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(2-ethoxy-5-{[3-(hydroxymethyl)-3-(3-phenylpropyl)piperidin-1-yl]methyl}phenyl)methanol
4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-N-(2,3,5-trifluorophenyl)piperidine-1-carboxamide
[(2S,6S)-4-(4-chloro-3-fluorobenzoyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
2-[5-(1H-imidazol-4-yl)-4-phenyl-1H-imidazol-1-yl]acetic acid
{[(3S,4R)-1-(2-methoxy-4-methylbenzoyl)-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl}dimethylamine
(4aR,7aS)-1-acetyl-4-(5-methyl-1H-indazole-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-4-[(3-methylpyridin-2-yl)methyl]piperazine
3-methyl-1-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)-1H-1,2,4-triazole
N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-2-oxo-1-phenylpyrrolidine-3-carboxamide
methyl 4-methyl-2-{2-[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]acetamido}-1,3-thiazole-5-carboxylate
N-{2-methyl-[1,2,4]triazolo[1,5-a]pyridin-8-yl}-2-(1,3-thiazol-2-yl)piperidine-1-carboxamide
1-[2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]piperidin-4-amine
6-methyl-N-[1-(morpholine-4-carbonyl)piperidin-4-yl]-2-oxo-1,2-dihydropyridine-4-carboxamide
(2S,4S,5R)-2-ethyl-5-(4-methoxyphenyl)-1-methyl-4-[(oxan-4-yl)carbamoyl]pyrrolidine-2-carboxylic acid
1-(2-{[1-methyl-3-(trifluoromethyl)-1H-pyrazol-5-yl]formamido}ethyl)piperidine-3-carboxamide
5-[1-(5-methyl-1,3,4-oxadiazole-2-carbonyl)pyrrolidin-2-yl]-N-(1-methyl-1H-pyrazol-5-yl)thiophene-2-carboxamide
(3R,4R)-1-[2-(1H-imidazol-1-yl)ethyl]-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
1-methyl-5-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-3-phenyl-1H-pyrazole
N-[1-(1-{[(2-methylpropyl)carbamoyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]cyclopentanecarboxamide
(3S,4R)-1-(dimethyl-1,2-oxazole-4-carbonyl)-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
4-{1-[(3-chloro-1-benzothiophen-2-yl)methyl]azetidin-3-yl}morpholine
N-[2-(furan-2-yl)ethyl]-3-{2-[(4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
N-[1-(1-methyl-1H-pyrazol-4-yl)propyl]-5-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
1-[(3S,4R)-1-(5-ethylthiophene-3-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
2-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-5,8-dimethoxy-4-methylquinoline
3-[5-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
(1R,3S)-3-(2-hydroxyethoxy)-7-[4-methyl-6-(methylamino)pyrimidin-2-yl]-7-azaspiro[3.5]nonan-1-ol
N,1,3,6-tetramethyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H-pyrazolo[3,4-b]pyridine-4-carboxamide
2-{[5-(1-methoxyethyl)-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
N-[(3S,4R)-4-propyl-1-(quinoline-3-carbonyl)pyrrolidin-3-yl]methanesulfonamide
N,N-dimethyl-4-[4-(1,2-oxazolidine-2-carbonyl)phenoxy]piperidine-1-sulfonamide
1-[(3-methoxyphenyl)methyl]-4-[3-(2-oxo-1,2-dihydropyridin-1-yl)propanoyl]piperazin-2-one
7-[(2,3-difluorophenyl)methyl]-2-(pyridin-2-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
N-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}prop-2-ene-1-sulfonamide
ethyl 4-(1-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)piperazine-1-carboxylate
1-(4-aminopyrimidin-2-yl)-4-(hydroxymethyl)piperidin-4-ol
1-(benzenesulfonyl)-4-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}piperazine
2-{methyl[(5-{pyrazolo[1,5-a]pyridine-7-carbonyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methyl]amino}ethan-1-ol
5-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
N-(2-methoxyethyl)-4-methyl-3-{[methyl(2-methylpropyl)carbamoyl]methyl}-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
2-{2-oxo-8-[4-(1H-1,2,4-triazol-3-yl)benzoyl]-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}acetic acid
N-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]furan-2-carboxamide
1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-8-[5-(trifluoromethyl)pyridin-2-yl]-1,8-diazaspiro[4.5]decane
(2R,3S,6R)-3-(2,3-difluorophenyl)-5-(1,2-oxazole-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-{[2-fluoro-5-(trifluoromethyl)phenyl]methyl}-5-(piperidin-1-yl)-2,3-dihydropyridazin-3-one
1-[(2-ethyl-1,3-thiazol-4-yl)methyl]-3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
3-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-3-methyl-1-[4-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]urea
(2S,4R)-1-[(2-chloro-6-fluorophenyl)methyl]-N-(2-methyl-1,3-benzothiazol-5-yl)-4-(pyridin-2-ylsulfanyl)pyrrolidine-2-carboxamide
2-amino-3-ethyl-N-{[1-(morpholin-4-yl)cyclopentyl]methyl}-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide