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(2S)-3-(4-hydroxyphenyl)-2-{[1-(propan-2-yl)piperidin-4-yl]formamido}propanoic acid
2-(4-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazin-1-yl)pyridine-3-carboxamide
4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}piperidine
N-[(5-{[(4-fluorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]cyclohexanecarboxamide
N-[(2-methyl-1H-1,3-benzodiazol-6-yl)methyl]-2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
2,4-dimethoxy-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}benzene-1-sulfonamide
3-[(3R,4R)-3-hydroxypiperidin-4-yl]-1-[3-(3-methoxyphenyl)phenyl]urea
(1R,3S)-3-(2-hydroxyethoxy)-7-[5-(hydroxymethyl)furan-2-carbonyl]-7-azaspiro[3.5]nonan-1-ol
2-({2-[1-(3-ethyl-1,2-oxazole-5-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
N-{[6-chloro-4-(cyclopentylamino)quinazolin-2-yl]methyl}-1,3-thiazole-5-carboxamide
N-{4-[2-(2H-1,3-benzodioxol-5-yloxy)propanamido]-2-methylphenyl}pentanamide
(1S,5R)-6-(1H-indol-5-ylmethyl)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-[(4aR,7aS)-4-(3-methoxypropyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
5-ethyl-N-{[4-(piperidine-1-carbonyl)phenyl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
(3aR,6aR)-2-[(2-ethyl-1,3-thiazol-4-yl)methyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-{[3-methoxy-4-(propan-2-yloxy)phenyl]methyl}-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide
1-{1-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-1-oxopropan-2-yl}pyrrolidin-2-one
[(2S)-1-{2-[benzyl(methyl)amino]-2,3-dihydro-1H-indene-2-carbonyl}pyrrolidin-2-yl]methanol
2-methyl-3-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]pyrazine
2-{2-[1-(2,5-difluorobenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
(4aR,8aS)-6-[3-(4-fluorophenyl)benzoyl]-1-[2-(4-methoxyphenyl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-2-[1-(3-methoxypropyl)-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]acetamide
N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
2-{[4-(ethylamino)pyrimidin-2-yl]amino}-N-(2-methylphenyl)acetamide
N,3-dimethyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]furan-2-carboxamide
5-[1-(2H-1,3-benzodioxol-5-yloxy)ethyl]-3-benzyl-1H-1,2,4-triazole
4-chlorophenyl (7R,9aR)-7-(2-methylpropyl)-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
methyl 2-[(3,5-dimethylphenyl)sulfamoyl]-6-[(2-hydroxyphenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-[4-(methylsulfanyl)benzoyl]-1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidine
(3aR,7aS)-2-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carbonyl}-2,3,3a,4,7,7a-hexahydro-1H-isoindole
1-{2-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]-2-oxoethyl}-5-(trifluoromethyl)-1,2-dihydropyridin-2-one
9-methoxy-4-[(2-methoxyphenyl)methyl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(1R,5S,6R)-N-[(3,4-dichlorophenyl)methyl]-3-azabicyclo[3.1.0]hexane-6-carboxamide
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-(5-oxo-2-phenylcyclopent-1-en-1-yl)acetamide
N-(1-methyl-1H-indazol-3-yl)-2-[3-(pyrimidin-5-yl)-1H-indazol-1-yl]acetamide
4-[(2-ethyl-1H-imidazol-1-yl)methyl]-5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazole
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}acetamide
(3aS,7aR)-2-(1H-imidazole-2-carbonyl)-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
9-[1-(4-chlorophenyl)cyclobutanecarbonyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
2-(3-phenylpyrrolidin-1-yl)-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]acetamide
2-[2-({methyl[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]amino}methyl)phenoxy]ethan-1-ol
2-chloro-N-{[1-(2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carbonyl)piperidin-3-yl]methyl}benzamide
5-{[4-(4-methylphenoxy)piperidin-1-yl]methyl}-N-(propan-2-yl)pyrimidin-2-amine
N,N-dimethyl-3-(5-methyl-2-oxo-5-phenylpiperidin-1-yl)propanamide
N-{4-[2-(3-methoxyphenyl)azetidine-1-carbonyl]phenyl}-2-methylfuran-3-carboxamide
N-[2-(6-hydroxypyrimidin-4-yl)ethyl]-1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
7-(cyclobutylmethyl)-2-(8-methoxy-4-methylquinolin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
N-(3-carbamoyl-4-methoxyphenyl)-2-(propan-2-yl)-2,5-dihydro-1H-pyrrole-1-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{1-[(5-ethylfuran-2-yl)methyl]piperidin-3-yl}piperazine
1-[(3R,4R)-3-hydroxy-4-methyl-3-(propan-2-yl)pyrrolidin-1-yl]-2-[methyl(pyridin-3-ylmethyl)amino]ethan-1-one