)-2-(2-methylphenyl)acetyl]piperazine-1-carboxamide
3-[({1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)methyl]-1λ6-thiolane-1,1-dione
3-(2-{[(2,4-dimethoxyphenyl)methyl]carbamoyl}ethyl)-N-(propan-2-yl)piperidine-1-carboxamide
1-{2-[1-(2-methyl-1,3-benzothiazol-6-yl)-1H-1,2,4-triazol-5-yl]ethyl}piperidine-4-carboxamide
N3-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]piperidine-1,3-dicarboxamide
2-(pyrimidin-2-ylmethyl)-5-(1,2,3,4-tetrahydroisoquinolin-2-yl)-2,3-dihydropyridazin-3-one
1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4-[1-(pyrrolidin-1-yl)ethyl]piperidine
2-[3-(2H-1,3-benzodioxole-5-carbonyl)piperidin-1-yl]-N,6-dimethylpyrimidin-4-amine
N-(5-acetyl-2-ethoxyphenyl)-4-[(1S,2S)-2-hydroxycyclohexyl]piperazine-1-carboxamide
N-[2-(azepan-1-yl)ethyl]-2-methyl-6-(piperidin-4-yl)pyrimidin-4-amine
1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-{1H-pyrrolo[2,3-b]pyridin-6-yl}piperazine
2-amino-6-methyl-4-[3-(pyridin-2-yl)phenyl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
N3,N3-diethyl-N1-(3-methyl-1,2,4-thiadiazol-5-yl)piperidine-1,3-dicarboxamide
1-(4-chlorophenyl)-N-{[5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclobutane-1-carboxamide
3-[({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(oxolan-2-ylmethyl)carbamoyl]pyridin-1-ium-1-olate
2-(2-methoxyethyl)-8-[2-(3-oxopiperazin-1-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one