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1-cyclopentanecarbonyl-N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-4-carboxamide
(3aR,6aR)-2-(2-cyclopentylacetyl)-5-(2-methoxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-cyclopropyl-3-methyl-N-[2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]-1H-pyrazole-4-carboxamide
3-{1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidin-3-yl}-N-[4-(trifluoromethyl)phenyl]propanamide
8-[3-(5-methyl-1H-pyrazol-1-yl)propanoyl]-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
N-[(1-cyclohexylpiperidin-3-yl)methyl]-3,5-dimethyl-N-(pyridin-3-ylmethyl)-1,2-oxazole-4-carboxamide
N-[2-(4-chlorophenyl)ethyl]-2-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]acetamide
[2-({4-[(3,5-dimethyl-1-benzofuran-2-yl)methyl]piperazin-1-yl}methyl)phenyl]methanol
5-(1-methyl-1H-pyrazol-4-yl)-N-(pyridin-3-yl)furan-2-carboxamide
3-[(4-fluorophenyl)formamido]-N-[1-(pyridin-3-yl)pentyl]propanamide
3-[3-(4-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1,2-dihydroquinoxalin-2-one
1-methyl-4-{4-[1-(propan-2-yl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]phenyl}piperazine
1-(2-methoxyethyl)-3-methyl-8-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2R,3R,6R)-3-(2-methoxyphenyl)-5-(pyridine-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[(5-amino-1,3,4-thiadiazol-2-yl)(phenyl)methyl]-2-(dimethylamino)-4-methylpyrimidine-5-carboxamide
2-amino-6-(4-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)-3,4-dihydropyrimidin-4-one
N,N-dimethyl-5-[3-(1-methylpiperidin-2-yl)propanoyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-2-(1-methyl-1H-pyrrol-3-yl)acetamide
3-[1-(4-methoxy-3-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
6-[4-(1-benzofuran-2-ylmethyl)piperazin-1-yl]pyridine-3-carbonitrile
N-ethyl-5-[4-(4-methoxyphenoxy)piperidine-1-carbonyl]pyrimidin-2-amine
ethyl 1-[(2,4-difluorophenyl)carbamoyl]-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
1-(cyclopropylmethyl)-N-ethyl-5-[2-(pyridin-2-ylsulfanyl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[4-(1-hydroxy-3-methylbutyl)piperidin-1-yl]ethan-1-one
(1-{5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1H-pyrazole-3-carbonyl}-2,5-dihydro-1H-pyrrol-2-yl)methanol
3-[2-methyl-4-(2-methylphenyl)piperazine-1-carbonyl]-1,2,5,6,7,8-hexahydroquinolin-2-one
N-[(4-phenyloxan-4-yl)methyl]-4-(pyridin-2-yl)pyrimidin-2-amine
4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)-N-(thiophen-2-yl)piperazine-1-carboxamide
1-{2-[4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]-2-oxoethyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
(3S,9aR)-3-(cyclohexylmethyl)-8-(4-ethylbenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-hydroxy-N-({2-methoxy-5-oxo-6-[2-(pyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)butanamide
3-(5-methanesulfonamido-2-methylphenyl)-1-[1-(3-methylpyridin-2-yl)propan-2-yl]urea
1-[3-(furan-2-yl)phenyl]-N-(1,2-oxazol-3-ylmethyl)piperidin-4-amine
N-[(1-benzylpiperidin-4-yl)methyl]-4-methylpyrimidin-2-amine
4-{[2-(3-hydroxypropyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]methyl}-N-methylbenzamide
(1R,5R)-3-(2-chloro-4-fluorobenzoyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonane
2-methoxy-4-{1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl}pyridine-3-carbonitrile
8-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-1-oxa-8-azaspiro[4.5]decan-3-ol
N-phenyl-4-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)piperidine-1-carboxamide
4-[4-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-3-methylpyridine
N-{2-[(5-chlorothiophen-2-yl)sulfonyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}pyridine-2-carboxamide
methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]({2-[4-(morpholin-4-yl)butoxy]phenyl}methyl)amine
4-methyl-7-{[methyl({[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl})amino]methyl}-2H-chromen-2-one
4-(1-{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)morpholine
4-[3-(1H-pyrazol-1-yl)azetidine-1-carbonyl]-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[2-(1H-pyrazol-4-yl)ethyl]acetamide
3-hydroxy-3-(hydroxymethyl)-N-[2-(3-methylphenoxy)phenyl]pyrrolidine-1-carboxamide
(3S,4S)-1-(2,2-diphenylethyl)-4-(1,4-oxazepan-4-yl)pyrrolidin-3-ol
1-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-4-(propan-2-yl)-1,2,3-thiadiazole-5-carboxamide