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ethyl 4-[(4-chlorophenyl)methyl]-1-propylpiperidine-4-carboxylate
3-{1-[5-(methylcarbamoyl)furan-2-yl]-1H-pyrazol-4-yl}benzoic acid
1-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-N-(pyridin-2-ylmethyl)piperazine-2-carboxamide
{1-[(2,3-dimethoxyphenyl)methyl]-4-(3-phenylpropyl)piperidin-4-yl}methanol
3-(azocan-1-yl)-N-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]propanamide
N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
3-(3-cyanopiperidine-1-carbonyl)-N-(1,2-oxazol-3-ylmethyl)benzene-1-sulfonamide
2,4-dimethyl-6-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}pyrimidine
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(4-methylpyrimidin-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-methyl-6-[4-(pyridin-3-ylmethyl)-1,4-diazepane-1-carbonyl]-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
3-(cyclopropylmethyl)-5-[2-fluoro-4-(pyrrolidin-1-ylmethyl)phenoxymethyl]-1,2,4-oxadiazole
4-[(1R,5S,8S)-8-methoxy-3-azabicyclo[3.2.1]octan-3-yl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaene
N-(pyridin-2-ylmethyl)-1-[1-(thiophen-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
3-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-1-{2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl}urea
2-methyl-6-{[1-methyl-5-(trifluoromethyl)-1H-1,3-benzodiazol-2-yl]methyl}-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
5-{[benzyl(methyl)amino]methyl}-N-(furan-3-ylmethyl)-N-methyl-1,2-oxazole-3-carboxamide
9-[(3-methylquinoxalin-2-yl)methyl]-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-(5-methoxy-1-methyl-1H-indole-2-carbonyl)-6-(methylsulfanyl)-1,2,3,4-tetrahydroisoquinoline
1-(4-methoxyphenyl)-6,6-dimethyl-4-{spiro[2.4]heptane-1-carbonyl}piperazin-2-one
4-(3-benzyl-1H-pyrazol-5-yl)-1-(1-ethyl-1H-pyrazole-4-carbonyl)piperidine
N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
5-chloro-2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-methyl-N-(oxan-2-ylmethyl)benzamide
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(3-methylpyridin-2-yl)methyl]acetamide
(5S,9aS,9bS)-5-(2,1,3-benzothiadiazol-5-yl)-2-[(2-methylphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]piperazine-1-sulfonamide
4-[3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)propanoyl]piperazin-2-one
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-(1-ethyl-5-methyl-1H-pyrazol-4-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N'-ethyl-N-(2-methylphenyl)-N'-(pyridin-2-ylmethyl)propanediamide
3-[(3R,4S)-1-[(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
(3S,4R)-1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
2-[2-(1H-imidazol-4-yl)ethyl]-8-(pyridine-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
2-[(3,4-difluorophenyl)methyl]-8-(3-fluoropropyl)-2,8-diazaspiro[4.5]decan-3-one
2-{[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
1-cyclopentyl-N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-6-oxopiperidine-3-carboxamide
4-(2,2-dimethylpropyl)-3-{2-oxo-2-[4-(2-phenoxyethyl)piperazin-1-yl]ethyl}piperazin-2-one
2-(2-methoxyethyl)-8-({4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-2,8-diazaspiro[5.5]undecan-3-one
8-methoxy-N-[3-(methylsulfanyl)propyl]-3,4-dihydro-2H-1-benzopyran-3-amine
3-(1,4-dimethyl-3-phenyl-1H-pyrazol-5-yl)-1-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]urea
2-(dimethyl-1,2-oxazol-4-yl)-N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}acetamide
N-(2-methoxyethyl)-3-phenyl-N-(pyridin-4-ylmethyl)-1H-pyrazole-4-carboxamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-2-hydroxy-4-(methylsulfanyl)butanamide
1-[3-(hydroxymethyl)-3-(3-methoxypropyl)piperidin-1-yl]-2-methoxy-2-methylpropan-1-one
methyl 2-chloro-5-{[3-hydroxy-3-(hydroxymethyl)pyrrolidine-1-carbonyl]amino}benzoate
3-{2-[(2-methylprop-2-en-1-yl)oxy]phenyl}-1-(oxan-4-yl)urea
(2S,4R)-4-amino-1-{6-chloro-2-methylimidazo[1,2-a]pyridine-3-carbonyl}-N-methylpyrrolidine-2-carboxamide
1,6-dimethyl-2-oxo-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1,2-dihydropyridine-3-carboxamide
{1-[2-(morpholin-4-yl)ethyl]-3-(prop-2-en-1-yl)piperidin-3-yl}methanol
N-(butan-2-yl)-5-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
5-methyl-3-[4-(thiophen-2-ylmethyl)-1,4-diazepane-1-carbonyl]-4,5,6,7-tetrahydro-2H-indazole
N-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]-4,5,6,7-tetrahydro-1,2-benzoxazole-3-carboxamide