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2-{3-[3-(methylsulfanyl)phenyl]phenoxy}acetamide
1-{2-[2-(azetidin-1-ylmethyl)phenoxy]ethyl}-3-methylpiperidine
N-[2-(morpholin-4-ylmethyl)phenyl]-4-phenylpiperidine-1-carboxamide
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
2-(4-cyclopentyl-3-oxopiperazin-1-yl)-2-(4-methoxy-2-methylphenyl)acetic acid
N-[(3S,5S,9R)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]-4-fluoro-3-(trifluoromethyl)benzamide
(4S)-3-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-4-phenyl-1,3-oxazolidin-2-one
1-(3-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)-3-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}urea
3-(4-methyl-1,3-thiazol-5-yl)-1-[4-(thiophen-3-ylmethyl)piperazin-1-yl]propan-1-one
4-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzoyl]morpholine
1-(2-methylpyrimidin-4-yl)-4-(3-phenylpropyl)piperidine-4-carboxylic acid
propan-2-yl 3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxylate
N-methyl-2-{4-[methyl(2-phenylethyl)amino]-6-oxo-1,6-dihydropyridazin-1-yl}propanamide
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}(2-methoxyethyl)(1H-pyrazol-3-ylmethyl)amine
({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amine
5-(cyclopropylmethyl)-3-[4-(trifluoromethyl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-(1,4-oxazepan-4-yl)pyridine-3-carboxamide
(3S,9aR)-3-benzyl-8-(2,3-difluorobenzoyl)-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-oxo-2-[4-(pyridin-4-yl)piperidin-1-yl]-S-(thiophen-2-yl)ethane-1-sulfonamido
2-[4-(2-butoxy-4-fluorophenyl)-1H-pyrazol-1-yl]propanamide
2-amino-1-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-methylpropan-1-one
(1R,4S)-1,7,7-trimethyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-3-oxo-2-oxabicyclo[2.2.1]heptane-4-carboxamide
1-(2-aminoethyl)-N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-cyclobutanecarbonyl-4-[2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]piperidine
2-(3-methylbutyl)-8-[2-(3-oxopiperazin-1-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
5-(2-methyl-1H-imidazol-4-yl)-4-phenyl-1H-imidazole
3-(prop-2-en-1-yl)-1-(1-propyl-1H-pyrazole-5-carbonyl)piperidine-3-carboxylic acid
1-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]piperidine-3-carboxamide
(2S,4R)-1-(2,3-dihydro-1H-inden-2-yl)-N-(2-methoxyethyl)-4-[(naphthalen-2-ylmethyl)amino]pyrrolidine-2-carboxamide
1-methyl-6-oxo-N-[1-(thiophen-2-ylmethyl)piperidin-4-yl]-1,6-dihydropyridazine-3-carboxamide
1-{3-fluoro-5-methylimidazo[1,2-a]pyridine-2-carbonyl}-3-phenylpiperazine
N-cyclopropyl-N-{[3-(oxolan-2-ylmethoxy)phenyl]methyl}furan-2-carboxamide
2-{2-[3-(ethoxymethyl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-1,3-benzodiazole
(1R,3s,6r,8S)-4-[7-fluoro-2-(1H-pyrazol-4-yl)quinoline-4-carbonyl]-4-azatricyclo[4.3.1.13,8]undecane
2-(1H-1,3-benzodiazol-2-ylmethoxy)-1-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]ethan-1-one
6-{[2-(1-ethylpiperidin-4-yl)ethyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(1-cyclopentanecarbonylpiperidin-3-yl)piperazine
N-[2-(cyclohex-1-en-1-yl)ethyl]-2-cyclopropyl-N-(cyclopropylmethyl)-4-hydroxypyrimidine-5-carboxamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-3-(2-oxoimidazolidin-1-yl)benzamide
2-{3,5-dimethyl-4-[3-(propan-2-yloxy)phenyl]-1H-pyrazol-1-yl}acetamide
(3aS,6aR)-3-cyclopentyl-5-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-methyl-5-({2-oxo-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}methyl)furan-2-carboxamide
1-(morpholin-4-yl)-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propan-1-one
3-(3-chlorobenzoyl)-N-(2,5-dimethylphenyl)piperidine-1-carboxamide
1-{5,7-dimethyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carbonyl}-4-(1-methyl-1H-imidazol-2-yl)piperidine
5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-1-(prop-2-en-1-yl)pyrrolidin-2-one
methyl (2S)-2-({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amino)-3-phenylpropanoate
methyl 4-{4-[1-(methoxymethyl)cyclobutanecarbonyl]piperazin-1-yl}benzoate
N-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]-3-phenyl-1H-pyrazole-4-carboxamide