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N-[(2-aminopyrimidin-5-yl)methyl]-1-(4-fluorophenyl)-N-methylcyclopropane-1-carboxamide
N-[2-(6-oxo-1,6-dihydropyrimidin-4-yl)ethyl]-2-{3-oxo-2-azatricyclo[6.3.1.04,12]dodeca-1(12),4,6,8,10-pentaen-2-yl}propanamide
3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1-[(1S,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]propan-1-one
8-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}-1,3-dioxa-8-azaspiro[4.5]decan-2-one
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-5-(methoxymethyl)thiophene-2-carboxamide
N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-1-(2-methylpropyl)-5-oxopyrrolidine-3-carboxamide
N-{2-[4-(4-fluorophenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]ethyl}-3-methylthiophene-2-carboxamide
[2-({4-[4-methyl-2-(propan-2-yl)pyrimidine-5-carbonyl]piperazin-1-yl}methyl)phenyl]methanol
1-ethyl-3-(hydroxymethyl)-N-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carboxamide
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
1-cyclopentanecarbonyl-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidine-4-carboxamide
1-{6-[4-(piperidine-1-carbonyl)piperidin-1-yl]pyrimidin-4-yl}piperidin-4-ol
2-(cyclopropylmethyl)-N-[2-methyl-2-(morpholin-4-yl)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-(4-methylpiperazin-1-yl)pyridine-3-carboxamide
8-(3,3-dimethylbutanoyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
(3aS,6aR)-5-benzoyl-3-[2-(3-chlorophenyl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
ethyl(1H-imidazol-4-ylmethyl){[2-(prop-2-en-1-yloxy)phenyl]methyl}amine
6-[1-(2-ethoxypyridine-3-carbonyl)piperidin-3-yl]-2-methylpyrimidin-4-ol
(1S,5R)-6-(cyclobutylmethyl)-3-(4-methylpyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}-2-(3-hydroxyphenyl)ethan-1-one
2-chloro-5-acetamido-N-{1-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}benzamide
2-ethoxy-3-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]pyridine
2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-(pyrimidin-4-ylmethyl)acetamide
1-[(2-{[3-(2-methylphenoxy)azetidin-1-yl]methyl}phenyl)methyl]-1H-pyrazole
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(thiophen-2-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(3-chloro-4-methoxyphenyl)-3-{1-[2-(1H-imidazol-2-yl)ethyl]piperidin-3-yl}propanamide
2-[4-({[(3-chlorophenyl)methyl](propyl)carbamoyl}amino)phenyl]-N-methylacetamide
1-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one
2-{[1-(cyclopentylmethyl)piperidin-4-yl]oxy}-N-cyclopropyl-4-methoxybenzamide
2-(3-{1-[(5-chlorothiophen-2-yl)methyl]-1H-imidazol-2-yl}phenoxy)acetamide
3-[3-(benzyloxy)azetidine-1-carbonyl]piperidine-1-carboxamide
8-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(1S,5R)-3-(4-methanesulfonylbenzoyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[2-(2-fluoro-3-methoxyphenyl)pyrimidin-4-yl]piperidin-4-ol
3-[1-(2-methoxyacetyl)piperidin-3-yl]-1-methyl-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{2-[(2-methylpyrrolidin-1-yl)methyl]phenyl}-6-propyl-3,4-dihydropyrimidin-4-one
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-3-(2-hydroxyphenyl)-N-methyl-1H-pyrazole-5-carboxamide
4-(4-chlorophenyl)-N-[2-(1H-pyrrol-1-yl)ethyl]butanamide
1-[1-(1-benzothiophen-2-ylmethyl)piperidin-4-yl]-N-(3-hydroxypropyl)-1H-1,2,3-triazole-4-carboxamide
N-[(2,3-difluoro-4-methoxyphenyl)methyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
6-ethyl-2-methyl-4-[3-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]quinoline
4-chloro-N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1-methyl-1H-pyrazole-5-carboxamide
4-(1-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-1H-imidazol-2-yl)-2,1,3-benzoxadiazole
N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-1H-indole-6-carboxamide
N-cyclohexyl-1-ethyl-3-(4-methyl-1,4-diazepane-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-cyclopentyl-2-(5-oxopyrrolidin-2-yl)-N-propylacetamide
3-chloro-N-(3-methoxypropyl)-N-(1-methylpiperidin-4-yl)thiophene-2-carboxamide
2-({5-acetyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)benzonitrile
1-[4-(1-methoxypropan-2-yl)piperidin-1-yl]-2-(methylamino)ethan-1-one
N-[(1-ethyl-1H-imidazol-5-yl)methyl]-5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine