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4-(1-{[3-(morpholin-4-yl)phenyl]methyl}piperidin-3-yl)benzoic acid
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-6-methylpyridine-3-carboxamide
6-[(3aS,6aR)-3-[3-(morpholin-4-yl)propyl]-2-oxo-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-5-yl]pyridine-3-carbonitrile
1-methyl-N-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl}azepane-2-carboxamide
N-[2-({4-[(2-chlorophenyl)methyl]-4-(hydroxymethyl)piperidin-1-yl}methyl)quinolin-5-yl]acetamide
4-(cyclopropylmethyl)-1-(3-phenyl-1,2-oxazole-5-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
6-ethoxy-3-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
dimethyl({1-[4-(1-propyl-1H-1,2,4-triazol-5-yl)phenyl]ethyl})amine
1-(cyclohex-1-ene-1-carbonyl)-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-3-carboxamide
N-[2-(3-chlorophenoxy)ethyl]-N-methyl-4-(piperidin-3-yl)benzamide
3-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butan-1-amine
1-[(3R,4S)-4-(dimethylamino)-3-(3-hydroxypropyl)piperidin-1-yl]-2-(3-fluoro-4-methylphenyl)ethan-1-one
3-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-4,5,6,7-tetrahydro-1H-indazole
5-(5,6-dimethyl-1H-1,3-benzodiazol-1-yl)pyridin-2-ol
4-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-(3-propylpyrrolidin-1-yl)pyrimidine
2-oxo-N-[3-(pyridin-3-yl)propyl]-2-(pyrrolidin-1-yl)acetamide
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-1H-pyrrole-3-carboxamide
N,N,2-trimethyl-7-(morpholine-4-sulfonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-[1-(3-methoxyphenyl)ethyl]-N-methyl-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanamide
(4aS,8aR)-6-(3-fluoropyridine-4-carbonyl)-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
3-{2-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
[(3-chloro-4-ethoxyphenyl)methyl](1H-imidazol-2-ylmethyl)methylamine
4-({4-methyl-5-[1-(1,3-thiazol-2-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
2-[3-cyclopropyl-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-1,2,4-triazol-5-yl]phenol
N-{2-[7-(cyclohexylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-2-oxoethyl}acetamide
1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-4-(pyridin-3-yl)piperidin-4-ol
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-(4-methoxyphenoxymethyl)piperidine
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-6-(2-methoxyphenyl)-N-methylimidazo[2,1-b][1,3]thiazole-3-carboxamide
5-phenyl-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}-1,2-oxazole-3-carboxamide
1-[(1S,5R)-6-[(2,5-dimethylthiophen-3-yl)sulfonyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
(3aS,6aR)-3-[2-(4-fluorophenyl)ethyl]-5-(isoquinolin-5-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
6-{1-[2-(1H-imidazol-2-yl)benzoyl]piperidin-4-yl}-2-methylpyrimidin-4-ol
[(2S)-1-(4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)pyrrolidin-2-yl]methanol
1-(5-ethyl-2,6-dimethylpyrimidin-4-yl)-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-4-ol
4-(1-methyl-1H-1,2,4-triazol-5-yl)-2-[4-(piperidine-1-carbonyl)piperidin-1-yl]pyrimidine
3-({2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}methyl)phenol
7-(2-benzyl-1,3-thiazole-4-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
(3S,4R)-4-methyl-1-(4-methyl-1H-imidazole-5-carbonyl)-3-(2-methylpropyl)piperidin-4-ol
3-[2-(2-methyl-3-oxo-4-phenylpiperazin-1-yl)-2-oxoethyl]-1,3-diazinane-2,4-dione
N-methyl-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[(4-methyl-1H-imidazol-2-yl)methyl]acetamide
8-[(5-methylthiophen-2-yl)methyl]-1-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(1,3-benzothiazol-2-ylmethyl)(1H-imidazol-4-ylmethyl)methylamine
4-({methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)-1H-pyrazole-3-carboxylic acid
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
2-methyl-8-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzoyl]-2,8-diazaspiro[4.5]decan-3-one
N-[2-oxo-2-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)ethyl]methanesulfonamide
ethyl 4-[4-(4-{[2-(1H-pyrazol-1-yl)ethyl]amino}piperidin-1-yl)benzoyl]piperazine-1-carboxylate
5-methanesulfonyl-N-methyl-N-[(2-methylphenyl)methyl]-4-(piperidin-3-yl)pyrimidin-2-amine
2-[(4-methyl-1,3-thiazol-2-yl)methyl]-4-{4-[1-(2-phenylethyl)piperidin-4-yl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
5-(dimethylamino)-2-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2,3-dihydropyridazin-3-one