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(4aR,7aS)-1-cyclobutanecarbonyl-4-(1-methyl-1H-pyrazole-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-[1-(3-methylbutyl)-1H-pyrazol-5-yl]-3-propoxypiperidine-1-carboxamide
2-(2,3-dihydro-1H-inden-5-yloxy)-N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-2-methylpropanamide
1-[2-(dimethylamino)-2-(2-fluorophenyl)acetamido]cyclopentane-1-carboxamide
4-[(3S,4S)-4-hydroxy-1-[(5-phenylthiophen-2-yl)methyl]pyrrolidin-3-yl]piperazin-2-one
3-(1H-imidazol-4-yl)-2-{[3-(5-methylfuran-2-yl)-1H-pyrazol-5-yl]formamido}propanoic acid
2-[3-(1H-1,3-benzodiazol-5-yl)-1,2,4-oxadiazol-5-yl]-N,N-dimethyl-2,3-dihydro-1H-inden-2-amine
2-{1-[1-(2,5-difluorobenzoyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-2-ol
4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-1-[3-(3-methylphenyl)-1H-pyrazole-4-carbonyl]piperidine
4-(4-methanesulfonylphenyl)-2-methyl-5-propylpyrimidine
1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methoxyethan-1-one
4-[1-(2,3-dihydro-1H-inden-2-yl)-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]pyridine
(2S)-2-[4-(4-hydroxyquinolin-2-yl)-1H-1,2,3-triazol-1-yl]-4-methylpentanamide
(cyclobutylmethyl)({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)(oxolan-2-ylmethyl)amine
(4aS,8aR)-6-[3-(1,2-oxazolidin-2-yl)propanoyl]-1-propyl-decahydro-1,6-naphthyridin-2-one
2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decane
(2E)-1-{4-[2-(2H-1,3-benzodioxol-5-yl)-5-fluoro-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}-3-(thiophen-2-yl)prop-2-en-1-one
N-[4-(2,1,3-benzothiadiazol-4-yl)-7-methoxy-2-oxo-1,2,3,4-tetrahydroquinolin-6-yl]butanamide
4-[(2-fluorophenyl)methyl]-1-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidine
3-(2,5-dimethoxyphenyl)-1-[5-(methoxymethyl)thiophene-2-carbonyl]pyrrolidine
8-[(5-methoxy-1,3,4-thiadiazol-2-yl)methyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
4-[(3-fluorophenyl)methyl]-1-(1H-indol-2-ylmethyl)-1,4-diazepan-5-one
(2R)-1-({3-[(2-methoxy-6-methylphenyl)carbamoyl]phenyl}methyl)pyrrolidine-2-carboxamide
ethyl 1-[3-({[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)-6,7-dimethoxyquinolin-2-yl]piperidine-3-carboxylate
6-(1,2-oxazinan-2-yl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
2-(4-ethylpiperazin-1-yl)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}acetamide
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-[(propan-2-yl)amino]pyrimidine-5-carboxamide
4-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine-1-sulfonamide
1-ethyl-3-(2-methylpropyl)-N-{[3-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}-1H-pyrazole-5-carboxamide
N-[5-(pentan-2-yl)-1,3,4-thiadiazol-2-yl]-1H-1,2,4-triazole-5-carboxamide
4-(2,5-dimethoxyphenyl)-3-[(trimethyl-1H-pyrazol-1-yl)methyl]-4H-1,2,4-triazole
methyl 2-({1-methyl-1H-pyrazolo[1,5-a]imidazol-7-yl}formamido)-2-(3-methylphenyl)acetate
1-ethyl-3-[4-(1-hydroxy-2-phenylethyl)piperidine-1-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
2-(2-{2-azaspiro[4.4]nonan-2-ylmethyl}phenyl)-5-methyl-6-(trifluoromethyl)-3,4-dihydropyrimidin-4-one
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[3-(1H-imidazol-1-yl)butyl]benzamide
(3R,4S)-1-(4-methyl-2-phenylpyrimidine-5-carbonyl)-4-phenylpyrrolidin-3-amine
3-{4-[3-(furan-2-yl)phenyl]-1H-1,2,3-triazol-1-yl}propane-1,2-diol
(2S,4R)-4-{4-[({[(2R)-3-methylbutan-2-yl]carbamoyl}amino)methyl]-1H-1,2,3-triazol-1-yl}-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-(4-fluoro-2-methylphenyl)-4-hydroxy-4-(pyrrolidin-1-ylmethyl)piperidine-1-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}thiophene-2-carboxamide
6-[(3-fluorophenyl)methoxy]-1-(2-phenylethyl)-4-(pyridine-2-carbonyl)-1,4-diazepan-2-one
(3S,4R)-4-methyl-3-(2-methylpropyl)-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidin-4-ol
N3-cyclooctyl-N5-[2-(2-fluorophenyl)ethyl]-4-oxo-1-(oxolan-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
4-[(2-fluoro-4-methoxyphenyl)methyl]-3-[2-(1,2-oxazolidin-2-yl)-2-oxoethyl]piperazin-2-one
1-{1-[(2-aminopyridin-3-yl)methyl]piperidin-3-yl}-2-phenylethan-1-one
4-[(5-ethylpyridin-2-yl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
3-{[(2H-1,3-benzodioxol-5-ylmethyl)amino]methyl}-1-(2-cyclohexylethyl)-3-hydroxypiperidin-2-one
3-[4-(4-fluorophenyl)-4-hydroxypiperidine-1-carbonyl]-N,N-dimethylpiperidine-1-carboxamide