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{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}[(4-fluorophenyl)methyl](prop-2-en-1-yl)amine
4-{4-[(2-fluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}-2-methoxypyridine-3-carbonitrile
5-(3-fluoro-4-methoxyphenyl)thiophene-2-carboxamide
N-cyclopropyl-5-methyl-6-(pyrrolidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-amine
1-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-yl]-2-(pyridin-4-yl)ethan-1-one
(3R,5S)-N-cyclopropyl-1-[(3,4-dimethoxyphenyl)methyl]-5-(morpholin-4-ylmethyl)piperidine-3-carboxamide
1-(cyclobutylmethyl)-3-(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-1-(oxolan-2-ylmethyl)urea
[(3R,5R)-5-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-(3-methyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]methanol
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-4-(4-fluorophenyl)-N-methyloxane-4-carboxamide
5-{5,7-dimethylpyrazolo[1,5-a]pyrimidin-2-yl}-3-(oxolan-3-yl)-1,2,4-oxadiazole
[(3R,4R)-4-(piperidin-1-ylmethyl)-1-(pyrimidin-2-yl)pyrrolidin-3-yl]methanol
5-fluoro-2-({[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methoxy}methyl)-1H-1,3-benzodiazole
3,5-dimethoxy-N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)benzamide
8-fluoro-2-[2-(thiophen-2-yl)azetidine-1-carbonyl]quinoline
{[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}(methyl)[2-(4-methylphenoxy)ethyl]amine
N-methyl-2-(oxan-2-ylmethoxy)-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]acetamide
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-(4-methyl-1,4-diazepan-1-yl)acetamide
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]acetamide
(2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}quinolin-3-yl)methanol
N-cyclopentyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-1H-pyrrole-2-carboxamide
(1R,5R)-N,N-dimethyl-6-(4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-(furan-2-ylmethyl)-1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidine-4-carboxamide
1-[(2-fluorophenyl)methyl]-5-[4-(3-methoxypropyl)piperidine-1-carbonyl]piperidin-2-one
2-[4-(3-methylbutanoyl)piperazin-1-yl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
1-benzyl-5-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)-4-oxo-N-(prop-2-en-1-yl)-1,4-dihydropyridine-3-carboxamide
N-[3-(methylsulfanyl)propyl]-2-[3-oxo-1-(pyridin-3-ylmethyl)piperazin-2-yl]acetamide
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-5-methanesulfonyl-2-methylpyrimidin-4-amine
4-(1,3-benzothiazole-6-carbonyl)-3-(3-fluorophenyl)piperazin-2-one
1-(2,3-dihydro-1H-inden-2-yl)-4-{[(1-methyl-1H-imidazol-2-yl)methyl]amino}pyrrolidin-2-one
4,6-dimethyl-5-{[4-(1H-pyrazol-1-yl)butan-2-yl]amino}-1,2-dihydropyridin-2-one
1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}-2-(1H-pyrazol-1-yl)butan-1-one
8-[2-(methylsulfanyl)pyrimidine-5-carbonyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-1-(propan-2-yl)piperidine-3-carboxamide
4-{[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-2,1,3-benzoxadiazole
2-(4-methoxyphenyl)-5-{[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]methyl}pyrimidine
2-ethoxy-6-({4-[(4-fluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenol
1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(pyridin-2-yl)ethan-1-one
1-(4-aminopyrimidin-2-yl)-4-(4-methylpiperazine-1-carbonyl)-1,4-diazepan-6-ol
1-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
5-methyl-2-[1-(piperidin-4-yl)-1H-1,2,3-triazol-4-yl]-1H-1,3-benzodiazole
N-[3-(4-chlorophenoxy)-2-hydroxypropyl]-2-(2,4-difluorophenoxy)acetamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]quinoxaline-6-carboxamide
N-methyl-5-[(1-oxo-1,2-dihydrophthalazin-2-yl)methyl]-1,2,4-oxadiazole-3-carboxamide
5-butyl-N4,6-dimethyl-N4-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]pyrimidine-2,4-diamine
[(3R,4R)-1-(2-methyl-1-benzofuran-5-carbonyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
(1S,5R)-3-[(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)methyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
4-(4-chlorophenyl)-1-[(2S)-2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl]butan-1-one
3-{3-[({[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}carbamoyl)amino]phenyl}-N,N-dimethylpropanamide
N-(2-{[(3-chlorophenyl)methyl]sulfanyl}ethyl)-2,2-dimethyloxane-4-carboxamide