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5,6-dimethyl-2-oxo-N-[1-(3-phenylpropyl)piperidin-3-yl]-1,2-dihydropyridine-3-carboxamide
ethyl 1-(1-benzothiophene-2-sulfonyl)-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(4-hydroxy-3-methylbenzoyl)pyrrolidine-3-carboxylic acid
2-(2-methoxyphenyl)-5-[1-(pyridin-3-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]pyrimidine
[1-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)ethyl][(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]amine
methyl(pyridin-4-ylmethyl)[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]amine
5-[5-(1-methyl-1H-1,3-benzodiazol-2-yl)-4-phenyl-1H-imidazol-1-yl]pentan-1-amine
1-[2-(furan-2-yl)-4-[(3-methoxypropyl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]ethan-1-one
3-chloro-N-(2-methoxyethyl)-N-(thiophen-2-ylmethyl)pyridine-4-carboxamide
[2-(3,4-dimethoxyphenyl)ethyl]({[7-methoxy-2-(thiophen-3-yl)quinolin-3-yl]methyl})amine
3-({[(2-chlorophenyl)methyl]amino}methyl)-1-(cyclobutylmethyl)-3-hydroxypiperidin-2-one
2-{5-[3-(2-methoxyphenyl)phenyl]-3-methyl-1H-1,2,4-triazol-1-yl}ethan-1-ol
1-{[5-(oxan-2-yl)furan-2-yl]methyl}-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
3-[4-(azepan-1-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-yl]-1H-indole
4-{[2-(dimethylamino)ethyl]amino}-N-(3-methoxypropyl)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
5-{6-methyl-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole
N-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-1-[3-(2-methylpyrimidin-4-yl)phenyl]piperidin-4-amine
(2E)-3-(3-fluorophenyl)-1-[4-(3-{[methyl(2-phenylethyl)amino]methyl}phenoxy)piperidin-1-yl]prop-2-en-1-one
(1S,5R)-6-(cyclopropylmethyl)-3-(3,6-dimethyl-1-benzofuran-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[(cyclopropylmethyl)sulfanyl]-1-[4-(3-methoxybenzoyl)piperazin-1-yl]ethan-1-one
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}furan-2-carboxamide
4-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-[4-(2,6-difluoro-3-methylbenzoyl)-1-[(4-fluorophenyl)methyl]piperazin-2-yl]ethan-1-ol
2-({[(3R,4R)-1-[(2,3-difluoro-4-methylphenyl)methyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
1-{furo[3,2-c]pyridin-4-yl}-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
2-[2-({3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}methyl)phenoxy]ethan-1-ol
1-[(5-methylpyrazin-2-yl)methyl]-3-[2-(pyrrolidin-1-ylmethyl)phenyl]urea
N'-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-N,N-dimethylbutanediamide
1-[3-(morpholin-4-yl)propyl]-5-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]piperidin-2-one
4-[6-(2H-1,3-benzodioxol-5-yl)pyrazine-2-carbonyl]morpholine
1-{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidine-2-carboxamide
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
2-[(4-chlorophenyl)methyl]-8-(2-methoxybutanoyl)-2,8-diazaspiro[4.5]decan-3-one
3-{2-[4-(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]-2-oxoethyl}-2,3-dihydro-1,3-benzoxazol-2-one
4-(3-{2-[(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]phenoxy}propyl)morpholine
5-{[(5-chloropyridin-3-yl)oxy]methyl}-N-(oxolan-2-ylmethyl)-N-(pyridin-4-ylmethyl)-1,2-oxazole-3-carboxamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]-2,6-dimethylpyrimidine-4-carboxamide
3-ethyl-1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-3-methylpiperidine
3-cyclopropyl-1-methyl-5-[2-(trifluoromethoxy)phenyl]-1H,4H-pyrazolo[3,4-d]imidazole
2-[(2-fluoro-2-phenylacetamido)methyl]-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
2-{1-[(1-{8-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}ethan-1-ol
3-[({1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}oxy)methyl]pyridine
8-methyl-3-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}-1,2-dihydroquinolin-2-one
(2-methoxyethyl)[(3-methyl-1-benzofuran-2-yl)methyl][(trimethyl-1H-pyrazol-4-yl)methyl]amine
(2S)-1-[3-(2-ethylphenoxy)azetidin-1-yl]-2-(methylamino)propan-1-one
2-[4-(1-benzofuran-3-carbonyl)piperazin-1-yl]-4,6-dimethylpyrimidine
4-methyl-N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-3-(2-oxoimidazolidin-1-yl)benzamide
1-[4-(pyridin-2-yl)pyrimidin-2-yl]azetidine-2-carboxylic acid
9-(2-hydroxy-3-methylbutanoyl)-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]-N-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]acetamide