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[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]({[4-methoxy-3-(methoxymethyl)phenyl]methyl})methylamine
2-[2-(1H-imidazol-4-yl)ethyl]-8-(2-methylpyridin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
[(4aS,8aR)-1-(1,3-benzothiazole-5-carbonyl)-6-propyl-decahydro-1,6-naphthyridin-4a-yl]methanol
(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)({[2-(propylsulfanyl)pyrimidin-5-yl]methyl})amine
2-(1-benzylpyrrolidin-3-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-(5-{[({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)amino]methyl}-1,2,4-oxadiazol-3-yl)benzoic acid
5-(2H-1,3-benzodioxol-5-yl)-1-butyl-3-(ethoxymethyl)-1H-1,2,4-triazole
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
1-{2-[2-(3,4-dimethoxyphenyl)acetamido]ethyl}-N-[1-(thiophen-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
5-[3-(morpholin-4-yl)azetidin-1-yl]-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
methyl 1-[(3-methoxyphenyl)methoxy]-2-oxo-8-(thiophen-3-ylmethyl)-1,8-diazaspiro[4.5]decane-4-carboxylate
4-[1-methyl-4-(3-propoxypiperidin-1-yl)-1H-pyrazolo[3,4-d]pyrimidin-6-yl]pyridine
5-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-methylpyrimidin-4-amine
(3S,4S)-4-cyclopropyl-1-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)pyrrolidine-3-carboxylic acid
[1-(2-methyl-1-benzofuran-5-carbonyl)-3-(2-phenoxyethyl)piperidin-3-yl]methanol
methyl 2-(benzylsulfamoyl)-6-(3-phenylpropanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4-(morpholin-4-yl)benzamide
N-[(2-ethoxyphenyl)methyl]-N-(prop-2-en-1-yl)-3-(1H-pyrrol-1-yl)propanamide
[(3R,4R)-4-[(4-methylpiperazin-1-yl)methyl]-1-(oxane-4-carbonyl)pyrrolidin-3-yl]methanol
5-chloro-3-ethyl-4-{[2-(3-methoxyphenyl)azetidin-1-yl]methyl}-1-methyl-1H-pyrazole
N-[3-(4-{[3-(1H-1,3-benzodiazol-1-yl)propanamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]-2-methylfuran-3-carboxamide
2-{2-[1-(2-propyl-1,3-thiazole-4-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]({[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl})amine
1-methyl-N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]-3-propyl-1H-pyrazole-5-carboxamide
8-[6-(2-methyl-1H-imidazol-1-yl)pyridazin-3-yl]quinoline
3-{2-[4-(furan-3-carbonyl)-1,4-diazepan-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
N-{2-[(2S)-pyrrolidin-2-yl]ethyl}-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
4-(2,2-difluoro-2H-1,3-benzodioxol-5-yl)-N-(2-methoxyethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-4-oxo-1,4-dihydroquinoline-2-carboxamide
1-(2-fluoropyridin-3-yl)-3-[1-(4-methyl-1H-imidazol-2-yl)propyl]urea
N-ethyl-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
2-[4-(4-cyclopentylpiperazine-1-carbonyl)-5-methyl-1H-pyrazol-1-yl]-4-(5-methylfuran-2-yl)pyrimidine
1-(2-ethoxyethyl)-3-(3-{thieno[2,3-d]pyrimidin-4-yl}phenyl)-1H-pyrazole
2-cyclopropanecarbonyl-8-(1H-pyrazole-3-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
5-({2-[2-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-1H-imidazol-1-yl]ethyl}sulfanyl)-1H-1,2,3-triazole
2-(2-{[(3S,4R)-4-amino-3-methoxypiperidin-1-yl]methyl}-4-(pyrimidin-5-yl)phenoxy)acetic acid
2-(dimethylamino)-2-(3-fluorophenyl)-N-methyl-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}acetamide
2-(cyclopentylmethyl)-6-methyl-5-[5-(pyrazin-2-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
9-(6-methyl-2-propylpyrimidin-4-yl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-({4-methyl-5-[1-(pyrazin-2-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-2-cyclohexyl-1,3-benzoxazole-6-carboxamide
1-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]-3-{imidazo[1,2-a]pyridin-2-yl}propan-1-one
N-{2-[4-(4-fluorophenyl)-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl]ethyl}-2-(1H-pyrazol-1-yl)benzamide
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]propanamide
N-[2-(diethylamino)ethyl]-N-ethyl-1-[2-(2-methoxyethyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]piperidine-4-carboxamide
N-ethyl-2-[(prop-2-en-1-yl)amino]-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]benzamide
methyl 4-(4-{[(2-methoxyethyl)(propan-2-yl)amino]methyl}-5-methyl-1,3-oxazol-2-yl)benzoate
2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)-N-[2-(propan-2-yloxy)ethyl]acetamide
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-amine
2-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-6-methoxyphenol