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8-chloro-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}quinoline-2-carboxamide
4-(4-methyl-1,3-thiazole-5-carbonyl)-1-(4-methylphenyl)piperazin-2-one
(3aS,6aS)-2-(oxan-4-yl)-5-(pyridin-2-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(1-benzyl-1H-imidazol-2-yl)-1-[(2-methyl-1,3-oxazol-4-yl)methyl]piperidine
2-[3-({3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}methyl)phenoxy]ethan-1-ol
(3aR,6aR)-2-methyl-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
N-cyclopentyl-1-(furan-2-ylmethyl)-N-(thiophen-3-ylmethyl)piperidine-3-carboxamide
3-ethyl-1-(2-phenylethyl)-8-{[2-(trifluoromethyl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-[(2,3-dihydro-1H-inden-2-yl)amino]-1-ethyl-N-(furan-2-ylmethyl)-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-4-[(2-methylpyrrolidin-1-yl)methyl]-1,3-oxazole
2,6-dimethoxy-N-[2-(4-methylmorpholin-2-yl)ethyl]pyrimidine-4-carboxamide
4-[3-({1,9-dioxaspiro[5.5]undecan-4-yl}amino)propyl]-1,3-thiazol-2-amine
N-ethyl-7,8-dimethyl-N-(pyridin-3-ylmethyl)-2-(pyrimidin-5-yl)quinoline-4-carboxamide
4-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-1,4-oxazepan-6-ol
{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amine
1-{1-[(5-methylthiophen-2-yl)methyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
2,5-dimethyl-3-{4-[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperazin-1-yl}pyrazine
2-{4-[(2,5-difluorophenyl)methyl]-1-[(4-methoxy-3-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
2-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridin-3-ol
methyl[(2-methyl-2,3-dihydro-1-benzofuran-5-yl)methyl]{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}amine
N-{[1-(4-methoxyphenyl)cyclopentyl]methyl}-2-oxo-1-oxaspiro[4.4]nonane-4-carboxamide
(2E)-3-(3,4-dimethoxyphenyl)-N-{[8-(3-phenylpropyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}prop-2-enamide
1-benzyl-3-[2-(1,4-diazepan-1-yl)-2-oxoethyl]-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
3-[(3R,4S)-1-(5-methyl-1,3-benzoxazol-2-yl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
1-[2-(pyridin-2-yl)ethyl]-5-(thiomorpholine-4-carbonyl)piperidin-2-one
N-cyclobutyl-2-(4-methoxyphenoxymethyl)-1,3-oxazole-4-carboxamide
N-methyl-4-[(3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)methyl]-1,3-thiazol-2-amine
(1R,3S)-3-(2-aminoethoxy)-7-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-7-azaspiro[3.5]nonan-1-ol
N-(1,3-benzothiazol-6-yl)-4-[(3S,4R)-4-hydroxyoxolan-3-yl]-1,4-diazepane-1-carboxamide
N-benzyl-2-[2-(1H-imidazol-4-yl)ethyl]-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
1-[1-(6-methylpyridin-3-yl)ethyl]-3-(3,4,5-trimethoxyphenyl)urea
N-[2-(pyrrolidine-3-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]pyridine-2-carboxamide
N-{[1-(1H-imidazol-4-ylmethyl)piperidin-4-yl]methyl}-1-phenylcyclopropane-1-carboxamide
2-({[4-(methylsulfanyl)phenyl]methyl}({[1-(propan-2-yl)piperidin-4-yl]methyl})amino)ethan-1-ol
7-(3-phenylpropyl)-2-(pyridine-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-(3-fluoro-4-methoxyphenyl)-3-(pyrrolidine-1-carbonyl)pyridine
1-(2,5-dimethylbenzoyl)-3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
N-{2-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]-2-oxoethyl}methanesulfonamide
1'-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-4-one
5-{[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}-N,N-dimethylpyrimidin-2-amine
N-[(3S,4R)-4-(propan-2-yl)-1-[2-(pyridin-2-yl)ethyl]pyrrolidin-3-yl]methanesulfonamide
(1S,5R)-6-(2H-1,3-benzodioxole-5-carbonyl)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
5-fluoro-2-methoxy-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]benzamide
2-(ethylamino)-N-[1-(6-methoxynaphthalen-2-yl)ethyl]pyrimidine-5-carboxamide
6-({[2-(1H-indol-3-yl)ethyl]amino}methyl)-1,4-oxazepan-6-ol
(1S,5R)-3-benzyl-6-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-cyclopropyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
3-(2H-1,3-benzodioxol-5-yl)-N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-phenylpropanamide
N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-4-(1H-1,2,4-triazol-1-yl)butanamide
4-[hydroxy(pyridin-2-yl)methyl]-N-{2-[(2-methylprop-2-en-1-yl)oxy]phenyl}piperidine-1-carboxamide