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1-({[(2-methylphenyl)methyl](prop-2-en-1-yl)carbamoyl}methyl)piperidine-4-carboxamide
2-[ethyl({[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl})amino]ethan-1-ol
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-(pyridin-4-yl)acetamide
2-{5-[1-(2-hydroxyethyl)-1H-1,3-benzodiazol-5-yl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl}acetic acid
2-{[(2,3-dihydro-1H-inden-2-yl)amino]methyl}-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
3-[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]propanamide
methyl 4-({6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carbonyl}amino)benzoate
1-(1-benzothiophen-2-ylmethyl)-3-(pyrrolidin-1-yl)piperidine
N-[(4-hydroxyazepan-4-yl)methyl]-3-(3-methoxyphenyl)benzamide
7-(5-chloropyridin-2-yl)-4-(thiophen-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-{[(3S)-3-(dimethylamino)pyrrolidin-1-yl]methyl}-7-methoxy-1,2-dihydroquinolin-2-one
2-cyclopropyl-4-[3-(4-phenylazepane-1-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
N4-[(4-methanesulfonylmorpholin-2-yl)methyl]-N2,N2,5,6-tetramethylpyrimidine-2,4-diamine
N-[(3R,4S)-1-(2-carbamoylethyl)-4-cyclopropylpyrrolidin-3-yl]-4,5-dimethylthiophene-2-carboxamide
3-ethyl-N-[1-(methoxymethyl)cyclopentyl]-1H-pyrazole-5-carboxamide
1-(4-{[(2-hydroxyethyl)(methyl)amino]methyl}-2-methoxyphenoxy)-3-(thiomorpholin-4-yl)propan-2-ol
N-methyl-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]-N-[2-(1H-pyrazol-4-yl)ethyl]piperidine-3-carboxamide
2-[2-(dimethylamino)ethyl]-9-(2-hydroxy-3-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
8-[4-(3,5-dimethyl-1H-pyrazol-1-yl)butanoyl]-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one
(3aR,6aR)-2-methyl-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1-(4-methylphenyl)cyclopropane-1-carboxamide
2-methyl-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)oxolane-2-carboxamide
1-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-3-(2-methylphenoxy)propan-1-one
3-phenyl-N-[3-(pyridin-2-yl)propyl]-1H-pyrazole-4-carboxamide
(1R,5R)-N,N-dimethyl-6-{2-[methyl(phenyl)amino]acetyl}-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
4-benzyl-3-[1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{[3-(2-chlorophenyl)-1,2-oxazol-5-yl]methyl}-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-1-(2-methoxyphenyl)-1H-pyrazole-4-carboxamide
(2S,4R)-4-amino-1-(2-{[(2-chlorophenyl)methyl]sulfanyl}acetyl)-N-methylpyrrolidine-2-carboxamide
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-hydroxyacetamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]acetamide
1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
N-(2-cyclopentylethyl)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-[3-(5-methylfuran-2-yl)butyl]piperazine-1-sulfonamide
4-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]pyrimidin-2-amine
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carboxamide
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-2-(morpholin-4-yl)-2-oxoacetamide
N-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-4-sulfamoylbenzamide
(3S,4R)-4-(3-fluorophenyl)-1-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}pyrrolidine-3-carboxylic acid
1-[(4-chlorophenyl)methyl]-N-[1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
(3S,4R)-1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-4-phenylpyrrolidine-3-carboxylic acid
1-(1-cyclobutylpiperidin-4-yl)-N-cyclopropylpiperidine-3-carboxamide
N-ethyl-N-(2-hydroxyethyl)-5-[3-(trifluoromethyl)phenoxymethyl]-1H-pyrazole-3-carboxamide
4-(2-methoxyphenoxy)-1-{[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl}piperidine
dimethyl[(2-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl}phenyl)methyl]amine
2-[2-(4-methyl-2-phenylpiperazin-1-yl)-2-oxoethyl]-1,2-dihydrophthalazin-1-one
1-[2-({methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
(3R,4R)-1-(2-cyclopropyl-4-methylpyrimidine-5-carbonyl)-4-methyl-3-(propan-2-yl)pyrrolidin-3-ol
N-[(4-hydroxyazepan-4-yl)methyl]-1-methyl-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
N-{[1-(5-acetyl-2,4-dimethyl-1H-pyrrole-3-carbonyl)piperidin-3-yl]methyl}thiophene-2-sulfonamide