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N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-3-acetamidobenzamide
4-[(1-benzylpiperidin-4-yl)oxy]-N-(pyridin-2-ylmethyl)benzamide
(1S,4S)-2-(2-{3-[3-(3-methylpyridin-2-yl)phenyl]-1H-pyrazol-1-yl}ethyl)-2-azabicyclo[2.2.1]heptane
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N,2,5-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-N-(2-hydroxy-2-phenylethyl)-N,5-dimethyl-1H-pyrazole-4-carboxamide
N-methyl-N-[2-(pyridin-2-yl)ethyl]-1,4-dioxane-2-carboxamide
1-(1-{[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)piperidin-3-ol
N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)-3-(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)propanamide
N,N-dimethyl-2-({[4-(propan-2-yl)phenyl]formamido}methyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
5-methoxy-9-(5-methoxy-1,2-dimethyl-1H-indole-3-carbonyl)-1-oxa-9-azaspiro[5.5]undecane
2-cyclopropyl-9-(3-hydroxypropyl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
1-{1-[1-(2-methoxy-4-methylbenzoyl)piperidin-4-yl]ethyl}-4-methylpiperazine
N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-2,3-dimethylquinoxaline-6-carboxamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-(1-methyl-1H-pyrrol-2-yl)-2-oxoacetamide
2-[(3-fluorophenyl)methyl]-4-{4-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
methyl 5-cyano-6-({1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}amino)-2-methylpyridine-3-carboxylate
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[2-(1H-imidazol-1-yl)acetyl]pyrrolidin-3-yl]-5-methyl-1,2-oxazole-4-carboxamide
1-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(pyridin-3-yl)ethan-1-one
3-[(3S,4R)-1-[(3-chlorophenyl)methyl]-4-(pyrrolidin-1-yl)piperidin-3-yl]-N-[2-(morpholin-4-yl)ethyl]propanamide
4-(4-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperazine-1-carbonyl)morpholine
methyl 2-{5-[1-(2-fluoro-5-methylbenzenesulfonyl)piperidin-4-yl]-1H-pyrazol-3-yl}acetate
2-(4-chloro-1-methyl-1H-pyrazol-3-yl)-7-methyl-1H-1,3-benzodiazole
5-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
(2S,4R)-N,N-diethyl-4-(3-hydroxypropanamido)-1-[(5-methylthiophen-2-yl)methyl]pyrrolidine-2-carboxamide
1-{3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}-2-(furan-2-yl)azepane
2,6-dimethyl-4-({3-oxo-2,8-diazaspiro[4.5]decan-8-yl}methyl)phenyl acetate
3-fluoro-N-{1-[1-(2-hydroxypropyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
N-[3-(2,4-dimethylphenoxy)-2-hydroxypropyl]-3-(1H-pyrazol-1-yl)benzamide
methyl 4-{[(2-{5-oxo-1-[3-(propan-2-yloxy)propyl]pyrrolidin-2-yl}ethyl)amino]methyl}benzoate
N-cyclopentyl-1-(2-methylpropyl)-5-(prop-2-en-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[(4-fluorophenyl)methyl]-4-(6-methoxypyrimidin-4-yl)piperazin-2-one
N-(cyclohexylmethyl)-1-cyclopropyl-4-oxo-5-[4-(propan-2-yl)piperazine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
N-[2-(dimethylsulfamoyl)ethyl]-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
6-methyl-N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}imidazo[1,2-a]pyridine-2-carboxamide
9-(4-methylpiperazine-1-carbonyl)-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
6-(1-methyl-1H-imidazol-2-yl)-N-[1-(3-methylpyridin-2-yl)propan-2-yl]pyridazin-3-amine
{1-[(3-chloro-5-fluoro-4-methoxyphenyl)methyl]-3-(3-methylbut-2-en-1-yl)piperidin-3-yl}methanol
7-(cyclohexylmethyl)-2-(2-methoxyacetyl)-2,7-diazaspiro[4.5]decan-6-one
4-{[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1H-imidazole
N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5,6,7,8-tetrahydroquinoline-3-carboxamide
8-[5-(ethylsulfanyl)thiophene-2-carbonyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-[(4-methyl-1H-imidazol-5-yl)methyl]cyclopropanamine
N-[4-(3-fluorophenyl)phenyl]-1-(thiophene-2-carbonyl)piperidine-3-carboxamide
methyl N-{2-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]-2-oxoethyl}carbamate
2-({5-[(dimethylamino)methyl]-4-[2-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-3-yl}sulfanyl)acetic acid
6-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-5-chloropyridine-3-carboxylic acid
(2R)-2-acetamido-N-{[1-(hydroxymethyl)cyclobutyl]methyl}-N-methylpropanamide
N-[1-(furan-2-ylmethyl)piperidin-4-yl]-4-hydroxy-2-phenylpyrimidine-5-carboxamide
5-[2,2-bis(prop-2-en-1-yl)pyrrolidine-1-carbonyl]-4,6-dimethyl-1,2,3,4-tetrahydropyrimidin-2-one
7-(7-fluoro-4-methylquinolin-2-yl)-4-[(5-methylthiophen-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol