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1-methyl-4-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine-1-carbonyl)piperidine
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
N-cyclopentyl-N-[(2-methoxyphenyl)methyl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
4-(pyridin-2-yl)-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}pyrimidin-2-amine
5-(2-fluorophenoxymethyl)-N-[2-hydroxy-1-(pyridin-3-yl)ethyl]-1H-pyrazole-3-carboxamide
(3R,4R)-1-{[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-3-methyl-4-(oxan-4-yl)piperidin-4-ol
ethyl 4-[1-(6-methoxypyrimidin-4-yl)piperidin-4-yl]piperazine-1-carboxylate
N-[(6-chloro-1H-1,3-benzodiazol-2-yl)methyl]-5-(methoxymethyl)pyrazolo[1,5-a]pyrimidin-7-amine
2-{1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]pyrrolidin-3-yl}benzoic acid
4-[4-(3-methyl-1H-1,2,4-triazol-5-yl)piperidine-1-carbonyl]-5,6,7,8-tetrahydroquinazolin-2-amine
2-({[3-cyclopropyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}sulfanyl)-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-ol
1-(2,3-dimethylquinoxalin-6-yl)-3-(3-methyl-1,1-dioxo-1λ6-thiolan-3-yl)urea
3-methyl-4-(1-{[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl)-1,2,5-oxadiazole
1-[(6-ethoxyquinolin-2-yl)methyl]-3-methylpiperidine-3-carboxamide
N-[3-(1H-imidazol-1-yl)-1-phenylpropyl]-2-[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetamide
N-(4-methoxyphenyl)-3-(naphthalene-2-carbonyl)piperidine-1-carboxamide
1-(adamantan-1-yl)-2-{[6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}ethan-1-ol
1-[1-(2,6-difluorobenzoyl)piperidin-4-yl]-3-phenylpropan-1-ol
4-[2-(4-fluorophenyl)-2-hydroxyacetyl]-1-phenylpiperazin-2-one
6-{[3-(2-chlorophenyl)-1,2-oxazol-5-yl]methyl}-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-{[5-(5-chloro-3-fluoropyridin-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}cyclobutanecarboxamide
ethyl 5-[2-(4-chloro-2-methylphenoxy)propanoyl]-1-(cyclopropylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-[2-(4-methyl-5-{[2-(morpholin-4-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)ethyl]naphthalene-1-carboxamide
1-(4-methoxyphenyl)-6,6-dimethyl-N-(1,3-thiazol-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
(2S,3S)-3-methyl-2-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamido}pentanoic acid
3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]propan-1-one
(1S,5R)-6-[(2-ethylphenyl)methyl]-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-(3-hydroxyphenyl)-5-oxo-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]pyrrolidine-3-carboxamide
N-ethyl-2-(1H-indol-4-yl)pyrimidin-4-amine
3-(2-methylphenyl)-1-{6-methylpyrazolo[1,5-a]pyrimidine-3-carbonyl}pyrrolidin-3-ol
5-chloro-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-oxo-N-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl)[2-(piperidin-1-yl)ethyl]amine
2-(3-chlorophenyl)-2-hydroxy-N-[1-(2-methylpropanoyl)piperidin-4-yl]acetamide
9-[6-methyl-1-(propan-2-yl)-1H-pyrazolo[3,4-b]pyridine-4-carbonyl]-3,9-diazaspiro[5.6]dodecane
N-[2-(ethanesulfonyl)ethyl]-6-(piperidin-1-yl)pyrimidin-4-amine
2-(2,5-dimethoxyphenyl)-2-[4-(6-methylpyridin-2-yl)piperazin-1-yl]acetic acid
1-(2-phenylethyl)-N-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-4-carboxamide
3-(2-ethyl-1H-1,3-benzodiazol-6-yl)-1-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)urea
(4aS,7aR)-1-[(5-fluoro-2-methoxyphenyl)methyl]-4-(1H-imidazol-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[(2-chloro-6-fluorophenyl)methyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decane
(4aS,8aR)-1-butyl-6-{2-[4-(hydroxymethyl)phenyl]acetyl}-decahydro-1,6-naphthyridin-2-one
1-[2-(4-chlorophenyl)morpholin-4-yl]-4-(1H-pyrazol-1-yl)butan-1-one
2-(2-chloro-4-fluorophenyl)-1-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]ethan-1-one
10-methoxy-5-{1H-pyrrolo[2,3-b]pyridin-6-yl}-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
3-[2-(3-methyl-4H-1,2,4-triazol-4-yl)ethyl]-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(3-{[(1-hydroxybutan-2-yl)(pyridin-2-ylmethyl)amino]methyl}phenoxy)acetamide
2-methyl-N-{1-[1-(1H-pyrrole-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
2-(3-phenyl-1,2,4-oxadiazol-5-yl)-1,2,3,4-tetrahydroisoquinolin-4-ol
1-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}but-2-yn-1-one
(2R,4S)-1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-4-hydroxypiperidine-2-carboxylic acid